NO325656B1 - Anti-syrefaste bakterielle midler inneholdende pyridonkarboksylsyrer som den aktive bestanddel - Google Patents
Anti-syrefaste bakterielle midler inneholdende pyridonkarboksylsyrer som den aktive bestanddel Download PDFInfo
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- NO325656B1 NO325656B1 NO20023764A NO20023764A NO325656B1 NO 325656 B1 NO325656 B1 NO 325656B1 NO 20023764 A NO20023764 A NO 20023764A NO 20023764 A NO20023764 A NO 20023764A NO 325656 B1 NO325656 B1 NO 325656B1
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Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
- A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
- A61K31/4545—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring hetero atom, e.g. pipamperone, anabasine
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/4709—Non-condensed quinolines and containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/4995—Pyrazines or piperazines forming part of bridged ring systems
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
- A61K31/5375—1,4-Oxazines, e.g. morpholine
- A61K31/5383—1,4-Oxazines, e.g. morpholine ortho- or peri-condensed with heterocyclic ring systems
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- A61P31/06—Antibacterial agents for tuberculosis
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- A61P31/08—Antibacterial agents for leprosy
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/48—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
- C07D215/54—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3
- C07D215/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3 with oxygen atoms in position 4
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/08—Bridged systems
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Epidemiology (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Pulmonology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Jellies, Jams, And Syrups (AREA)
- Medicines Containing Material From Animals Or Micro-Organisms (AREA)
- Coloring Foods And Improving Nutritive Qualities (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2000038099 | 2000-02-09 | ||
| PCT/JP2001/000861 WO2001058876A1 (en) | 2000-02-09 | 2001-02-07 | Anti-acid-fast bacterial agents containing pyridonecarboxylic acids as the active ingredient |
Publications (3)
| Publication Number | Publication Date |
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| NO20023764D0 NO20023764D0 (no) | 2002-08-08 |
| NO20023764L NO20023764L (no) | 2002-10-09 |
| NO325656B1 true NO325656B1 (no) | 2008-06-30 |
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| NO20023764A NO325656B1 (no) | 2000-02-09 | 2002-08-08 | Anti-syrefaste bakterielle midler inneholdende pyridonkarboksylsyrer som den aktive bestanddel |
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| EP (1) | EP1262477B1 (de) |
| KR (1) | KR100817425B1 (de) |
| CN (1) | CN1312131C (de) |
| AT (1) | ATE407121T1 (de) |
| AU (2) | AU2001232238B2 (de) |
| CA (1) | CA2398988C (de) |
| DE (1) | DE60135640D1 (de) |
| DK (1) | DK1262477T3 (de) |
| ES (1) | ES2312411T3 (de) |
| HK (1) | HK1048118B (de) |
| IL (2) | IL151035A0 (de) |
| MX (1) | MXPA02007667A (de) |
| NO (1) | NO325656B1 (de) |
| PT (1) | PT1262477E (de) |
| RU (2) | RU2297420C2 (de) |
| TW (1) | TWI283668B (de) |
| WO (1) | WO2001058876A1 (de) |
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| US7459005B2 (en) | 2002-11-22 | 2008-12-02 | Akzo Nobel N.V. | Chemical composition and method |
| DE10314634A1 (de) * | 2003-04-01 | 2004-10-14 | Khs Maschinen- Und Anlagenbau Ag, Patentabteilung | Spülbares Huborgan |
| SG144936A1 (en) | 2003-09-10 | 2008-08-28 | Kyorin Seiyaku Kk | 7-(4-substituted-3-cyclopropylaminomethyl-1- pyrrolidinyl)quinolonecarboxylic acid derivative |
| JP4619952B2 (ja) * | 2003-09-29 | 2011-01-26 | 第一三共株式会社 | ８−シアノキノロンカルボン酸誘導体 |
| ITMI20032259A1 (it) * | 2003-11-20 | 2005-05-21 | Chemi Spa | Nuovo polimorfo dell'acido 1-ciclopropil-7-(s,s-2,8-diazabciclo-4.3.0-non-8-il)-6-fluoro-1,4-diidro-8-metossi-4-oxo-chinolin carbossilico cloridrato e metodi per la sua preparazione |
| TW200640899A (en) * | 2005-01-21 | 2006-12-01 | Daiichi Seiyaku Co | Fluoroalkylpyrrolidine derivative |
| US8129533B2 (en) | 2005-09-28 | 2012-03-06 | Dalichi Sankyo Company, Limited | Method for production of quinolone-containing lyophilized preparation |
| JP5174365B2 (ja) * | 2007-03-23 | 2013-04-03 | 第一三共株式会社 | キノロン含有凍結乾燥製剤の製造方法 |
| RU2318513C1 (ru) * | 2007-04-10 | 2008-03-10 | Автономная некоммерческая организация "Институт молекулярной диагностики" (АНО "ИнМоДи") | Лекарственное средство на основе d-циклосерина, препарат пролонгированного действия, содержащий наночастицы, способ его получения |
| CA2688008A1 (en) * | 2007-05-24 | 2008-11-27 | Kyorin Pharmaceutical Co., Ltd. | Mutilin derivative having heterocyclic aromatic ring carboxylic acid structure in substituent at 14-position |
| EP2310388B1 (de) * | 2008-06-17 | 2015-08-05 | Institut Pasteur Korea | Pyridopyrimidinverbindungen als mittel gegen tuberkulose |
| CA2762022A1 (en) | 2009-05-15 | 2010-11-18 | Redx Pharma Limited | Redox drug derivatives |
| AU2011206761A1 (en) * | 2010-01-13 | 2012-07-12 | Institut National De La Sante Et De La Recherche Medicale (Inserm) | Anti - infective pyrido (1,2 -a) pyrimidines |
| CA2904387C (en) | 2013-03-15 | 2021-12-07 | Melinta Therapeutics, Inc. | Methods of treating infections in overweight and obese patients using antibiotics |
| CN103381169A (zh) * | 2013-07-04 | 2013-11-06 | 丁圣雨 | Chukrasone A在抗结核菌药物中的应用 |
| KR20230085439A (ko) | 2021-12-07 | 2023-06-14 | 대한민국(국립마산병원장) | 비결핵 항산균 감염 질환의 예방 또는 치료용 조성물 |
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| JPS5872589A (ja) * | 1981-10-28 | 1983-04-30 | Dai Ichi Seiyaku Co Ltd | ピリド〔１，２，３−ｄｅ〕〔１，４〕ベンゾオキサジン誘導体 |
| JPS6212760A (ja) | 1984-12-14 | 1987-01-21 | Dai Ichi Seiyaku Co Ltd | １−（２−ハロゲノシクロプロピル）キノリンカルボン酸誘導体 |
| JPS61205258A (ja) | 1985-03-08 | 1986-09-11 | Kyorin Pharmaceut Co Ltd | キノロンカルボン酸誘導体及びその製造方法 |
| US4977154A (en) | 1985-12-12 | 1990-12-11 | Warner-Lambert Company | 5-amino and 5-hydroxy-6-fluoroquinolones as antibacterial agents |
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| DE3705621C2 (de) * | 1986-02-25 | 1997-01-09 | Otsuka Pharma Co Ltd | Heterocyclisch substituierte Chinoloncarbonsäurederivate |
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| NO885426L (no) | 1987-12-11 | 1989-06-12 | Dainippon Pharmaceutical Co | Kinolinderivater, samt fremgangsmaate ved fremstilling derav. |
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| DE68907996T2 (de) | 1988-05-11 | 1994-01-05 | Abbott Lab | Verfahren zur Erhöhung der Spezifizität in kompetitiven Immuntests. |
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| DE4120646A1 (de) * | 1991-06-22 | 1992-12-24 | Bayer Ag | 7-isoindolinyl-chinolon- und naphthyridoncarbonsaeure-derivate |
| US6075024A (en) * | 1991-11-27 | 2000-06-13 | Sepracor Inc. | Methods for treating infection using optically pure (S)-lomefloxacin |
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| TW252107B (de) * | 1993-08-27 | 1995-07-21 | Hokuriku Pharmacetical Co Ltd | |
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-
2001
- 2001-02-07 AT AT01904335T patent/ATE407121T1/de active
- 2001-02-07 HK HK03100293.1A patent/HK1048118B/en not_active IP Right Cessation
- 2001-02-07 KR KR1020027010292A patent/KR100817425B1/ko not_active Expired - Fee Related
- 2001-02-07 PT PT01904335T patent/PT1262477E/pt unknown
- 2001-02-07 ES ES01904335T patent/ES2312411T3/es not_active Expired - Lifetime
- 2001-02-07 EP EP01904335A patent/EP1262477B1/de not_active Expired - Lifetime
- 2001-02-07 MX MXPA02007667A patent/MXPA02007667A/es active IP Right Grant
- 2001-02-07 WO PCT/JP2001/000861 patent/WO2001058876A1/ja not_active Ceased
- 2001-02-07 RU RU2004137055/04A patent/RU2297420C2/ru not_active IP Right Cessation
- 2001-02-07 AU AU2001232238A patent/AU2001232238B2/en not_active Ceased
- 2001-02-07 DK DK01904335T patent/DK1262477T3/da active
- 2001-02-07 CA CA2398988A patent/CA2398988C/en not_active Expired - Fee Related
- 2001-02-07 DE DE60135640T patent/DE60135640D1/de not_active Expired - Lifetime
- 2001-02-07 US US10/203,199 patent/US7176313B2/en not_active Expired - Fee Related
- 2001-02-07 IL IL15103501A patent/IL151035A0/xx unknown
- 2001-02-07 AU AU3223801A patent/AU3223801A/xx active Pending
- 2001-02-07 CN CNB018077331A patent/CN1312131C/zh not_active Expired - Fee Related
- 2001-02-07 RU RU2002121245/04A patent/RU2299205C2/ru not_active IP Right Cessation
- 2001-02-09 TW TW090102897A patent/TWI283668B/zh not_active IP Right Cessation
-
2002
- 2002-08-01 IL IL151035A patent/IL151035A/en not_active IP Right Cessation
- 2002-08-08 NO NO20023764A patent/NO325656B1/no not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| RU2002121245A (ru) | 2004-04-10 |
| CN1312131C (zh) | 2007-04-25 |
| CA2398988C (en) | 2010-06-22 |
| US20030119848A1 (en) | 2003-06-26 |
| CN1422256A (zh) | 2003-06-04 |
| IL151035A0 (en) | 2003-04-10 |
| KR20020074517A (ko) | 2002-09-30 |
| DE60135640D1 (de) | 2008-10-16 |
| PT1262477E (pt) | 2008-11-14 |
| RU2297420C2 (ru) | 2007-04-20 |
| IL151035A (en) | 2008-12-29 |
| NO20023764L (no) | 2002-10-09 |
| DK1262477T3 (da) | 2008-12-01 |
| US7176313B2 (en) | 2007-02-13 |
| AU3223801A (en) | 2001-08-20 |
| EP1262477A4 (de) | 2003-07-02 |
| WO2001058876A1 (en) | 2001-08-16 |
| HK1048118B (en) | 2009-01-09 |
| ATE407121T1 (de) | 2008-09-15 |
| KR100817425B1 (ko) | 2008-03-27 |
| ES2312411T3 (es) | 2009-03-01 |
| AU2001232238B2 (en) | 2005-03-24 |
| MXPA02007667A (es) | 2003-04-14 |
| NO20023764D0 (no) | 2002-08-08 |
| CA2398988A1 (en) | 2001-08-16 |
| RU2004137055A (ru) | 2006-05-27 |
| RU2299205C2 (ru) | 2007-05-20 |
| EP1262477A1 (de) | 2002-12-04 |
| EP1262477B1 (de) | 2008-09-03 |
| HK1048118A1 (en) | 2003-03-21 |
| TWI283668B (en) | 2007-07-11 |
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