NO972169L - Acylerte insulinanaloger - Google Patents

Acylerte insulinanaloger

Info

Publication number
NO972169L
NO972169L NO972169A NO972169A NO972169L NO 972169 L NO972169 L NO 972169L NO 972169 A NO972169 A NO 972169A NO 972169 A NO972169 A NO 972169A NO 972169 L NO972169 L NO 972169L
Authority
NO
Norway
Prior art keywords
chain
insulin analogues
acylated insulin
insulin
acylated
Prior art date
Application number
NO972169A
Other languages
English (en)
Other versions
NO972169D0 (no
Inventor
Jeffrey Clayton Baker
Jose Michel Hanquier
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of NO972169L publication Critical patent/NO972169L/no
Publication of NO972169D0 publication Critical patent/NO972169D0/no

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • A61K38/22—Hormones
    • A61K38/28—Insulins
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/575—Hormones
    • C07K14/62—Insulins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/38—Drugs for disorders of the endocrine system of the suprarenal hormones
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

Abstract

Monomer insulinanalog for bruk i forbindelse med diabetes og hvori A-kjeden er den naturlig forekommende sekvensen i den humane insulin A-kjeden og B-kjeden er modifisert ved enten stilling B28 og B29 eller begge. Analogen er monoacylert ved N- terminalen i A-kjeden eller B-kjeden eller ved lysindelen. De acylerte insulinanalogene har en langvarig virkningsvarighet.
NO972169A 1994-11-17 1997-05-12 Acylerte insulinanaloger NO972169D0 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US08/342,931 US5693609A (en) 1994-11-17 1994-11-17 Acylated insulin analogs
PCT/US1995/014873 WO1996015804A1 (en) 1994-11-17 1995-11-14 Acylated insulin analogs

Publications (2)

Publication Number Publication Date
NO972169L true NO972169L (no) 1997-05-12
NO972169D0 NO972169D0 (no) 1997-05-12

Family

ID=23343907

Family Applications (1)

Application Number Title Priority Date Filing Date
NO972169A NO972169D0 (no) 1994-11-17 1997-05-12 Acylerte insulinanaloger

Country Status (25)

Country Link
US (2) US5693609A (no)
EP (1) EP0712861B1 (no)
JP (1) JPH10511644A (no)
KR (1) KR970706842A (no)
AR (1) AR002700A1 (no)
AT (1) ATE237635T1 (no)
AU (1) AU711282B2 (no)
BR (1) BR9509653A (no)
CA (1) CA2205060A1 (no)
CO (1) CO4520284A1 (no)
CZ (1) CZ145797A3 (no)
DE (1) DE69530353T2 (no)
ES (1) ES2194890T3 (no)
FI (1) FI972031A (no)
HU (1) HUT77030A (no)
IL (1) IL115973A (no)
NO (1) NO972169D0 (no)
NZ (1) NZ297257A (no)
PL (1) PL320644A1 (no)
RU (1) RU2160118C2 (no)
TR (1) TR199501420A2 (no)
TW (1) TW434259B (no)
WO (1) WO1996015804A1 (no)
YU (1) YU71395A (no)
ZA (1) ZA959679B (no)

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WO1996015804A1 (en) 1996-05-30
FI972031A0 (fi) 1997-05-13
AR002700A1 (es) 1998-04-29
AU4237396A (en) 1996-06-17
IL115973A (en) 2001-08-26
US5693609A (en) 1997-12-02
MX9703508A (es) 1997-07-31
US5922675A (en) 1999-07-13
AU711282B2 (en) 1999-10-07
DE69530353T2 (de) 2004-02-19
YU71395A (sh) 1998-07-10
DE69530353D1 (de) 2003-05-22
NO972169D0 (no) 1997-05-12
BR9509653A (pt) 1997-09-16
TW434259B (en) 2001-05-16
EP0712861A3 (en) 1998-03-11
NZ297257A (en) 1999-05-28
ATE237635T1 (de) 2003-05-15
EP0712861B1 (en) 2003-04-16
CO4520284A1 (es) 1997-10-15
FI972031A (fi) 1997-05-14
IL115973A0 (en) 1996-01-31
TR199501420A2 (tr) 1996-06-21
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ZA959679B (en) 1997-05-14
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HUT77030A (hu) 1998-03-02
RU2160118C2 (ru) 2000-12-10

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