MXPA01006472A - Combinaciones de inhibidores de transporte de acido biliar ileal y derivados de acido fibrico para indicaciones cardiovasculares. - Google Patents

Combinaciones de inhibidores de transporte de acido biliar ileal y derivados de acido fibrico para indicaciones cardiovasculares.

Info

Publication number
MXPA01006472A
MXPA01006472A MXPA01006472A MXPA01006472A MXPA01006472A MX PA01006472 A MXPA01006472 A MX PA01006472A MX PA01006472 A MXPA01006472 A MX PA01006472A MX PA01006472 A MXPA01006472 A MX PA01006472A MX PA01006472 A MXPA01006472 A MX PA01006472A
Authority
MX
Mexico
Prior art keywords
combinations
ileal bile
transport inhibitors
bile acid
fibric
Prior art date
Application number
MXPA01006472A
Other languages
English (en)
Inventor
Bradley T Keller
Original Assignee
Searle Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=26811676&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MXPA01006472(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Searle Llc filed Critical Searle Llc
Publication of MXPA01006472A publication Critical patent/MXPA01006472A/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19—Carboxylic acids, e.g. valproic acid
    • A61K31/192—Carboxylic acids, e.g. valproic acid having aromatic groups, e.g. sulindac, 2-aryl-propionic acids, ethacrynic acid 
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/21—Esters, e.g. nitroglycerine, selenocyanates
    • A61K31/215—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
    • A61K31/216—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acids having aromatic rings, e.g. benactizyne, clofibrate
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A61K31/554—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having at least one nitrogen and one sulfur as ring hetero atoms, e.g. clothiapine, diltiazem
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/02—Non-specific cardiovascular stimulants, e.g. drugs for syncope, antihypotensives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Abstract

La presente invencion proporciona combinaciones de compuestos terapeuticos cardiovasculares para la profilaxis o el tratamiento de enfermedades cardiovasculares incluyendo hipercolesterolemia, aterosclerosis, o hiperlipidemia. Las combinaciones descritas incluyen un inhibidor de transporte de acido biliar ileal combinado con un derivado de acido fibrico.
MXPA01006472A 1998-12-23 1999-12-17 Combinaciones de inhibidores de transporte de acido biliar ileal y derivados de acido fibrico para indicaciones cardiovasculares. MXPA01006472A (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US11395598P 1998-12-23 1998-12-23
US14260399P 1999-07-07 1999-07-07
PCT/US1999/027948 WO2000038727A1 (en) 1998-12-23 1999-12-17 Combinations of ileal bile acid transport inhibitors and fibric acid derivatives for cardiovascular indications

Publications (1)

Publication Number Publication Date
MXPA01006472A true MXPA01006472A (es) 2004-03-10

Family

ID=26811676

Family Applications (1)

Application Number Title Priority Date Filing Date
MXPA01006472A MXPA01006472A (es) 1998-12-23 1999-12-17 Combinaciones de inhibidores de transporte de acido biliar ileal y derivados de acido fibrico para indicaciones cardiovasculares.

Country Status (24)

Country Link
US (2) US6638969B1 (es)
EP (2) EP1336413A1 (es)
JP (1) JP2002533413A (es)
KR (1) KR20010102964A (es)
CN (1) CN1342090A (es)
AR (1) AR022023A1 (es)
AT (1) ATE240120T1 (es)
AU (1) AU776658B2 (es)
BR (1) BR9916565A (es)
CA (1) CA2356607A1 (es)
CZ (1) CZ20012342A3 (es)
DE (1) DE69907960T2 (es)
DK (1) DK1140189T3 (es)
EA (1) EA200100707A1 (es)
ES (1) ES2200588T3 (es)
HK (2) HK1040926B (es)
HU (1) HUP0104793A2 (es)
IL (1) IL143947A0 (es)
MX (1) MXPA01006472A (es)
NO (1) NO20013162L (es)
NZ (1) NZ512537A (es)
PL (1) PL348580A1 (es)
PT (1) PT1140189E (es)
WO (1) WO2000038727A1 (es)

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