ATE178897T1 - Hypolipidämische benzothiazepin verbindungen - Google Patents

Hypolipidämische benzothiazepin verbindungen

Info

Publication number
ATE178897T1
ATE178897T1 AT93904212T AT93904212T ATE178897T1 AT E178897 T1 ATE178897 T1 AT E178897T1 AT 93904212 T AT93904212 T AT 93904212T AT 93904212 T AT93904212 T AT 93904212T AT E178897 T1 ATE178897 T1 AT E178897T1
Authority
AT
Austria
Prior art keywords
integer
pct
alkyl
phenylalkoxy
alkoxy
Prior art date
Application number
AT93904212T
Other languages
German (de)
English (en)
Inventor
Lawrence Edward Brieaddy
Original Assignee
Wellcome Found
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wellcome Found filed Critical Wellcome Found
Application granted granted Critical
Publication of ATE178897T1 publication Critical patent/ATE178897T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D281/00—Heterocyclic compounds containing rings of more than six members having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D281/02—Seven-membered rings
    • C07D281/04—Seven-membered rings having the hetero atoms in positions 1 and 4
    • C07D281/08—Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D281/10—Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Vascular Medicine (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Urology & Nephrology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Saccharide Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Steroid Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
AT93904212T 1992-02-17 1993-02-16 Hypolipidämische benzothiazepin verbindungen ATE178897T1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB929203347A GB9203347D0 (en) 1992-02-17 1992-02-17 Hypolipidaemic compounds

Publications (1)

Publication Number Publication Date
ATE178897T1 true ATE178897T1 (de) 1999-04-15

Family

ID=10710542

Family Applications (1)

Application Number Title Priority Date Filing Date
AT93904212T ATE178897T1 (de) 1992-02-17 1993-02-16 Hypolipidämische benzothiazepin verbindungen

Country Status (21)

Country Link
US (2) US5663165A (en:Method)
EP (1) EP0626952B1 (en:Method)
JP (1) JP2904926B2 (en:Method)
KR (1) KR100265529B1 (en:Method)
AT (1) ATE178897T1 (en:Method)
AU (1) AU675419B2 (en:Method)
CA (1) CA2117485A1 (en:Method)
DE (1) DE69324479T2 (en:Method)
DK (1) DK0626952T3 (en:Method)
ES (1) ES2131106T3 (en:Method)
FI (1) FI943775A7 (en:Method)
GB (1) GB9203347D0 (en:Method)
GR (1) GR3030491T3 (en:Method)
HU (1) HUT71487A (en:Method)
IL (1) IL104740A (en:Method)
MX (1) MX9300821A (en:Method)
MY (1) MY129970A (en:Method)
NZ (1) NZ249189A (en:Method)
TW (1) TW274547B (en:Method)
WO (1) WO1993016055A1 (en:Method)
ZA (1) ZA931073B (en:Method)

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WO2025146507A1 (en) 2024-01-05 2025-07-10 Albireo Ab Benzothia(di)azepine compounds and their use as bile acid modulators
WO2025146508A1 (en) 2024-01-05 2025-07-10 Albireo Ab Benzothia(di)azepine compounds and their use as bile acid modulators

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US3362962A (en) * 1964-01-24 1968-01-09 Hoffmann La Roche Certain benzothiazepine derivatives
US5276025A (en) * 1992-09-09 1994-01-04 Merck & Co., Inc. Heterobicyclic sulfonamides

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FI943775A0 (fi) 1994-08-16
JPH07503724A (ja) 1995-04-20
US5663165A (en) 1997-09-02
MY129970A (en) 2007-05-31
DK0626952T3 (da) 1999-10-25
EP0626952A1 (en) 1994-12-07
TW274547B (en:Method) 1996-04-21
AU3508293A (en) 1993-09-03
CA2117485A1 (en) 1993-08-19
AU675419B2 (en) 1997-02-06
GR3030491T3 (en) 1999-10-29
KR100265529B1 (ko) 2000-11-01
KR950700265A (ko) 1995-01-16
NZ249189A (en) 1996-02-27
EP0626952B1 (en) 1999-04-14
JP2904926B2 (ja) 1999-06-14
US5859240A (en) 1999-01-12
ZA931073B (en) 1994-08-16
GB9203347D0 (en) 1992-04-01
DE69324479T2 (de) 1999-09-16
HUT71487A (en) 1995-11-28
FI943775L (fi) 1994-08-16
HU9402365D0 (en) 1994-10-28
IL104740A (en) 1996-09-12
HK1004217A1 (en) 1998-11-20
MX9300821A (es) 1993-09-01
DE69324479D1 (de) 1999-05-20
WO1993016055A1 (en) 1993-08-19
IL104740A0 (en) 1993-06-10
ES2131106T3 (es) 1999-07-16
FI943775A7 (fi) 1994-08-16

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