NO20021728L - Pyrimidin derivater - Google Patents
Pyrimidin derivaterInfo
- Publication number
- NO20021728L NO20021728L NO20021728A NO20021728A NO20021728L NO 20021728 L NO20021728 L NO 20021728L NO 20021728 A NO20021728 A NO 20021728A NO 20021728 A NO20021728 A NO 20021728A NO 20021728 L NO20021728 L NO 20021728L
- Authority
- NO
- Norway
- Prior art keywords
- halogeno
- pyrimidine derivatives
- trifluoromethyl
- cyano
- hydroxy
- Prior art date
Links
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- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/32—One oxygen, sulfur or nitrogen atom
- C07D239/42—One nitrogen atom
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- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
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---|---|---|---|
GBGB9924092.1A GB9924092D0 (en) | 1999-10-13 | 1999-10-13 | Pyrimidine derivatives |
PCT/GB2000/003929 WO2001027089A1 (en) | 1999-10-13 | 2000-10-10 | Pyrimidine derivatives |
Publications (3)
Publication Number | Publication Date |
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NO20021728D0 NO20021728D0 (no) | 2002-04-12 |
NO20021728L true NO20021728L (no) | 2002-06-12 |
NO322808B1 NO322808B1 (no) | 2006-12-11 |
Family
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Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
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NO20021728A NO322808B1 (no) | 1999-10-13 | 2002-04-12 | Pyrimidin derivater, samt anvendelse derav og farmasoytisk preparat. |
Country Status (18)
Country | Link |
---|---|
US (1) | US6846827B1 (no) |
EP (1) | EP1226126B1 (no) |
JP (1) | JP2003511442A (no) |
KR (1) | KR100738862B1 (no) |
CN (1) | CN100415724C (no) |
AT (1) | ATE286501T1 (no) |
AU (1) | AU772293B2 (no) |
BR (1) | BR0014596A (no) |
CA (1) | CA2382605A1 (no) |
DE (1) | DE60017279T2 (no) |
GB (1) | GB9924092D0 (no) |
HK (1) | HK1045511B (no) |
IL (2) | IL148428A0 (no) |
MX (1) | MXPA02003533A (no) |
NO (1) | NO322808B1 (no) |
NZ (1) | NZ517572A (no) |
WO (1) | WO2001027089A1 (no) |
ZA (1) | ZA200201557B (no) |
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SK286247B6 (sk) | 1998-05-15 | 2008-06-06 | Astrazeneca Ab | Benzamidové deriváty, spôsob ich prípravy, farmaceutické prostriedky, ktoré ich obsahujú a ich použitie pri príprave liečiva na liečbu chorobných stavov sprostredkovaných cytokínmi |
KR20010099609A (ko) | 1998-08-04 | 2001-11-09 | 다비드 에 질레스 | 사이토킨의 생성 억제제로서 유용한 아미드 유도체 |
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TR200102568T2 (tr) | 1999-03-17 | 2002-05-21 | Astrazeneca Ab | Amid türevleri. |
US7008945B1 (en) | 1999-03-17 | 2006-03-07 | Astrazeneca Ab | Amide derivatives |
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GB9816837D0 (en) | 1998-08-04 | 1998-09-30 | Zeneca Ltd | Amide derivatives |
AU661533B2 (en) | 1992-01-20 | 1995-07-27 | Astrazeneca Ab | Quinazoline derivatives |
JP2000506532A (ja) * | 1996-03-13 | 2000-05-30 | スミスクライン・ビーチャム・コーポレイション | サイトカイン介在疾患の治療にて有用な新規ピリミジン化合物 |
GB9623833D0 (en) | 1996-11-16 | 1997-01-08 | Zeneca Ltd | Chemical compound |
JP2002510322A (ja) | 1997-07-03 | 2002-04-02 | デュポン ファーマシューティカルズ カンパニー | 副腎皮質刺激ホルモン放出ホルモン拮抗剤としてのアリールおよびアリールアミノ置換複素環 |
NZ502702A (en) | 1997-09-23 | 2002-10-25 | Astrazeneca Ab | Amide derivatives for the treatment of diseases mediated by TNF, IL-1, IL-6 or IL-8 |
DK0945443T3 (da) * | 1998-03-27 | 2003-06-02 | Janssen Pharmaceutica Nv | HIV-hæmmende pyrimidinderivater |
SK286247B6 (sk) | 1998-05-15 | 2008-06-06 | Astrazeneca Ab | Benzamidové deriváty, spôsob ich prípravy, farmaceutické prostriedky, ktoré ich obsahujú a ich použitie pri príprave liečiva na liečbu chorobných stavov sprostredkovaných cytokínmi |
HUP0102295A3 (en) | 1998-05-15 | 2002-11-28 | Astrazeneca Ab | Benzamide derivatives for the treatment of diseases mediated by cytokines |
KR20010099609A (ko) | 1998-08-04 | 2001-11-09 | 다비드 에 질레스 | 사이토킨의 생성 억제제로서 유용한 아미드 유도체 |
JP4497340B2 (ja) | 1998-08-27 | 2010-07-07 | 大日本住友製薬株式会社 | ピリミジン誘導体 |
AU5438499A (en) | 1998-08-29 | 2000-03-21 | Astrazeneca Ab | Pyrimidine compounds |
JP2002523497A (ja) | 1998-08-29 | 2002-07-30 | アストラゼネカ・アクチエボラーグ | ピリミジン化合物 |
WO2000018738A1 (en) | 1998-09-25 | 2000-04-06 | Astrazeneca Ab | Benzamide derivatives and their use as cytokine inhibitors |
PT1117653E (pt) | 1998-10-01 | 2003-06-30 | Astrazeneca Ab | Derivados de quinolina e quinazolina e sua utilizacao como inibidores de doencas mediadas pela citosina |
TR200102568T2 (tr) | 1999-03-17 | 2002-05-21 | Astrazeneca Ab | Amid türevleri. |
US7008945B1 (en) | 1999-03-17 | 2006-03-07 | Astrazeneca Ab | Amide derivatives |
GB9906566D0 (en) | 1999-03-23 | 1999-05-19 | Zeneca Ltd | Chemical compounds |
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1999
- 1999-10-13 GB GBGB9924092.1A patent/GB9924092D0/en not_active Ceased
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2000
- 2000-10-10 CA CA002382605A patent/CA2382605A1/en not_active Abandoned
- 2000-10-10 DE DE60017279T patent/DE60017279T2/de not_active Expired - Fee Related
- 2000-10-10 NZ NZ517572A patent/NZ517572A/en unknown
- 2000-10-10 KR KR1020027004779A patent/KR100738862B1/ko not_active IP Right Cessation
- 2000-10-10 AT AT00968084T patent/ATE286501T1/de not_active IP Right Cessation
- 2000-10-10 JP JP2001530109A patent/JP2003511442A/ja active Pending
- 2000-10-10 US US10/070,360 patent/US6846827B1/en not_active Expired - Fee Related
- 2000-10-10 EP EP00968084A patent/EP1226126B1/en not_active Expired - Lifetime
- 2000-10-10 MX MXPA02003533A patent/MXPA02003533A/es active IP Right Grant
- 2000-10-10 AU AU78042/00A patent/AU772293B2/en not_active Ceased
- 2000-10-10 BR BR0014596-3A patent/BR0014596A/pt not_active Application Discontinuation
- 2000-10-10 WO PCT/GB2000/003929 patent/WO2001027089A1/en active IP Right Grant
- 2000-10-10 CN CNB008141452A patent/CN100415724C/zh not_active Expired - Fee Related
- 2000-10-10 IL IL14842800A patent/IL148428A0/xx active IP Right Grant
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2002
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- 2002-02-27 IL IL148428A patent/IL148428A/en not_active IP Right Cessation
- 2002-04-12 NO NO20021728A patent/NO322808B1/no not_active IP Right Cessation
- 2002-09-25 HK HK02107003.8A patent/HK1045511B/zh not_active IP Right Cessation
Also Published As
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ZA200201557B (en) | 2003-07-30 |
EP1226126B1 (en) | 2005-01-05 |
BR0014596A (pt) | 2002-06-11 |
AU772293B2 (en) | 2004-04-22 |
DE60017279D1 (en) | 2005-02-10 |
EP1226126A1 (en) | 2002-07-31 |
CA2382605A1 (en) | 2001-04-19 |
US6846827B1 (en) | 2005-01-25 |
AU7804200A (en) | 2001-04-23 |
IL148428A (en) | 2006-12-10 |
IL148428A0 (en) | 2002-09-12 |
ATE286501T1 (de) | 2005-01-15 |
CN100415724C (zh) | 2008-09-03 |
CN1378537A (zh) | 2002-11-06 |
MXPA02003533A (es) | 2002-08-20 |
HK1045511A1 (en) | 2002-11-29 |
JP2003511442A (ja) | 2003-03-25 |
NO20021728D0 (no) | 2002-04-12 |
GB9924092D0 (en) | 1999-12-15 |
KR20020091830A (ko) | 2002-12-06 |
DE60017279T2 (de) | 2005-12-08 |
HK1045511B (zh) | 2005-06-03 |
WO2001027089A1 (en) | 2001-04-19 |
NO322808B1 (no) | 2006-12-11 |
KR100738862B1 (ko) | 2007-07-13 |
NZ517572A (en) | 2003-11-28 |
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