NO332757B1 - 3-substituerte 2(arylalkyl)-1-azabicykloalkaner,farmasoytiske preparater omfattende slike, slike forbindelser for anvendelse som medikament samt slike forbindelser for behandling av sykdom. - Google Patents

3-substituerte 2(arylalkyl)-1-azabicykloalkaner,farmasoytiske preparater omfattende slike, slike forbindelser for anvendelse som medikament samt slike forbindelser for behandling av sykdom. Download PDF

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Publication number
NO332757B1
NO332757B1 NO20054052A NO20054052A NO332757B1 NO 332757 B1 NO332757 B1 NO 332757B1 NO 20054052 A NO20054052 A NO 20054052A NO 20054052 A NO20054052 A NO 20054052A NO 332757 B1 NO332757 B1 NO 332757B1
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NO
Norway
Prior art keywords
compounds
pyridinyl
azabicyclo
compound according
methyl
Prior art date
Application number
NO20054052A
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English (en)
Norwegian (no)
Other versions
NO20054052L (no
NO20054052D0 (no
Inventor
Craig H Miller
Anatoly A Mazurov
Jozef Klucik
Lan Miao
Angela S Seamans
Teresa Youngpeter Phillips
Jeffrey Daniel Schmitt
Original Assignee
Targacept Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Publication date
Application filed by Targacept Inc filed Critical Targacept Inc
Publication of NO20054052D0 publication Critical patent/NO20054052D0/no
Publication of NO20054052L publication Critical patent/NO20054052L/no
Publication of NO332757B1 publication Critical patent/NO332757B1/no

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/08—Bridged systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K51/00—Preparations containing radioactive substances for use in therapy or testing in vivo
    • A61K51/02—Preparations containing radioactive substances for use in therapy or testing in vivo characterised by the carrier, i.e. characterised by the agent or material covalently linked or complexing the radioactive nucleus
    • A61K51/04—Organic compounds
    • A61K51/041—Heterocyclic compounds
    • A61K51/044—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins
    • A61K51/0455—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
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    • C07D453/00—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
    • C07D453/02—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/08—Bridged systems

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NO20054052A 2003-02-21 2005-08-31 3-substituerte 2(arylalkyl)-1-azabicykloalkaner,farmasoytiske preparater omfattende slike, slike forbindelser for anvendelse som medikament samt slike forbindelser for behandling av sykdom. NO332757B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US10/372,642 US6953855B2 (en) 1998-12-11 2003-02-21 3-substituted-2(arylalkyl)-1-azabicycloalkanes and methods of use thereof
PCT/US2004/005044 WO2004076449A2 (en) 2003-02-21 2004-02-20 3-substituted-2(arylalkyl)-1-azabicycloalkanes and methods of use thereof

Publications (3)

Publication Number Publication Date
NO20054052D0 NO20054052D0 (no) 2005-08-31
NO20054052L NO20054052L (no) 2005-10-21
NO332757B1 true NO332757B1 (no) 2013-01-07

Family

ID=32926222

Family Applications (3)

Application Number Title Priority Date Filing Date
NO20054052A NO332757B1 (no) 2003-02-21 2005-08-31 3-substituerte 2(arylalkyl)-1-azabicykloalkaner,farmasoytiske preparater omfattende slike, slike forbindelser for anvendelse som medikament samt slike forbindelser for behandling av sykdom.
NO20110013A NO332759B1 (no) 2003-02-21 2011-01-06 3-substituerte 2(arylalkyl)-1-azabicykloalkaner, farmasoytiske preparater omfattende slike, slike forbindelser for anvendelse som medikament samt slike forbindelser for behandling av sykdom.
NO20110014A NO332760B1 (no) 2003-02-21 2011-01-06 3-substituerte 2(arylalkyl)-1-azabicykloalkaner, farmasoytiske preparater omfattende slike, slike forbindelser for anvendelse som medikament samt slike forbindelser for behandling av sykdom.

Family Applications After (2)

Application Number Title Priority Date Filing Date
NO20110013A NO332759B1 (no) 2003-02-21 2011-01-06 3-substituerte 2(arylalkyl)-1-azabicykloalkaner, farmasoytiske preparater omfattende slike, slike forbindelser for anvendelse som medikament samt slike forbindelser for behandling av sykdom.
NO20110014A NO332760B1 (no) 2003-02-21 2011-01-06 3-substituerte 2(arylalkyl)-1-azabicykloalkaner, farmasoytiske preparater omfattende slike, slike forbindelser for anvendelse som medikament samt slike forbindelser for behandling av sykdom.

Country Status (22)

Country Link
US (11) US6953855B2 (https=)
EP (1) EP1594869B9 (https=)
JP (3) JP4828407B2 (https=)
KR (3) KR101098490B1 (https=)
CN (2) CN101220026A (https=)
AT (1) ATE381563T1 (https=)
AU (1) AU2004215386B2 (https=)
BR (1) BRPI0407708A (https=)
CA (1) CA2514135C (https=)
CY (1) CY1107175T1 (https=)
DE (1) DE602004010787T2 (https=)
DK (1) DK1594869T3 (https=)
EA (1) EA011033B1 (https=)
ES (1) ES2300749T3 (https=)
IL (3) IL169797A (https=)
MX (1) MXPA05008926A (https=)
NO (3) NO332757B1 (https=)
NZ (3) NZ565178A (https=)
PL (3) PL378145A1 (https=)
PT (1) PT1594869E (https=)
WO (1) WO2004076449A2 (https=)
ZA (1) ZA200506515B (https=)

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DE10164139A1 (de) 2001-12-27 2003-07-10 Bayer Ag 2-Heteroarylcarbonsäureamide
GB0220581D0 (en) 2002-09-04 2002-10-09 Novartis Ag Organic Compound
MXPA05003317A (es) * 2002-09-25 2005-07-05 Memory Pharm Corp Indazoles, benzotiazoles y benzoisotiazoles asi como preparacion y usos de los mismos.
DE602004031124D1 (de) 2003-08-13 2011-03-03 Neurosearch As Neue chinuklidinderivative und deren pharmazeutische verwendung
DE602004010299T2 (de) 2003-12-22 2008-09-18 Memory Pharmaceuticals Corp. Indole, 1h-indazole, 1,2-benzisoxazole und 1,2-benzisothiazole und deren herstellung und anwendungen
SE0400708D0 (sv) * 2004-03-22 2004-03-22 Aprea Ab New compounds and use thereof
NZ550534A (en) * 2004-03-25 2009-07-31 Memory Pharm Corp Indazoles, benzothiazoles, benzoisothiazoles, benzisoxazoles, and preparation and uses thereof
WO2006001894A1 (en) * 2004-04-22 2006-01-05 Memory Pharmaceutical Corporation Indoles, 1h-indazoles, 1,2-benzisoxazoles, 1,2-benzoisothiazoles, and preparation and uses thereof
JP2007538011A (ja) * 2004-05-07 2007-12-27 メモリー・ファーマシューティカルズ・コーポレイション １ｈ−インダゾール、ベンゾチアゾール、１，２−ベンゾイソキサゾール、１，２−ベンゾイソチアゾール、およびクロモン、ならびにそれらの調製および使用
PE20060437A1 (es) 2004-06-18 2006-06-08 Novartis Ag COMPUESTOS AZA-BICICLONONANOS COMO LIGANDOS COLINERGICOS DE nAChR
GB0415746D0 (en) 2004-07-14 2004-08-18 Novartis Ag Organic compounds
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