NO982580D0 - Nye taxoider, deres fremstilling samt farmas°ystiske preparater inneholdende taxoidene - Google Patents

Nye taxoider, deres fremstilling samt farmas°ystiske preparater inneholdende taxoidene

Info

Publication number
NO982580D0
NO982580D0 NO982580A NO982580A NO982580D0 NO 982580 D0 NO982580 D0 NO 982580D0 NO 982580 A NO982580 A NO 982580A NO 982580 A NO982580 A NO 982580A NO 982580 D0 NO982580 D0 NO 982580D0
Authority
NO
Norway
Prior art keywords
taxoids
preparation
pharmaceutical preparations
preparations containing
new
Prior art date
Application number
NO982580A
Other languages
English (en)
Other versions
NO982580L (no
NO317358B1 (no
Inventor
Herve Bouchard
Alain Commercon
Original Assignee
Rhone Poulenc Rorer Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Rhone Poulenc Rorer Sa filed Critical Rhone Poulenc Rorer Sa
Publication of NO982580L publication Critical patent/NO982580L/no
Publication of NO982580D0 publication Critical patent/NO982580D0/no
Publication of NO317358B1 publication Critical patent/NO317358B1/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D493/00—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
    • C07D493/02—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains two hetero rings
    • C07D493/08—Bridged systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D305/00—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms
    • C07D305/14—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms condensed with carbocyclic rings or ring systems
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
NO19982580A 1995-12-22 1998-06-05 Nye taxoider, deres fremstilling samt farmasoystiske preparater inneholdende taxoidene NO317358B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9515379A FR2742751B1 (fr) 1995-12-22 1995-12-22 Nouveaux taxoides, leur preparation et les compositions pharmaceutiques qui les contiennent
PCT/FR1996/002031 WO1997023473A1 (fr) 1995-12-22 1996-12-19 Nouveaux taxoides, leur preparation et les compositions pharmaceutiques qui les contiennent

Publications (3)

Publication Number Publication Date
NO982580L NO982580L (no) 1998-06-05
NO982580D0 true NO982580D0 (no) 1998-06-05
NO317358B1 NO317358B1 (no) 2004-10-18

Family

ID=9485871

Family Applications (1)

Application Number Title Priority Date Filing Date
NO19982580A NO317358B1 (no) 1995-12-22 1998-06-05 Nye taxoider, deres fremstilling samt farmasoystiske preparater inneholdende taxoidene

Country Status (41)

Country Link
US (1) US5728849A (no)
EP (1) EP0876362B1 (no)
JP (1) JP3953106B2 (no)
KR (1) KR100500351B1 (no)
CN (1) CN1103766C (no)
AR (1) AR005197A1 (no)
AT (1) ATE250593T1 (no)
AU (1) AU712597B2 (no)
BG (1) BG63204B1 (no)
BR (1) BR9612135A (no)
CA (1) CA2238884C (no)
CO (1) CO4520184A1 (no)
CZ (1) CZ294972B6 (no)
DE (1) DE69630145T2 (no)
DK (1) DK0876362T3 (no)
DZ (1) DZ2149A1 (no)
EA (1) EA001533B1 (no)
ES (1) ES2202490T3 (no)
FR (1) FR2742751B1 (no)
HK (1) HK1017895A1 (no)
HU (1) HU225032B1 (no)
IL (1) IL124994A (no)
IN (4) IN186768B (no)
MA (1) MA26412A1 (no)
MX (1) MX9804688A (no)
MY (1) MY113934A (no)
NO (1) NO317358B1 (no)
NZ (1) NZ324337A (no)
OA (1) OA10700A (no)
PE (1) PE25198A1 (no)
PL (1) PL189311B1 (no)
PT (1) PT876362E (no)
RO (1) RO116194B1 (no)
SK (1) SK282835B6 (no)
TN (1) TNSN96169A1 (no)
TR (1) TR199801179T2 (no)
TW (1) TW371659B (no)
UA (1) UA48205C2 (no)
UY (1) UY24386A1 (no)
WO (1) WO1997023473A1 (no)
ZA (1) ZA9610737B (no)

Families Citing this family (39)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9920548D0 (en) * 1999-08-31 1999-11-03 Rhone Poulenc Rorer Sa Treatment of hepatocellular carcinoma
MXPA01009902A (es) 2000-02-02 2003-07-28 Univ Florida State Res Found Taxanos sustituidos con carbonato en c10 como agentes antitumor.
DK1368349T3 (da) * 2001-02-24 2007-05-21 Boehringer Ingelheim Pharma Xanthinderivater, deres fremstilling og deres anvendelse som lægemidler
US7407955B2 (en) 2002-08-21 2008-08-05 Boehringer Ingelheim Pharma Gmbh & Co., Kg 8-[3-amino-piperidin-1-yl]-xanthines, the preparation thereof and their use as pharmaceutical compositions
CA2526278A1 (en) * 2003-05-20 2004-12-02 Aronex Pharmaceuticals, Inc. Combination chemotherapy comprising a liposomal platinum complex
US7501426B2 (en) 2004-02-18 2009-03-10 Boehringer Ingelheim International Gmbh 8-[3-amino-piperidin-1-yl]-xanthines, their preparation and their use as pharmaceutical compositions
DE102004054054A1 (de) 2004-11-05 2006-05-11 Boehringer Ingelheim Pharma Gmbh & Co. Kg Verfahren zur Herstellung chiraler 8-(3-Amino-piperidin-1-yl)-xanthine
EP1669358A1 (en) * 2004-12-07 2006-06-14 Aventis Pharma S.A. Cytotoxic agents comprising new taxanes
DE102005035891A1 (de) 2005-07-30 2007-02-08 Boehringer Ingelheim Pharma Gmbh & Co. Kg 8-(3-Amino-piperidin-1-yl)-xanthine, deren Herstellung und deren Verwendung als Arzneimittel
EP1852108A1 (en) 2006-05-04 2007-11-07 Boehringer Ingelheim Pharma GmbH & Co.KG DPP IV inhibitor formulations
PE20110235A1 (es) 2006-05-04 2011-04-14 Boehringer Ingelheim Int Combinaciones farmaceuticas que comprenden linagliptina y metmorfina
MX2008014024A (es) 2006-05-04 2008-11-14 Boehringer Ingelheim Int Formas poliformas.
US20080207743A1 (en) * 2007-02-28 2008-08-28 Rodger Lamb Biologically Active Taxane Analogs and Methods of Treatment
AU2008290582B2 (en) * 2007-08-17 2014-08-14 Boehringer Ingelheim International Gmbh Purin derivatives for use in the treatment of fab-related diseases
PE20140960A1 (es) 2008-04-03 2014-08-15 Boehringer Ingelheim Int Formulaciones que comprenden un inhibidor de dpp4
PE20100156A1 (es) * 2008-06-03 2010-02-23 Boehringer Ingelheim Int Tratamiento de nafld
UY32030A (es) 2008-08-06 2010-03-26 Boehringer Ingelheim Int "tratamiento para diabetes en pacientes inapropiados para terapia con metformina"
KR20200118243A (ko) 2008-08-06 2020-10-14 베링거 인겔하임 인터내셔날 게엠베하 메트포르민 요법이 부적합한 환자에서의 당뇨병 치료
WO2010029089A2 (en) 2008-09-10 2010-03-18 Boehringer Ingelheim International Gmbh Combination therapy for the treatment of diabetes and related conditions
US20200155558A1 (en) 2018-11-20 2020-05-21 Boehringer Ingelheim International Gmbh Treatment for diabetes in patients with insufficient glycemic control despite therapy with an oral antidiabetic drug
WO2010072776A1 (en) 2008-12-23 2010-07-01 Boehringer Ingelheim International Gmbh Salt forms of organic compound
AR074990A1 (es) 2009-01-07 2011-03-02 Boehringer Ingelheim Int Tratamiento de diabetes en pacientes con un control glucemico inadecuado a pesar de la terapia con metformina
UY32048A (es) * 2009-01-08 2010-03-26 Boehringer Ingelheim Int Derivados sustituido de 1-(sustituido)-3-metil-7-(sustituido)-8-(3-(R)-amino-piperidin-1-il)cantina y derivados sustituidos de 1-(sustituido) - 4 - fluoropirrolidin- 2 - carbonitrilo y sus sales famacéuticamente aceptables como inhibidores de DPP-4 y aplicaciones.
CN102753161A (zh) 2009-11-27 2012-10-24 贝林格尔.英格海姆国际有限公司 基因型糖尿病患者利用dpp-iv抑制剂例如利拉利汀的治疗
ES2935300T3 (es) 2010-05-05 2023-03-03 Boehringer Ingelheim Int Combiterapia
CN106975074A (zh) 2010-06-24 2017-07-25 勃林格殷格翰国际有限公司 糖尿病治疗
US9034883B2 (en) 2010-11-15 2015-05-19 Boehringer Ingelheim International Gmbh Vasoprotective and cardioprotective antidiabetic therapy
WO2013010964A1 (en) 2011-07-15 2013-01-24 Boehringer Ingelheim International Gmbh Substituted quinazolines, the preparation thereof and the use thereof in pharmaceutical compositions
US9555001B2 (en) 2012-03-07 2017-01-31 Boehringer Ingelheim International Gmbh Pharmaceutical composition and uses thereof
WO2013171167A1 (en) 2012-05-14 2013-11-21 Boehringer Ingelheim International Gmbh A xanthine derivative as dpp -4 inhibitor for use in the treatment of podocytes related disorders and/or nephrotic syndrome
WO2013174767A1 (en) 2012-05-24 2013-11-28 Boehringer Ingelheim International Gmbh A xanthine derivative as dpp -4 inhibitor for use in modifying food intake and regulating food preference
CN105849086B (zh) 2012-11-24 2018-07-31 杭州多禧生物科技有限公司 亲水性链接体及其在药物分子和细胞结合分子共轭反应上的应用
FR3010839B1 (fr) * 2013-09-17 2017-04-21 Schneider Electric Ind Sas Dispositif de raccordement electrique d'au moins un conducteur dans une borne appartenant a un appareil electrique
US9526728B2 (en) 2014-02-28 2016-12-27 Boehringer Ingelheim International Gmbh Medical use of a DPP-4 inhibitor
DK3122757T3 (da) 2014-02-28 2023-10-09 Hangzhou Dac Biotech Co Ltd Ladede linkere og anvendelse deraf til konjugering
EP3319936A4 (en) 2015-07-12 2019-02-06 Suzhou M-conj Biotech Co., Ltd. PLACES OF CONDUCT FOR THE CONJUGATION OF CELL BINDING MOLECULES
US9839687B2 (en) 2015-07-15 2017-12-12 Suzhou M-Conj Biotech Co., Ltd. Acetylenedicarboxyl linkers and their uses in specific conjugation of a cell-binding molecule
BR112018072401A2 (pt) 2016-06-10 2019-02-19 Boehringer Ingelheim International Gmbh combinações de linagliptina e metformina
WO2018086139A1 (en) 2016-11-14 2018-05-17 Hangzhou Dac Biotech Co., Ltd Conjugation linkers, cell binding molecule-drug conjugates containing the likers, methods of making and uses such conjugates with the linkers

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RU2017724C1 (ru) * 1990-07-12 1994-08-15 Дзе Юниверсити оф Канзас Способ получения производных таксола
US5059699A (en) * 1990-08-28 1991-10-22 Virginia Tech Intellectual Properties, Inc. Water soluble derivatives of taxol
FR2678930B1 (fr) * 1991-07-10 1995-01-13 Rhone Poulenc Rorer Sa Procede de preparation de derives de la baccatine iii et de la desacetyl-10 baccatine iii.
RU2059631C1 (ru) * 1991-11-29 1996-05-10 Дзе Юниверсити оф Канзас Производные таксола и фармацевтическая композиция, обладающая противоопухолевой активностью
EP0639186B1 (en) * 1992-04-17 1999-06-23 Abbott Laboratories Taxol derivatives
US5254580A (en) * 1993-01-19 1993-10-19 Bristol-Myers Squibb Company 7,8-cyclopropataxanes
IL107950A (en) * 1992-12-15 2001-04-30 Upjohn Co b 7, b 8 - Matano - Taxols, their preparation and pharmaceutical preparations against malignant tumors containing them

Also Published As

Publication number Publication date
FR2742751B1 (fr) 1998-01-30
AR005197A1 (es) 1999-04-14
US5728849A (en) 1998-03-17
IN188469B (no) 2002-09-28
DE69630145T2 (de) 2004-07-15
HUP9904046A1 (hu) 2001-04-28
EA199800588A1 (ru) 1998-12-24
MY113934A (en) 2002-06-29
CA2238884C (fr) 2007-02-06
IN188470B (no) 2002-09-28
NO982580L (no) 1998-06-05
AU712597B2 (en) 1999-11-11
NZ324337A (en) 2000-03-27
CA2238884A1 (fr) 1997-07-03
WO1997023473A1 (fr) 1997-07-03
NO317358B1 (no) 2004-10-18
SK282835B6 (sk) 2002-12-03
IL124994A0 (en) 1999-01-26
MX9804688A (es) 1998-10-31
TNSN96169A1 (fr) 2005-03-15
CN1103766C (zh) 2003-03-26
BR9612135A (pt) 1999-07-13
IN188680B (no) 2002-10-26
IN186768B (no) 2001-11-03
CO4520184A1 (es) 1997-10-15
CZ294972B6 (cs) 2005-04-13
OA10700A (fr) 2002-11-27
BG102569A (en) 1999-04-30
PL327405A1 (en) 1998-12-07
TW371659B (en) 1999-10-11
FR2742751A1 (fr) 1997-06-27
AU1180997A (en) 1997-07-17
EP0876362A1 (fr) 1998-11-11
JP2000502671A (ja) 2000-03-07
PE25198A1 (es) 1998-05-10
HU225032B1 (en) 2006-05-29
KR100500351B1 (ko) 2005-12-21
DK0876362T3 (da) 2004-02-02
ATE250593T1 (de) 2003-10-15
IL124994A (en) 2000-12-06
EP0876362B1 (fr) 2003-09-24
HK1017895A1 (en) 1999-12-03
SK85398A3 (en) 1998-11-04
KR19990076680A (ko) 1999-10-15
JP3953106B2 (ja) 2007-08-08
DE69630145D1 (de) 2003-10-30
RO116194B1 (ro) 2000-11-30
DZ2149A1 (fr) 2002-10-23
BG63204B1 (bg) 2001-06-29
PT876362E (pt) 2004-02-27
ZA9610737B (en) 1997-06-27
CN1205697A (zh) 1999-01-20
CZ196198A3 (cs) 1998-09-16
ES2202490T3 (es) 2004-04-01
UA48205C2 (uk) 2002-08-15
MA26412A1 (fr) 2004-12-20
UY24386A1 (es) 2001-08-27
HUP9904046A3 (en) 2001-08-28
TR199801179T2 (xx) 1998-10-21
EA001533B1 (ru) 2001-04-23
PL189311B1 (pl) 2005-07-29

Similar Documents

Publication Publication Date Title
NO982580D0 (no) Nye taxoider, deres fremstilling samt farmas°ystiske preparater inneholdende taxoidene
NO973923D0 (no) Nye taxoider, deres fremstilling samt farmasöytiske preparater inneholdende forbindelsene
FI943570A0 (fi) 1-bentseenisulfonyyli-1,3-dihydroindol-2-onijohdannaisia, niiden valmistus ja niitä sisältäviä lääkeaineita
NO944700D0 (no) Nye tienotiazinderivater, fremgangsmåte for fremstilling derav samt farmasöytiske preparater inneholdende forbindelsene
NO973222D0 (no) Nye farnesyl-transferase-inhibitorer, deres fremstilling samt farmasöytiske preparater inneholdende inhibitorene
NO973608D0 (no) Nye farnesyl-transferaseinhibitorer, deres fremstilling samt farmasöytiske preparater inneholdende forbindelsene
NO2009028I1 (no) Kinazolin-derivater, anvendelse og fremstilling derav, samt farmasøytisk preparat
DE122005000024I1 (de) Darifenacin enthaltende Pharmazeutische Zubereitungen.
NL300249I2 (en) Cephalosporins and homologues, preparations and pharmaceutical preparations.
NO307459B1 (no) Piperazinderivater, samt farmasøytiske preparater inneholdende slike
NO952677D0 (no) Nye dihydropyrrolopyridinon- og oksazolopyridinonforbindelser, deres fremstilling og farmasöytiske preparater
NO305903B1 (no) Benzonitriler og benzofluorider, legemidler bestående av forbindelsene, farmasöytiske preparater inneholdende forbindelsene, samt anvendelse av forbindelsene for fremstilling av farmasöytiske preparater
NO951283D0 (no) Nye taxanderivater, deres fremstilling samt farmasöytiske preparater inneholdende derivatene
NO942910L (no) Nye baccatin-III- og 10-desacetyl-baccatin-III-derivater, deres fremstillinger, samt farmasöytiske preparater inneholdende derivatene
NO307510B1 (no) Bicykliske aromatiske forbindelser, deres anvendelse og farmasøytiske og kosmetiske preparater derav
DK0820448T3 (da) Nye taxoider, deres fremstilling og farmaceutiske præparater deraf
FI890488A (fi) Vaextextrakt innehaollande farmaceutiska preparat samt foerfarande foer framstaellning daerav.
NO20016247L (no) Streptograminderivater, deres fremstilling samt preparater inneholdende derivatene
NO983472D0 (no) Taxoider, deres fremstilling og farmas°ytiske preparater inneholdende taxoidene
NO974563D0 (no) Nye taxoider, deres fremstilling samt farmasöytiske preparater inneholdende forbindelsene
NO20003661D0 (no) Nye pentasakkarider, fremgangsmÕter for deres fremstilling og farmasøytiske preparater inneholdende de samme
NO308527B1 (no) Substituerte 2-naftoylguanidiner, deres anvendelse for fremstilling av et medikament samt legemidler og preparater inneholdende forbindelsene
FI955679A (fi) Piperidiinijohdannaisia, niiden valmistus ja käyttö
DK469189D0 (da) Substituerede thienopyraner, fremgangsmaade til fremstilling deraf samt farmaceutiske praeparater indeholdende samme
NO20024590L (no) Farmasöytiske preparater inneholdende oligosakkarider, de nye oligosakkarider samt deres fremstilling

Legal Events

Date Code Title Description
MM1K Lapsed by not paying the annual fees