NO991594L - Tiosyreavledede, monosykliske N-heterosykluser som antikoagulanter - Google Patents

Tiosyreavledede, monosykliske N-heterosykluser som antikoagulanter

Info

Publication number
NO991594L
NO991594L NO991594A NO991594A NO991594L NO 991594 L NO991594 L NO 991594L NO 991594 A NO991594 A NO 991594A NO 991594 A NO991594 A NO 991594A NO 991594 L NO991594 L NO 991594L
Authority
NO
Norway
Prior art keywords
thioacid
anticoagulants
heterocycles
monocyclic
derived
Prior art date
Application number
NO991594A
Other languages
English (en)
Norwegian (no)
Other versions
NO991594D0 (no
Inventor
Monica J Kochanny
Michael M Morrissey
Howard P Ng
Original Assignee
Schering Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Schering Ag filed Critical Schering Ag
Publication of NO991594D0 publication Critical patent/NO991594D0/no
Publication of NO991594L publication Critical patent/NO991594L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Silicates, Zeolites, And Molecular Sieves (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pyridine Compounds (AREA)
NO991594A 1996-10-09 1999-03-31 Tiosyreavledede, monosykliske N-heterosykluser som antikoagulanter NO991594L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US08/731,128 US6004985A (en) 1996-10-09 1996-10-09 Thio acid derived monocylic N-heterocyclics as anticoagulants
PCT/EP1997/005231 WO1998015547A1 (en) 1996-10-09 1997-09-24 Thio acid derived monocyclic n-heterocyclics as anticoagulants

Publications (2)

Publication Number Publication Date
NO991594D0 NO991594D0 (no) 1999-03-31
NO991594L true NO991594L (no) 1999-06-08

Family

ID=24938188

Family Applications (1)

Application Number Title Priority Date Filing Date
NO991594A NO991594L (no) 1996-10-09 1999-03-31 Tiosyreavledede, monosykliske N-heterosykluser som antikoagulanter

Country Status (21)

Country Link
US (6) US6004985A (cs)
EP (1) EP0934310B1 (cs)
JP (1) JP3768244B2 (cs)
KR (1) KR20000048966A (cs)
CN (1) CN1111159C (cs)
AT (1) ATE288908T1 (cs)
AU (1) AU730060B2 (cs)
CA (1) CA2268172A1 (cs)
CZ (1) CZ122799A3 (cs)
DE (1) DE69732490T2 (cs)
DK (1) DK0934310T3 (cs)
ES (1) ES2236828T3 (cs)
HK (1) HK1020958A1 (cs)
HU (1) HUP9904180A3 (cs)
IL (1) IL129056A0 (cs)
NO (1) NO991594L (cs)
NZ (1) NZ334758A (cs)
PL (1) PL332602A1 (cs)
PT (1) PT934310E (cs)
SK (1) SK46499A3 (cs)
WO (1) WO1998015547A1 (cs)

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DE69821985T2 (de) 1997-12-19 2005-05-04 Schering Ag Ortho-anthranilamide derivate als antikoagulantien
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DK1569912T3 (en) 2002-12-03 2015-06-29 Pharmacyclics Inc 2- (2-hydroxybiphenyl-3-yl) -1h-benzoimidazole-5-carboxamidine derivatives as factor VIIa inhibitors.
US6875781B2 (en) * 2003-04-04 2005-04-05 Cell Therapeutics, Inc. Pyridines and uses thereof
US8178671B2 (en) * 2003-07-30 2012-05-15 Rigel Pharmaceuticals, Inc. Methods of treating or preventing autoimmune diseases with 2, 4-pyrimidinediamine compounds
WO2006068770A1 (en) * 2004-11-24 2006-06-29 Rigel Pharmaceuticals, Inc. Spiro-2, 4-pyrimidinediamine compounds and their uses
DE602006010979D1 (de) 2005-01-19 2010-01-21 Rigel Pharmaceuticals Inc Prodrugs aus 2,4-pyrimidindiamin-verbindungen und ihre verwendungen
CA2604551A1 (en) * 2005-05-03 2007-03-08 Rigel Pharmaceuticals, Inc. Jak kinase inhibitors and their uses
US20070015834A1 (en) * 2005-07-18 2007-01-18 Moshe Flashner-Barak Formulations of fenofibrate containing PEG/Poloxamer
US8138339B2 (en) 2008-04-16 2012-03-20 Portola Pharmaceuticals, Inc. Inhibitors of protein kinases
BRPI0910921B1 (pt) 2008-04-16 2022-06-21 Portola Pharmaceuticals, Inc Inibidores de proteína syk quinase, composição farmacêutica, kit e usos dos referidos inibidores
SI2300013T1 (en) 2008-05-21 2018-03-30 Adriad Pharmacaceuticals, Inc. Phosphorus derivatives as kinase inhibitors
US9273077B2 (en) 2008-05-21 2016-03-01 Ariad Pharmaceuticals, Inc. Phosphorus derivatives as kinase inhibitors
EA201391626A1 (ru) 2011-05-04 2014-03-31 Ариад Фармасьютикалз, Инк. Соединения для ингибирования клеточной пролиферации в egfr-стимулированных типах рака
CA2856301C (en) 2011-11-23 2020-10-06 Portola Pharmaceuticals, Inc. Pyrazine kinase inhibitors
JP6469567B2 (ja) 2012-05-05 2019-02-13 アリアド・ファーマシューティカルズ・インコーポレイテッド Ｅｇｆｒ発動性がんの細胞増殖阻害用化合物
US9611283B1 (en) 2013-04-10 2017-04-04 Ariad Pharmaceuticals, Inc. Methods for inhibiting cell proliferation in ALK-driven cancers
US10676436B2 (en) * 2018-07-05 2020-06-09 Landos Biopharma, Inc. NLRX1 ligands
US10487057B1 (en) * 2018-07-05 2019-11-26 Landos Biopharma, Inc. NLRX1 ligands
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Also Published As

Publication number Publication date
CZ122799A3 (cs) 1999-09-15
US6162807A (en) 2000-12-19
AU4624097A (en) 1998-05-05
CN1111159C (zh) 2003-06-11
JP2001501632A (ja) 2001-02-06
DE69732490D1 (en) 2005-03-17
JP3768244B2 (ja) 2006-04-19
SK46499A3 (en) 2000-04-10
US6004985A (en) 1999-12-21
HK1020958A1 (en) 2004-03-19
WO1998015547A1 (en) 1998-04-16
EP0934310B1 (en) 2005-02-09
PL332602A1 (en) 1999-09-27
NZ334758A (en) 2000-11-24
DK0934310T3 (da) 2005-05-30
HUP9904180A2 (hu) 2000-09-28
ES2236828T3 (es) 2005-07-16
CN1233247A (zh) 1999-10-27
AU730060B2 (en) 2001-02-22
ATE288908T1 (de) 2005-02-15
CA2268172A1 (en) 1998-04-16
EP0934310A1 (en) 1999-08-11
HUP9904180A3 (en) 2000-11-28
US6221886B1 (en) 2001-04-24
DE69732490T2 (de) 2006-04-27
NO991594D0 (no) 1999-03-31
KR20000048966A (ko) 2000-07-25
US6034084A (en) 2000-03-07
US6150382A (en) 2000-11-21
US6166014A (en) 2000-12-26
PT934310E (pt) 2005-06-30
IL129056A0 (en) 2000-02-17

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