NO314999B1 - 5-substituerte-3-oksadiazolyl-1,6-naftyridin-2(1H)-on- derivater og farmasöytisk preparat inneholdende disse - Google Patents
5-substituerte-3-oksadiazolyl-1,6-naftyridin-2(1H)-on- derivater og farmasöytisk preparat inneholdende disse Download PDFInfo
- Publication number
- NO314999B1 NO314999B1 NO20000183A NO20000183A NO314999B1 NO 314999 B1 NO314999 B1 NO 314999B1 NO 20000183 A NO20000183 A NO 20000183A NO 20000183 A NO20000183 A NO 20000183A NO 314999 B1 NO314999 B1 NO 314999B1
- Authority
- NO
- Norway
- Prior art keywords
- group
- naphthyridin
- substituted
- oxadiazol
- alkyl
- Prior art date
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- -1 5-substituted-3-oxadiazolyl-1,6-naphthyridin-2 (1H) -one Chemical class 0.000 title claims description 21
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- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
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- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Hospice & Palliative Care (AREA)
- Psychiatry (AREA)
- Anesthesiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP20717997 | 1997-07-15 | ||
| PCT/JP1998/003134 WO1999003857A1 (fr) | 1997-07-15 | 1998-07-14 | Derives de 5-substitue-3-oxadiazolyl-1,6-naphtyridin-2(1h)-one |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| NO20000183D0 NO20000183D0 (no) | 2000-01-14 |
| NO20000183L NO20000183L (no) | 2000-03-07 |
| NO314999B1 true NO314999B1 (no) | 2003-06-23 |
Family
ID=16535559
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO20000183A NO314999B1 (no) | 1997-07-15 | 2000-01-14 | 5-substituerte-3-oksadiazolyl-1,6-naftyridin-2(1H)-on- derivater og farmasöytisk preparat inneholdende disse |
Country Status (29)
| Country | Link |
|---|---|
| US (2) | US6172079B1 (pt) |
| EP (1) | EP1010699B1 (pt) |
| JP (1) | JP3390453B2 (pt) |
| KR (1) | KR100508392B1 (pt) |
| CN (1) | CN1134437C (pt) |
| AR (1) | AR013222A1 (pt) |
| AT (1) | ATE297923T1 (pt) |
| AU (1) | AU735960B2 (pt) |
| BR (1) | BR9811474B1 (pt) |
| CA (1) | CA2296427C (pt) |
| DE (1) | DE69830595T2 (pt) |
| DK (1) | DK1010699T3 (pt) |
| EE (1) | EE04372B1 (pt) |
| ES (1) | ES2244065T3 (pt) |
| HK (1) | HK1028895A1 (pt) |
| HU (1) | HUP0004671A3 (pt) |
| ID (1) | ID24047A (pt) |
| IL (2) | IL133512A0 (pt) |
| NO (1) | NO314999B1 (pt) |
| NZ (1) | NZ501814A (pt) |
| PL (1) | PL191200B1 (pt) |
| PT (1) | PT1010699E (pt) |
| RU (1) | RU2188199C2 (pt) |
| SI (1) | SI1010699T1 (pt) |
| SK (1) | SK285913B6 (pt) |
| TR (1) | TR200000103T2 (pt) |
| TW (1) | TW486479B (pt) |
| WO (1) | WO1999003857A1 (pt) |
| ZA (1) | ZA985870B (pt) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TWI298068B (en) * | 2000-06-21 | 2008-06-21 | Dainippon Sumitomo Pharma Co | Pharmaceutical composition for schizophrenia |
| TW200533371A (en) * | 2004-04-15 | 2005-10-16 | Dainippon Pharmaceutical Co | Medicament comprising a combination of an acetylcholinesterase inhibitor and a 5-substituted-3-oxadiazolyl-1,6-naphthyridin-2(1h)-one derivative |
| CN101541311B (zh) | 2006-10-25 | 2013-01-23 | 大日本住友制药株式会社 | 不易结块的颗粒制剂 |
| MX2010009207A (es) * | 2008-02-22 | 2011-03-03 | Irm Llc | Compuestos y composiciones heterociclicos como inhibidores de c-kit y pdgfr cinasa. |
| WO2010002451A1 (en) * | 2008-07-01 | 2010-01-07 | Concert Pharmaceuticals, Inc. | Naphthyridin derivatives |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4415580A (en) | 1982-08-02 | 1983-11-15 | Sterling Drug Inc. | Certain 2-(1H)-pyridinones cardiotonic compositions containing same and method of using same |
| US4650806A (en) * | 1985-01-14 | 1987-03-17 | Sterling Drug Inc. | Cardiotonic 5-(heterylcarbonyl)-pyridones |
| US4567186A (en) * | 1985-01-14 | 1986-01-28 | Sterling Drug Inc. | 5-Heteryl-1,6-naphthyridin-2(1H)-ones, cardiotonic use thereof and intermediates therefor |
| DK151890D0 (da) * | 1990-06-22 | 1990-06-22 | Ferrosan As | Heterocykliske forbindelser deres fremstilling og brug |
| AU1625192A (en) * | 1991-05-31 | 1992-12-03 | Zeneca Limited | Heterocyclic derivatives |
| AU664912B2 (en) * | 1992-09-02 | 1995-12-07 | Dainippon Pharmaceutical Co. Ltd. | Novel 3-oxadiazolyl-1,6-naphthyridine derivatives |
| JP2002241379A (ja) * | 1997-03-21 | 2002-08-28 | Dainippon Pharmaceut Co Ltd | ３−オキサジアゾリルキノキサリン誘導体 |
-
1998
- 1998-07-03 TW TW087110767A patent/TW486479B/zh not_active IP Right Cessation
- 1998-07-03 ZA ZA985870A patent/ZA985870B/xx unknown
- 1998-07-14 TR TR2000/00103T patent/TR200000103T2/xx unknown
- 1998-07-14 PT PT98931076T patent/PT1010699E/pt unknown
- 1998-07-14 WO PCT/JP1998/003134 patent/WO1999003857A1/ja active IP Right Grant
- 1998-07-14 AT AT98931076T patent/ATE297923T1/de not_active IP Right Cessation
- 1998-07-14 AU AU81294/98A patent/AU735960B2/en not_active Ceased
- 1998-07-14 JP JP50689699A patent/JP3390453B2/ja not_active Expired - Fee Related
- 1998-07-14 NZ NZ501814A patent/NZ501814A/en unknown
- 1998-07-14 EP EP98931076A patent/EP1010699B1/en not_active Expired - Lifetime
- 1998-07-14 ID IDW991683A patent/ID24047A/id unknown
- 1998-07-14 ES ES98931076T patent/ES2244065T3/es not_active Expired - Lifetime
- 1998-07-14 BR BRPI9811474-3A patent/BR9811474B1/pt not_active IP Right Cessation
- 1998-07-14 US US09/462,412 patent/US6172079B1/en not_active Expired - Fee Related
- 1998-07-14 HU HU0004671A patent/HUP0004671A3/hu unknown
- 1998-07-14 KR KR10-2000-7000388A patent/KR100508392B1/ko not_active IP Right Cessation
- 1998-07-14 RU RU2000103445/04A patent/RU2188199C2/ru not_active IP Right Cessation
- 1998-07-14 EE EEP200000029A patent/EE04372B1/xx not_active IP Right Cessation
- 1998-07-14 CN CNB988072262A patent/CN1134437C/zh not_active Expired - Fee Related
- 1998-07-14 DK DK98931076T patent/DK1010699T3/da active
- 1998-07-14 IL IL13351298A patent/IL133512A0/xx active IP Right Grant
- 1998-07-14 CA CA002296427A patent/CA2296427C/en not_active Expired - Fee Related
- 1998-07-14 SI SI9830774T patent/SI1010699T1/xx unknown
- 1998-07-14 SK SK53-2000A patent/SK285913B6/sk not_active IP Right Cessation
- 1998-07-14 PL PL338085A patent/PL191200B1/pl not_active IP Right Cessation
- 1998-07-14 DE DE69830595T patent/DE69830595T2/de not_active Expired - Fee Related
- 1998-07-15 AR ARP980103452A patent/AR013222A1/es active IP Right Grant
-
1999
- 1999-12-14 IL IL133512A patent/IL133512A/en not_active IP Right Cessation
-
2000
- 2000-01-14 NO NO20000183A patent/NO314999B1/no not_active IP Right Cessation
- 2000-09-01 US US09/654,782 patent/US6277993B1/en not_active Expired - Fee Related
- 2000-12-21 HK HK00108261A patent/HK1028895A1/xx not_active IP Right Cessation
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| MM1K | Lapsed by not paying the annual fees |