NO322313B1 - Indol-derivater, bruk av disse som medikament, farmasoytiske preparater inneholdende disse samt anvendelse av disse for fremstilling av medikamenter for behandling og/eller forebygging av sykdommer - Google Patents
Indol-derivater, bruk av disse som medikament, farmasoytiske preparater inneholdende disse samt anvendelse av disse for fremstilling av medikamenter for behandling og/eller forebygging av sykdommer Download PDFInfo
- Publication number
- NO322313B1 NO322313B1 NO20016149A NO20016149A NO322313B1 NO 322313 B1 NO322313 B1 NO 322313B1 NO 20016149 A NO20016149 A NO 20016149A NO 20016149 A NO20016149 A NO 20016149A NO 322313 B1 NO322313 B1 NO 322313B1
- Authority
- NO
- Norway
- Prior art keywords
- indol
- dichloro
- pharmaceutically acceptable
- tetramethylpiperidin
- benzamide
- Prior art date
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- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/16—Antivirals for RNA viruses for influenza or rhinoviruses
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/18—Antivirals for RNA viruses for HIV
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Physical Education & Sports Medicine (AREA)
- Virology (AREA)
- Oncology (AREA)
- Rheumatology (AREA)
- Immunology (AREA)
- Communicable Diseases (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Pulmonology (AREA)
- Dermatology (AREA)
- Hematology (AREA)
- Urology & Nephrology (AREA)
- Neurosurgery (AREA)
- Molecular Biology (AREA)
- AIDS & HIV (AREA)
- Obesity (AREA)
- Hospice & Palliative Care (AREA)
- Cardiology (AREA)
- Vascular Medicine (AREA)
- Psychiatry (AREA)
- Pain & Pain Management (AREA)
- Heart & Thoracic Surgery (AREA)
- Ophthalmology & Optometry (AREA)
- Diabetes (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB9914371.1A GB9914371D0 (en) | 1999-06-18 | 1999-06-18 | Novel compounds |
| PCT/EP2000/005672 WO2001002388A1 (en) | 1999-06-18 | 2000-06-16 | Indole derivatives and their use for the treatment of osteoporosis amongst other applications |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| NO20016149L NO20016149L (no) | 2001-12-17 |
| NO20016149D0 NO20016149D0 (no) | 2001-12-17 |
| NO322313B1 true NO322313B1 (no) | 2006-09-11 |
Family
ID=10855696
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO20016149A NO322313B1 (no) | 1999-06-18 | 2001-12-17 | Indol-derivater, bruk av disse som medikament, farmasoytiske preparater inneholdende disse samt anvendelse av disse for fremstilling av medikamenter for behandling og/eller forebygging av sykdommer |
Country Status (30)
| Country | Link |
|---|---|
| US (2) | US6787550B1 (pt) |
| EP (1) | EP1212317B1 (pt) |
| JP (1) | JP2003503490A (pt) |
| KR (1) | KR100701109B1 (pt) |
| CN (1) | CN1179960C (pt) |
| AR (1) | AR024390A1 (pt) |
| AT (1) | ATE276245T1 (pt) |
| AU (1) | AU768726B2 (pt) |
| BR (1) | BR0011708A (pt) |
| CA (1) | CA2376657A1 (pt) |
| CO (1) | CO5200757A1 (pt) |
| CZ (1) | CZ301697B6 (pt) |
| DE (1) | DE60013859T2 (pt) |
| DK (1) | DK1212317T3 (pt) |
| ES (1) | ES2226870T3 (pt) |
| GB (1) | GB9914371D0 (pt) |
| GC (1) | GC0000341A (pt) |
| HK (2) | HK1048468B (pt) |
| HU (1) | HUP0202049A3 (pt) |
| IL (2) | IL147012A0 (pt) |
| MX (1) | MXPA01013277A (pt) |
| MY (1) | MY129425A (pt) |
| NO (1) | NO322313B1 (pt) |
| NZ (1) | NZ516131A (pt) |
| PL (1) | PL352964A1 (pt) |
| PT (1) | PT1212317E (pt) |
| TR (1) | TR200103683T2 (pt) |
| TW (1) | TWI248440B (pt) |
| WO (1) | WO2001002388A1 (pt) |
| ZA (1) | ZA200200177B (pt) |
Families Citing this family (27)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2004073611A2 (en) | 2003-02-13 | 2004-09-02 | Wellstat Therapeutics Corporation | Compounds for the treatment of metabolic disorders |
| MXPA06000538A (es) * | 2003-07-15 | 2006-03-30 | Smithkline Beecham Corp | Compuestos novedosos. |
| ITMI20040875A1 (it) * | 2004-04-30 | 2004-07-30 | Ist Naz Stud Cura Dei Tumori | Derivati indolici utili per il trattamento della resistenza agli agenti antitumorali |
| EP1961757B1 (en) | 2004-09-17 | 2010-09-01 | IDENIX Pharmaceuticals, Inc. | Phosphoindoles as HIV inhibitors |
| KR20070060156A (ko) * | 2004-10-04 | 2007-06-12 | 미리어드 제네틱스, 인크. | 알츠하이머병 치료용 화합물 |
| US7833805B2 (en) * | 2004-10-21 | 2010-11-16 | University Of Cincinnati | Selectively permeable membranes on porous substrates |
| EP1911744B1 (en) | 2005-07-20 | 2013-09-04 | Masanori Somei | Tryptophan derivative and use thereof |
| ITRM20050390A1 (it) | 2005-07-22 | 2007-01-23 | Giuliani Spa | Composti e loro sali specifici per i recettori ppar ed i recettori per l'egf e loro uso in campo medico. |
| ITRM20050389A1 (it) | 2005-07-22 | 2007-01-23 | Giuliani Spa | Composti e loro sali specifici per i recettori ppar ed i recettori per l'egf e loro uso in campo medico. |
| WO2007022269A2 (en) | 2005-08-15 | 2007-02-22 | Irm Llc | Compounds and compositions as tpo mimetics |
| EP1779849A1 (en) * | 2005-10-28 | 2007-05-02 | Nikem Research S.R.L. | V-ATPase inhibitors for the treatment of septic shock |
| EP1779848A1 (en) * | 2005-10-28 | 2007-05-02 | Nikem Research S.R.L. | V-ATPase inhibitors for the treatment of inflammatory and autoimmune diseases |
| EP1976377A4 (en) | 2006-01-25 | 2010-06-23 | Wellstat Therapeutics Corp | COMPOUNDS FOR THE TREATMENT OF METABOLIC DISORDERS |
| EP1976510A4 (en) | 2006-01-25 | 2010-06-09 | Wellstat Therapeutics Corp | COMPOUNDS FOR THE TREATMENT OF METABOLISM DISORDER |
| CN101378740A (zh) | 2006-02-02 | 2009-03-04 | 维尔斯达医疗公司 | 用于治疗代谢紊乱的化合物 |
| US8222261B2 (en) * | 2006-07-13 | 2012-07-17 | GlaxoSmithKline, LLC | Chemical compounds |
| ES2488922T3 (es) | 2006-09-29 | 2014-09-01 | Idenix Pharmaceuticals, Inc. | Fosfoindoles enantiómeramente puros como inhibidores del HIV |
| UA107562C2 (uk) | 2008-12-05 | 2015-01-26 | Спосіб лікування псоріазу | |
| ES2806691T3 (es) | 2009-02-16 | 2021-02-18 | Nogra Pharma Ltd | Compuestos de alquilamido y usos de los mismos |
| US20110038852A1 (en) * | 2009-06-10 | 2011-02-17 | 3-V Biosciences, Inc. | Antivirals that target transporters, carriers, and ion channels |
| CN103201268B (zh) * | 2010-09-08 | 2015-08-12 | 百时美施贵宝公司 | 作为广谱流感抗病毒药物的新型哌嗪类似物 |
| WO2012045451A1 (en) | 2010-10-05 | 2012-04-12 | Ludwig-Maximilians-Universitaet Muenchen | Novel therapeutic treatment of progranulin-dependent diseases |
| US20120142627A1 (en) * | 2010-12-06 | 2012-06-07 | Emory University | Monophosphate prodrugs of dapd and analogs thereof |
| WO2013117744A2 (en) | 2012-02-09 | 2013-08-15 | Nogra Pharma Limited | Methods of treating fibrosis |
| EP2844242A1 (en) | 2012-04-18 | 2015-03-11 | Nogra Pharma Limited | Methods of treating lactose intolerance |
| BR112021015609A2 (pt) | 2019-02-08 | 2021-10-05 | Nogra Pharma Limited | Processo de fabricação de ácido 3-(4?-aminofenil)-2-metoxipropiônico, e análogos e intermediários do mesmo |
| CN113024432A (zh) * | 2019-12-24 | 2021-06-25 | 上海科胜药物研发有限公司 | 一种氨磺必利药典杂质的制备方法 |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| RU2124511C1 (ru) * | 1993-05-14 | 1999-01-10 | Фармасьютикал Ко., Лтд | Производные пиперазина |
| PL321263A1 (en) * | 1995-01-10 | 1997-11-24 | Smithkline Beecham Spa | Derivatives of indole useful in treating osteoporosis |
| AU3620597A (en) * | 1996-07-09 | 1998-02-02 | Smithkline Beecham Laboratoires Pharmaceutiques | Indole derivatives for the treatment of osteoporosis |
| PL191633B1 (pl) | 1997-12-24 | 2006-06-30 | Nikem Res Srl | Pochodne indolu i kompozycja farmaceutyczna zawierająca pochodną indolu |
-
1999
- 1999-06-18 GB GBGB9914371.1A patent/GB9914371D0/en not_active Ceased
-
2000
- 2000-06-16 WO PCT/EP2000/005672 patent/WO2001002388A1/en active IP Right Grant
- 2000-06-16 DK DK00943839T patent/DK1212317T3/da active
- 2000-06-16 CO CO00045017A patent/CO5200757A1/es not_active Application Discontinuation
- 2000-06-16 AR ARP000103010A patent/AR024390A1/es not_active Application Discontinuation
- 2000-06-16 US US10/018,443 patent/US6787550B1/en not_active Expired - Fee Related
- 2000-06-16 DE DE60013859T patent/DE60013859T2/de not_active Expired - Lifetime
- 2000-06-16 IL IL14701200A patent/IL147012A0/xx active IP Right Grant
- 2000-06-16 MX MXPA01013277A patent/MXPA01013277A/es active IP Right Grant
- 2000-06-16 CA CA002376657A patent/CA2376657A1/en not_active Abandoned
- 2000-06-16 NZ NZ516131A patent/NZ516131A/en unknown
- 2000-06-16 AT AT00943839T patent/ATE276245T1/de not_active IP Right Cessation
- 2000-06-16 KR KR1020017016180A patent/KR100701109B1/ko not_active IP Right Cessation
- 2000-06-16 BR BR0011708-0A patent/BR0011708A/pt not_active IP Right Cessation
- 2000-06-16 MY MYPI20002728A patent/MY129425A/en unknown
- 2000-06-16 PT PT00943839T patent/PT1212317E/pt unknown
- 2000-06-16 TR TR2001/03683T patent/TR200103683T2/xx unknown
- 2000-06-16 ES ES00943839T patent/ES2226870T3/es not_active Expired - Lifetime
- 2000-06-16 HU HU0202049A patent/HUP0202049A3/hu unknown
- 2000-06-16 CN CNB008115974A patent/CN1179960C/zh not_active Expired - Fee Related
- 2000-06-16 CZ CZ20014496A patent/CZ301697B6/cs not_active IP Right Cessation
- 2000-06-16 EP EP00943839A patent/EP1212317B1/en not_active Expired - Lifetime
- 2000-06-16 AU AU58165/00A patent/AU768726B2/en not_active Ceased
- 2000-06-16 PL PL00352964A patent/PL352964A1/xx not_active IP Right Cessation
- 2000-06-16 JP JP2001507825A patent/JP2003503490A/ja active Pending
- 2000-06-18 GC GCP2000726 patent/GC0000341A/en active
- 2000-07-06 TW TW089113348A patent/TWI248440B/zh not_active IP Right Cessation
-
2001
- 2001-12-10 IL IL147012A patent/IL147012A/en not_active IP Right Cessation
- 2001-12-17 NO NO20016149A patent/NO322313B1/no not_active IP Right Cessation
-
2002
- 2002-01-09 ZA ZA200200177A patent/ZA200200177B/en unknown
- 2002-11-19 HK HK02108380.9A patent/HK1048468B/zh not_active IP Right Cessation
-
2003
- 2003-02-20 HK HK03101303.7A patent/HK1049164A1/zh unknown
-
2004
- 2004-06-24 US US10/875,356 patent/US20040235930A1/en not_active Abandoned
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Legal Events
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| MM1K | Lapsed by not paying the annual fees |