DE69231445D1 - Triazole enthaltende antifungizide mittel - Google Patents

Triazole enthaltende antifungizide mittel

Info

Publication number
DE69231445D1
DE69231445D1 DE69231445T DE69231445T DE69231445D1 DE 69231445 D1 DE69231445 D1 DE 69231445D1 DE 69231445 T DE69231445 T DE 69231445T DE 69231445 T DE69231445 T DE 69231445T DE 69231445 D1 DE69231445 D1 DE 69231445D1
Authority
DE
Germany
Prior art keywords
pct
image
date apr
sec
alkyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
DE69231445T
Other languages
English (en)
Other versions
DE69231445T2 (de
Inventor
Simon Bell
Kenneth Richardson
John Whittle
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Ltd
Pfizer Inc
Original Assignee
Pfizer Ltd
Pfizer Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Ltd, Pfizer Inc filed Critical Pfizer Ltd
Application granted granted Critical
Publication of DE69231445D1 publication Critical patent/DE69231445D1/de
Publication of DE69231445T2 publication Critical patent/DE69231445T2/de
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/62—Oxygen or sulfur atoms
    • C07D213/70—Sulfur atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/06—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Cephalosporin Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
DE69231445T 1991-10-10 1992-10-01 Triazole enthaltende antifungizide mittel Expired - Fee Related DE69231445T2 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB919121456A GB9121456D0 (en) 1991-10-10 1991-10-10 Triazole antifungal agents
PCT/EP1992/002278 WO1993007139A1 (en) 1991-10-10 1992-10-01 Triazole antifungal agents

Publications (2)

Publication Number Publication Date
DE69231445D1 true DE69231445D1 (de) 2000-10-19
DE69231445T2 DE69231445T2 (de) 2001-01-11

Family

ID=10702663

Family Applications (1)

Application Number Title Priority Date Filing Date
DE69231445T Expired - Fee Related DE69231445T2 (de) 1991-10-10 1992-10-01 Triazole enthaltende antifungizide mittel

Country Status (13)

Country Link
US (1) US5541203A (de)
EP (1) EP0607193B1 (de)
JP (1) JPH07502022A (de)
AT (1) ATE196293T1 (de)
CA (1) CA2118937C (de)
DE (1) DE69231445T2 (de)
DK (1) DK0607193T3 (de)
ES (1) ES2149777T3 (de)
FI (1) FI108131B (de)
GB (1) GB9121456D0 (de)
GR (1) GR3034769T3 (de)
PT (1) PT100942B (de)
WO (1) WO1993007139A1 (de)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9317491D0 (en) * 1993-08-23 1993-10-06 Fujisawa Pharmaceutical Co New compound and a process for preparation thereof
NZ270418A (en) * 1994-02-07 1997-09-22 Eisai Co Ltd Polycyclic triazole & imidazole derivatives, antifungal compositions
GB9512961D0 (en) * 1995-06-26 1995-08-30 Pfizer Ltd Antifungal agents
GB9605705D0 (en) * 1996-03-19 1996-05-22 Pfizer Ltd Therapeutic agents
KR100889937B1 (ko) * 2007-08-06 2009-03-20 한미약품 주식회사 보리코나졸의 제조방법
GB2452049A (en) * 2007-08-21 2009-02-25 Alpharma Aps Process for the preparation of voriconazole
WO2012177635A1 (en) * 2011-06-19 2012-12-27 Viamet Pharmaceuticals, Inc. Metalloenzyme inhibitor compounds
WO2012177603A2 (en) * 2011-06-19 2012-12-27 Viamet Pharmaceuticals, Inc. Metalloenzyme inhibitor compounds
ES2774267T3 (es) * 2012-01-20 2020-07-20 Mycovia Pharmaceuticals Inc Compuestos inhibidores de metaloenzimas
TWI561515B (en) * 2012-03-16 2016-12-11 Viamet Pharmaceuticals Inc Metalloenzyme inhibitor compounds
MX2017014848A (es) 2015-05-18 2018-04-20 Viamet Pharmaceuticals Nc Inc Compuestos antifungicos.
CN109996442A (zh) * 2016-11-22 2019-07-09 美国陶氏益农公司 用于谷物的真菌防治的杀真菌化合物和混合物
AR110209A1 (es) * 2016-11-22 2019-03-06 Viamet Pharmaceuticals Inc Uso de un compuesto de difluoro-(2-hidroxipropil)piridina como fungicida para el control de hongos fitopatógenos en maíz
WO2018098237A1 (en) * 2016-11-22 2018-05-31 Vps-3, Inc. Use of a difluoro-(2-hydroxypropyl)pyridine compound as a fungicide for control of leaf spot of sugar beets
UA124349C2 (uk) * 2016-11-22 2021-09-01 ДАУ АГРОСАЙЄНСІЗ ЕлЕлСі Застосування сполуки дифтор-(2-гідроксипропіл)піридину як фунгіциду для боротьби з фітопатогенним грибком ячменю
WO2018098256A1 (en) * 2016-11-22 2018-05-31 Vps-3, Inc. Use of a difluoro-(2-hydroxypropyl)pyridine compound as a fungicide for control of phytopathogenic fungi of rice
JP2019535756A (ja) * 2016-11-22 2019-12-12 ダウ アグロサイエンシィズ エルエルシー 殺真菌組成物および穀類における真菌防除のための混合物
AU2017363225A1 (en) * 2016-11-22 2019-06-20 Corteva Agriscience Llc Fungicidal compounds and mixtures for fungal control in cereals
US20230042961A1 (en) * 2016-11-22 2023-02-09 Dow Agrosciences Llc Fungicidal compounds and mixtures for fungal control in cereals
AR110206A1 (es) * 2016-11-22 2019-03-06 Viamet Pharmaceuticals Inc Uso de un compuesto de difluoro-(2-hidroxipropil)piridina como fungicida para el control de hongos fitopatógenos en trigo
EP3544426A4 (de) 2016-11-22 2020-04-29 Dow AgroSciences LLC Fungizide verbindungen und mischungen zur pilzbekämpfung in getreide

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE322526C (de) * 1918-08-31 1920-07-01 Hermann Meyer Sicherheitskettenverschluss fuer Korridortueren u. dgl.
EP0158741A3 (de) * 1980-11-19 1986-02-12 Imperial Chemical Industries Plc Zwischenprodukte für fungizide Triazol- und Imidazolverbindungen
ES8503680A1 (es) * 1982-06-17 1985-04-01 Pfizer Un procedimiento para la preparacion de un compuesto dotado de propiedades fungicidas
DE3245504A1 (de) * 1982-12-09 1984-06-14 Bayer Ag, 5090 Leverkusen Fungizide mittel, deren herstellung und verwendung
US4952232A (en) * 1987-04-29 1990-08-28 E. I. Du Pont De Nemours And Company Antifungal carbinols
DE3813841A1 (de) * 1987-06-03 1988-12-15 Bayer Ag Heterocyclische hydroxyethylazole
DE3732385A1 (de) * 1987-09-25 1989-04-06 Bayer Ag Hydroxyalkylcyclopropyl1-1,2,4-triazolyl- oder -imidazolyl-derivate und ihre verwendung als antimykotische mittel
EP0440608A1 (de) * 1987-12-17 1991-08-14 E.I. Du Pont De Nemours And Company Antifungale carbinole
NO171272C (no) * 1988-03-04 1993-02-17 Sankyo Co Analogifremgangsmaate til fremstilling av terapeutisk aktive 1,2,4-triazolforbindelser
GB8819308D0 (en) * 1988-08-13 1988-09-14 Pfizer Ltd Triazole antifungal agents
GB9002375D0 (en) * 1990-02-02 1990-04-04 Pfizer Ltd Triazole antifungal agents

Also Published As

Publication number Publication date
WO1993007139A1 (en) 1993-04-15
DE69231445T2 (de) 2001-01-11
FI941644A (fi) 1994-04-08
GR3034769T3 (en) 2001-02-28
FI941644A0 (fi) 1994-04-08
PT100942B (pt) 1999-07-30
DK0607193T3 (da) 2000-10-09
JPH07502022A (ja) 1995-03-02
GB9121456D0 (en) 1991-11-27
PT100942A (pt) 1993-10-29
EP0607193A1 (de) 1994-07-27
ES2149777T3 (es) 2000-11-16
CA2118937A1 (en) 1993-04-15
ATE196293T1 (de) 2000-09-15
EP0607193B1 (de) 2000-09-13
US5541203A (en) 1996-07-30
CA2118937C (en) 1998-04-28
FI108131B (fi) 2001-11-30

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