NO329984B1 - Sammensetning omfattende krystallinsk suberoylanilid hydroksaminsyre (SAHA) samt fremgangsmate for fremstilling derav - Google Patents

Sammensetning omfattende krystallinsk suberoylanilid hydroksaminsyre (SAHA) samt fremgangsmate for fremstilling derav Download PDF

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Publication number
NO329984B1
NO329984B1 NO20044112A NO20044112A NO329984B1 NO 329984 B1 NO329984 B1 NO 329984B1 NO 20044112 A NO20044112 A NO 20044112A NO 20044112 A NO20044112 A NO 20044112A NO 329984 B1 NO329984 B1 NO 329984B1
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Prior art keywords
saha
methanol
mixture
acid
water
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NO20044112A
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English (en)
Norwegian (no)
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NO20044112L (no
Inventor
Thomas A Miller
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Merck Hdac Res Llc
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Application filed by Merck Hdac Res Llc filed Critical Merck Hdac Res Llc
Publication of NO20044112L publication Critical patent/NO20044112L/no
Publication of NO329984B1 publication Critical patent/NO329984B1/no

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    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841—Filling excipients; Inactive ingredients
    • A61K9/4866—Organic macromolecular compounds
    • A—HUMAN NECESSITIES
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    • A61K31/13—Amines
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    • A61K31/164—Amides, e.g. hydroxamic acids of a carboxylic acid with an aminoalcohol, e.g. ceramides
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    • A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
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    • A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
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    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
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    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C259/00—Compounds containing carboxyl groups, an oxygen atom of a carboxyl group being replaced by a nitrogen atom, this nitrogen atom being further bound to an oxygen atom and not being part of nitro or nitroso groups
    • C07C259/04—Compounds containing carboxyl groups, an oxygen atom of a carboxyl group being replaced by a nitrogen atom, this nitrogen atom being further bound to an oxygen atom and not being part of nitro or nitroso groups without replacement of the other oxygen atom of the carboxyl group, e.g. hydroxamic acids
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NO20044112A 2002-03-04 2004-09-28 Sammensetning omfattende krystallinsk suberoylanilid hydroksaminsyre (SAHA) samt fremgangsmate for fremstilling derav NO329984B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US36175902P 2002-03-04 2002-03-04
PCT/US2003/006451 WO2003075839A2 (en) 2002-03-04 2003-03-04 Methods of inducing terminal differentiation

Publications (2)

Publication Number Publication Date
NO20044112L NO20044112L (no) 2004-11-30
NO329984B1 true NO329984B1 (no) 2011-01-31

Family

ID=27805074

Family Applications (2)

Application Number Title Priority Date Filing Date
NO20044112A NO329984B1 (no) 2002-03-04 2004-09-28 Sammensetning omfattende krystallinsk suberoylanilid hydroksaminsyre (SAHA) samt fremgangsmate for fremstilling derav
NO20092714A NO332749B1 (no) 2002-03-04 2009-07-20 Anvendelse av suberoylanilidhydroksaminsyre for fremstilling av et oralt medikament til behandling av kreft

Family Applications After (1)

Application Number Title Priority Date Filing Date
NO20092714A NO332749B1 (no) 2002-03-04 2009-07-20 Anvendelse av suberoylanilidhydroksaminsyre for fremstilling av et oralt medikament til behandling av kreft

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US (7) US20040072735A1 (US20040072735A1-20040415-C00053.png)
EP (4) EP2082737B1 (US20040072735A1-20040415-C00053.png)
JP (4) JP4732693B2 (US20040072735A1-20040415-C00053.png)
KR (2) KR100868813B1 (US20040072735A1-20040415-C00053.png)
CN (3) CN103393630A (US20040072735A1-20040415-C00053.png)
AU (1) AU2003213684C1 (US20040072735A1-20040415-C00053.png)
BR (1) BR0308250A (US20040072735A1-20040415-C00053.png)
CA (3) CA2671976C (US20040072735A1-20040415-C00053.png)
ES (1) ES2532607T3 (US20040072735A1-20040415-C00053.png)
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IL (3) IL163909A0 (US20040072735A1-20040415-C00053.png)
MX (1) MXPA04008577A (US20040072735A1-20040415-C00053.png)
NO (2) NO329984B1 (US20040072735A1-20040415-C00053.png)
NZ (3) NZ567758A (US20040072735A1-20040415-C00053.png)
PL (1) PL372239A1 (US20040072735A1-20040415-C00053.png)
RU (3) RU2394022C2 (US20040072735A1-20040415-C00053.png)
WO (1) WO2003075839A2 (US20040072735A1-20040415-C00053.png)
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KR20050022216A (ko) * 2003-08-25 2005-03-07 윤덕구 동결건조 즉석소면 및 그 제조방법
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