NO990484L - Aminosyreester inneholdende azol antisoppmiddel - Google Patents

Aminosyreester inneholdende azol antisoppmiddel

Info

Publication number
NO990484L
NO990484L NO990484A NO990484A NO990484L NO 990484 L NO990484 L NO 990484L NO 990484 A NO990484 A NO 990484A NO 990484 A NO990484 A NO 990484A NO 990484 L NO990484 L NO 990484L
Authority
NO
Norway
Prior art keywords
amino acid
acid ester
antifungal agent
ester containing
azole antifungal
Prior art date
Application number
NO990484A
Other languages
English (en)
Other versions
NO990484D0 (no
NO316668B1 (no
Inventor
Lieven Meerpoel
Jan Heeres
Robert Jozef Maria Hendrickx
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of NO990484D0 publication Critical patent/NO990484D0/no
Publication of NO990484L publication Critical patent/NO990484L/no
Publication of NO316668B1 publication Critical patent/NO316668B1/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D249/00Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/081,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10Antimycotics
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
NO19990484A 1997-02-11 1999-02-02 Aminosyreesterinneholdende azoler, deres mellomprodukter og anvendelse av forbindelsene, samt farmasoytiske blandinger NO316668B1 (no)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP97200374 1997-02-11
EP97203228 1997-10-15
PCT/EP1998/000646 WO1998034934A1 (en) 1997-02-11 1998-02-03 Amino acid ester containing azole antifungals

Publications (3)

Publication Number Publication Date
NO990484D0 NO990484D0 (no) 1999-02-02
NO990484L true NO990484L (no) 1999-10-11
NO316668B1 NO316668B1 (no) 2004-03-29

Family

ID=26146124

Family Applications (1)

Application Number Title Priority Date Filing Date
NO19990484A NO316668B1 (no) 1997-02-11 1999-02-02 Aminosyreesterinneholdende azoler, deres mellomprodukter og anvendelse av forbindelsene, samt farmasoytiske blandinger

Country Status (31)

Country Link
US (3) US6262052B1 (no)
EP (1) EP0958289B1 (no)
JP (1) JP4347911B2 (no)
KR (1) KR100509171B1 (no)
CN (1) CN1238353C (no)
AT (1) ATE270290T1 (no)
AU (1) AU725302C (no)
BG (1) BG63872B1 (no)
BR (1) BR9809744A (no)
CA (1) CA2262791C (no)
CZ (1) CZ297197B6 (no)
DE (1) DE69824834T2 (no)
DK (1) DK0958289T3 (no)
EE (1) EE03876B1 (no)
ES (1) ES2224364T3 (no)
HU (1) HU227744B1 (no)
ID (1) ID21755A (no)
IL (2) IL128513A (no)
MY (1) MY129537A (no)
NO (1) NO316668B1 (no)
NZ (1) NZ334477A (no)
PL (1) PL191152B1 (no)
PT (1) PT958289E (no)
RU (1) RU2197489C2 (no)
SI (1) SI0958289T1 (no)
SK (1) SK284910B6 (no)
TR (1) TR199900584T2 (no)
TW (1) TW495508B (no)
UA (1) UA61919C2 (no)
WO (1) WO1998034934A1 (no)
ZA (1) ZA981079B (no)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0957101A1 (en) * 1998-05-14 1999-11-17 Janssen Pharmaceutica N.V. Water soluble azoles as broad-spectrum antifungals
WO2000030655A1 (en) 1998-11-20 2000-06-02 Bristol-Myers Squibb Company Water soluble prodrugs of azole compounds
EA200101172A1 (ru) 1999-05-04 2002-04-25 Янссен Фармацевтика Н.В. Противогрибковые эфиры
WO2003052117A2 (en) * 2001-09-19 2003-06-26 Massachusetts Institute Of Technology Methods and products related to non-viral transfection
ITMI20032020A1 (it) * 2003-10-17 2005-04-18 Italfarmaco Spa Nuovi agenti antifungini azolici con diminuita interazione con i citocromi metabolici
RU2585760C2 (ru) * 2010-05-19 2016-06-10 Сандоз Аг Способ получения хиральных триазолонов
AU2015380298B2 (en) 2014-12-30 2019-02-21 Corteva Agriscience Llc Picolinamide compounds with fungicidal activity
BR102019004480B1 (pt) * 2018-03-08 2023-03-28 Dow Agrosciences Llc Picolinamidas como fungicidas
CN111138421A (zh) * 2019-12-26 2020-05-12 上海英诺富成生物科技有限公司 抗真菌水溶性化合物及其制备方法与应用

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4267179A (en) 1978-06-23 1981-05-12 Janssen Pharmaceutica, N.V. Heterocyclic derivatives of (4-phenylpiperazin-1-yl-aryloxymethyl-1,3-dioxolan-2-yl)methyl-1H-imidazoles and 1H-1,2,4-triazoles
US4791111A (en) * 1985-12-23 1988-12-13 Janssen Pharmaceutica, N.V. [[4-[4-(4-phenyl-1-piperazinyl)phenoxymethyl]-1,3-dioxolan-2-yl]methyl]-1H-imidazoles and 1H-1,2,4-triazoles having anti-microbial properties
US4916134A (en) 1987-03-25 1990-04-10 Janssen Pharmacuetica N.V. 4-[4-[4-[4-[[2-(2,4-difluorophenyl)-2-(1H-azolylmethyl)-1,3-dioxolan-4-yl]me]phenyl]-1-piperazinyl]phenyl]triazolones
CA1331757C (en) 1988-02-29 1994-08-30 Janssen Pharmaceutica Naamloze Vennootschap 5-lipoxygenase inhibiting 4-(4-phenyl-1-piperazinyl)phenols
HU221189B1 (en) 1992-03-18 2002-08-28 Janssen Pharmaceutica Nv Itraconazole and saperconazole stereoisomers, their cyclodextrin complexes and pharmaceutical compositions containing them and process for producing them
ES2159623T3 (es) * 1993-12-21 2001-10-16 Schering Corp Antifungicos de tetrahidrofurano.
WO1995019983A1 (en) * 1994-01-24 1995-07-27 Janssen Pharmaceutica N.V. Watersoluble azole antifungals
CA2197672C (en) * 1995-06-02 2011-05-17 Anil K. Saksena Tetrahydrofuran antifungals
AU6257396A (en) * 1995-06-19 1997-01-15 Schering Corporation Tetrahydrofuran antifungals

Also Published As

Publication number Publication date
US20010039281A1 (en) 2001-11-08
EP0958289B1 (en) 2004-06-30
US6703506B2 (en) 2004-03-09
PL332008A1 (en) 1999-08-16
MY129537A (en) 2007-04-30
CN1236366A (zh) 1999-11-24
ATE270290T1 (de) 2004-07-15
RU2197489C2 (ru) 2003-01-27
NZ334477A (en) 2001-05-25
CZ297197B6 (cs) 2006-09-13
EE9900100A (et) 1999-10-15
KR100509171B1 (ko) 2005-08-22
BG63872B1 (bg) 2003-04-30
NO990484D0 (no) 1999-02-02
BR9809744A (pt) 2000-06-20
IL149285A0 (en) 2002-11-10
IL149285A (en) 2007-08-19
US6512116B2 (en) 2003-01-28
SK284910B6 (sk) 2006-02-02
DK0958289T3 (da) 2004-11-01
EE03876B1 (et) 2002-10-15
HUP0001050A2 (hu) 2001-04-28
CZ283599A3 (cs) 2000-02-16
IL128513A0 (en) 2000-01-31
DE69824834T2 (de) 2005-07-21
IL128513A (en) 2002-11-10
TW495508B (en) 2002-07-21
HUP0001050A3 (en) 2001-07-30
EP0958289A1 (en) 1999-11-24
JP4347911B2 (ja) 2009-10-21
ZA981079B (en) 1999-08-10
HU227744B1 (en) 2012-02-28
JP2001508080A (ja) 2001-06-19
ES2224364T3 (es) 2005-03-01
DE69824834D1 (de) 2004-08-05
NO316668B1 (no) 2004-03-29
TR199900584T2 (xx) 1999-10-21
ID21755A (id) 1999-07-22
UA61919C2 (uk) 2003-12-15
PT958289E (pt) 2004-11-30
CN1238353C (zh) 2006-01-25
BG103171A (en) 1999-09-30
PL191152B1 (pl) 2006-03-31
CA2262791A1 (en) 1998-08-13
KR20000068526A (ko) 2000-11-25
US20030158210A1 (en) 2003-08-21
SI0958289T1 (en) 2004-12-31
AU725302B2 (en) 2000-10-12
WO1998034934A1 (en) 1998-08-13
SK105999A3 (en) 2000-06-12
US6262052B1 (en) 2001-07-17
AU6620798A (en) 1998-08-26
AU725302C (en) 2001-08-23
CA2262791C (en) 2008-10-28

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