NO328756B1 - Orale formuleringer for 3-(5-metoksy-1H-indol-3yl-metylen)-N-pentylkarbazimidamid og anvendelse derav - Google Patents
Orale formuleringer for 3-(5-metoksy-1H-indol-3yl-metylen)-N-pentylkarbazimidamid og anvendelse derav Download PDFInfo
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- NO328756B1 NO328756B1 NO20010863A NO20010863A NO328756B1 NO 328756 B1 NO328756 B1 NO 328756B1 NO 20010863 A NO20010863 A NO 20010863A NO 20010863 A NO20010863 A NO 20010863A NO 328756 B1 NO328756 B1 NO 328756B1
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Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
- A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
- A61K31/404—Indoles, e.g. pindolol
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- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2013—Organic compounds, e.g. phospholipids, fats
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- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2013—Organic compounds, e.g. phospholipids, fats
- A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
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- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/2027—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
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- A—HUMAN NECESSITIES
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- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
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- A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
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- A—HUMAN NECESSITIES
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- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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- A—HUMAN NECESSITIES
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- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Biophysics (AREA)
- Engineering & Computer Science (AREA)
- Molecular Biology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Indole Compounds (AREA)
- Cosmetics (AREA)
- Macromonomer-Based Addition Polymer (AREA)
- Peptides Or Proteins (AREA)
Applications Claiming Priority (5)
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| GBGB9818340.3A GB9818340D0 (en) | 1998-08-21 | 1998-08-21 | Organic compounds |
| GBGB9823477.6A GB9823477D0 (en) | 1998-10-27 | 1998-10-27 | Organic compounds |
| GBGB9910320.2A GB9910320D0 (en) | 1999-05-05 | 1999-05-05 | Organic compounds |
| GBGB9911059.5A GB9911059D0 (en) | 1999-05-12 | 1999-05-12 | Organic compounds |
| PCT/EP1999/006083 WO2000010526A2 (en) | 1998-08-21 | 1999-08-19 | New oral formulation for 5-ht4 agonists or antagonists |
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| NO20010863D0 NO20010863D0 (no) | 2001-02-20 |
| NO20010863L NO20010863L (no) | 2001-03-26 |
| NO328756B1 true NO328756B1 (no) | 2010-05-03 |
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| EP (1) | EP1104289B1 (es) |
| JP (1) | JP4048024B2 (es) |
| KR (1) | KR100529659B1 (es) |
| CN (2) | CN1165293C (es) |
| AT (1) | ATE316782T1 (es) |
| AU (4) | AU762829B2 (es) |
| BG (1) | BG65322B1 (es) |
| BR (1) | BR9913135A (es) |
| CA (1) | CA2338794C (es) |
| CZ (1) | CZ300647B6 (es) |
| DE (1) | DE69929703T2 (es) |
| DK (1) | DK1104289T3 (es) |
| EE (1) | EE05054B1 (es) |
| ES (1) | ES2257869T3 (es) |
| FR (3) | FR2782454B1 (es) |
| HK (1) | HK1038179A1 (es) |
| HR (1) | HRP20010123B1 (es) |
| HU (1) | HU228179B1 (es) |
| ID (1) | ID28510A (es) |
| IL (1) | IL141236A0 (es) |
| IS (1) | IS2369B (es) |
| IT (1) | IT1314185B1 (es) |
| NO (1) | NO328756B1 (es) |
| NZ (1) | NZ509832A (es) |
| PL (2) | PL194069B1 (es) |
| RS (1) | RS50104B (es) |
| SK (1) | SK285255B6 (es) |
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| US6743820B2 (en) | 2000-07-07 | 2004-06-01 | University Of Toledo | Methods for protection of stratified squamous epithelium against injury by noxious substances and novel agents for use therefor |
| AU2002231627A1 (en) * | 2000-11-24 | 2002-06-03 | Janssen Pharmaceutica N.V. | Use of a triple combination comprising a 5HT3 antagonist, a 5HT4 agonist and a laxative for promoting intestinal lavage |
| EP1321142A1 (en) * | 2001-12-21 | 2003-06-25 | Novartis AG | Solid pharmaceutical composition for oral administration of Tegaserod |
| EP1598074B1 (en) * | 2003-02-28 | 2019-01-02 | Chugai Seiyaku Kabushiki Kaisha | Stabilized protein-containing formulations |
| WO2004085393A1 (en) * | 2003-03-25 | 2004-10-07 | Hetero Drugs Limited | Novel crystalline forms of tegaserod maleate |
| GB0307440D0 (en) * | 2003-03-31 | 2003-05-07 | Novartis Ag | Organic compounds |
| MY137386A (en) * | 2003-07-24 | 2009-01-30 | Novartis Ag | Stable modifications of tegaserod hydrogen maleate |
| US8591974B2 (en) | 2003-11-21 | 2013-11-26 | Kraft Foods Global Brands Llc | Delivery system for two or more active components as part of an edible composition |
| US8591973B2 (en) | 2005-05-23 | 2013-11-26 | Kraft Foods Global Brands Llc | Delivery system for active components and a material having preselected hydrophobicity as part of an edible composition |
| US8597703B2 (en) | 2005-05-23 | 2013-12-03 | Kraft Foods Global Brands Llc | Delivery system for active components as part of an edible composition including a ratio of encapsulating material and active component |
| US8591968B2 (en) | 2005-05-23 | 2013-11-26 | Kraft Foods Global Brands Llc | Edible composition including a delivery system for active components |
| US20050112236A1 (en) | 2003-11-21 | 2005-05-26 | Navroz Boghani | Delivery system for active components as part of an edible composition having preselected tensile strength |
| US8591972B2 (en) | 2005-05-23 | 2013-11-26 | Kraft Foods Global Brands Llc | Delivery system for coated active components as part of an edible composition |
| US8389032B2 (en) | 2005-05-23 | 2013-03-05 | Kraft Foods Global Brands Llc | Delivery system for active components as part of an edible composition having selected particle size |
| US8216610B2 (en) | 2004-05-28 | 2012-07-10 | Imaginot Pty Ltd. | Oral paracetamol formulations |
| EP3263117A1 (en) | 2005-11-28 | 2018-01-03 | Imaginot Pty Ltd. | Oral therapeutic compound delivery system |
| EP3332772A1 (en) | 2009-10-30 | 2018-06-13 | IX Biopharma Ltd | Fast dissolving solid dosage form |
| WO2013026565A1 (de) | 2011-08-20 | 2013-02-28 | Advanced Medical Balloons | Trans-analer einlaufkatheter und verfahren zur intermittierenden auslösung einer reflexkoordinierten defäkation |
| UA118339C2 (uk) * | 2012-09-03 | 2019-01-10 | Біогайа Аб | Бактеріальний штам lactobacillus gasseri для лікування порушення моторики кишечнику (варіанти) |
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| US552398A (en) * | 1895-12-31 | Riveting-machine | ||
| JP2708803B2 (ja) * | 1987-09-02 | 1998-02-04 | 中外製薬株式会社 | 持続放出製剤 |
| DK0472502T3 (da) * | 1990-08-24 | 1995-10-09 | Spirig Ag | Fremgangsmåde til fremstilling af pellets |
| HUT64023A (en) * | 1991-03-22 | 1993-11-29 | Sandoz Ag | Process for producing aminoguanidine derivatives and pharmaceutical compositions comprising such compounds |
| US5523289A (en) * | 1991-04-15 | 1996-06-04 | Abbott Laboratories | Pharmaceutical composition |
| US20020128172A1 (en) * | 1991-12-21 | 2002-09-12 | Smithkline Beecham Plc | Use of 5-HT4 modulators for the manufacture of a medicament for the treatment of the bladder diseases |
| FR2710915B1 (fr) * | 1993-10-04 | 1995-11-24 | Synthelabo | Dérivés de pipéridine, leur préparation et leur utilisation en thérapeutique. |
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-
1999
- 1999-08-19 ES ES99942892T patent/ES2257869T3/es not_active Expired - Lifetime
- 1999-08-19 PL PL99346764A patent/PL194069B1/pl unknown
- 1999-08-19 WO PCT/EP1999/006083 patent/WO2000010526A2/en active Application Filing
- 1999-08-19 CZ CZ20010619A patent/CZ300647B6/cs not_active IP Right Cessation
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- 1999-08-19 DK DK99942892T patent/DK1104289T3/da active
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- 1999-08-19 HU HU0103431A patent/HU228179B1/hu unknown
- 1999-08-19 IT IT1999MI001826A patent/IT1314185B1/it active
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- 1999-08-19 BR BR9913135-8A patent/BR9913135A/pt not_active Application Discontinuation
- 1999-08-19 CN CNA2004100638733A patent/CN1589906A/zh active Pending
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- 1999-08-20 FR FR9910666A patent/FR2782454B1/fr not_active Expired - Lifetime
- 1999-11-26 FR FR9914897A patent/FR2784899B1/fr not_active Expired - Lifetime
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2000
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- 2000-08-21 FR FR0010748A patent/FR2799123B1/fr not_active Expired - Lifetime
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2001
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2003
- 2003-07-15 US US10/620,178 patent/US20030236183A1/en not_active Abandoned
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2006
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2007
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2009
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2011
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2013
- 2013-01-31 US US13/755,444 patent/US20130158092A1/en not_active Abandoned
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| MK1K | Patent expired |