NO322808B1 - Pyrimidin derivater, samt anvendelse derav og farmasoytisk preparat. - Google Patents

Pyrimidin derivater, samt anvendelse derav og farmasoytisk preparat. Download PDF

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Publication number
NO322808B1
NO322808B1 NO20021728A NO20021728A NO322808B1 NO 322808 B1 NO322808 B1 NO 322808B1 NO 20021728 A NO20021728 A NO 20021728A NO 20021728 A NO20021728 A NO 20021728A NO 322808 B1 NO322808 B1 NO 322808B1
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Norway
Prior art keywords
pyrrolidin
group
methyl
formula
substituent
Prior art date
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NO20021728A
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English (en)
Norwegian (no)
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NO20021728D0 (no
NO20021728L (no
Inventor
John Graham Cumming
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Astrazeneca Ab
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Publication of NO20021728D0 publication Critical patent/NO20021728D0/no
Publication of NO20021728L publication Critical patent/NO20021728L/no
Publication of NO322808B1 publication Critical patent/NO322808B1/no

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    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/32—One oxygen, sulfur or nitrogen atom
    • C07D239/42—One nitrogen atom
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
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    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
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NO20021728A 1999-10-13 2002-04-12 Pyrimidin derivater, samt anvendelse derav og farmasoytisk preparat. NO322808B1 (no)

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EP1226126A1 (en) 2002-07-31
AU7804200A (en) 2001-04-23
KR100738862B1 (ko) 2007-07-13
US6846827B1 (en) 2005-01-25
NO20021728D0 (no) 2002-04-12
CA2382605A1 (en) 2001-04-19
AU772293B2 (en) 2004-04-22
EP1226126B1 (en) 2005-01-05
NZ517572A (en) 2003-11-28
ATE286501T1 (de) 2005-01-15
IL148428A (en) 2006-12-10
MXPA02003533A (es) 2002-08-20
CN1378537A (zh) 2002-11-06
KR20020091830A (ko) 2002-12-06
IL148428A0 (en) 2002-09-12
DE60017279T2 (de) 2005-12-08
NO20021728L (no) 2002-06-12
GB9924092D0 (en) 1999-12-15
CN100415724C (zh) 2008-09-03
DE60017279D1 (en) 2005-02-10
JP2003511442A (ja) 2003-03-25
HK1045511A1 (en) 2002-11-29
HK1045511B (zh) 2005-06-03
BR0014596A (pt) 2002-06-11

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