NO303013B1 - Tiadiazinonderivater, farmas÷ytiske preparater som inneholder minst ett av derivatene, samt anvendelse av derivater til fremstilling av legemidler - Google Patents

Tiadiazinonderivater, farmas÷ytiske preparater som inneholder minst ett av derivatene, samt anvendelse av derivater til fremstilling av legemidler Download PDF

Info

Publication number
NO303013B1
NO303013B1 NO924098A NO924098A NO303013B1 NO 303013 B1 NO303013 B1 NO 303013B1 NO 924098 A NO924098 A NO 924098A NO 924098 A NO924098 A NO 924098A NO 303013 B1 NO303013 B1 NO 303013B1
Authority
NO
Norway
Prior art keywords
derivatives
formula
compounds
methoxy
thiadiazin
Prior art date
Application number
NO924098A
Other languages
English (en)
Norwegian (no)
Other versions
NO924098D0 (no
NO924098L (no
Inventor
Rochus Jonas
Michael Klockow
Joachim Leibrock
Hans-Jochen Schliep
Christoph Seyfried
Michael Wolf
Original Assignee
Merck Patent Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck Patent Gmbh filed Critical Merck Patent Gmbh
Publication of NO924098D0 publication Critical patent/NO924098D0/no
Publication of NO924098L publication Critical patent/NO924098L/no
Publication of NO303013B1 publication Critical patent/NO303013B1/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D285/00Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
    • C07D285/15Six-membered rings
    • C07D285/16Thiadiazines; Hydrogenated thiadiazines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/06Antiasthmatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/26Psychostimulants, e.g. nicotine, cocaine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/04Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/08Vasodilators for multiple indications

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Biomedical Technology (AREA)
  • Cardiology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Pulmonology (AREA)
  • Psychiatry (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pain & Pain Management (AREA)
  • Hospice & Palliative Care (AREA)
  • Rheumatology (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Saccharide Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
NO924098A 1991-10-23 1992-10-22 Tiadiazinonderivater, farmas÷ytiske preparater som inneholder minst ett av derivatene, samt anvendelse av derivater til fremstilling av legemidler NO303013B1 (no)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE4134893A DE4134893A1 (de) 1991-10-23 1991-10-23 Thiadiazinone

Publications (3)

Publication Number Publication Date
NO924098D0 NO924098D0 (no) 1992-10-22
NO924098L NO924098L (no) 1993-04-26
NO303013B1 true NO303013B1 (no) 1998-05-18

Family

ID=6443196

Family Applications (1)

Application Number Title Priority Date Filing Date
NO924098A NO303013B1 (no) 1991-10-23 1992-10-22 Tiadiazinonderivater, farmas÷ytiske preparater som inneholder minst ett av derivatene, samt anvendelse av derivater til fremstilling av legemidler

Country Status (16)

Country Link
US (1) US5276027A (pl)
EP (1) EP0539806B1 (pl)
JP (1) JP3193789B2 (pl)
AT (1) ATE116644T1 (pl)
AU (1) AU653444B2 (pl)
CA (1) CA2081049A1 (pl)
CZ (1) CZ281377B6 (pl)
DE (2) DE4134893A1 (pl)
DK (1) DK0539806T3 (pl)
ES (1) ES2066540T3 (pl)
HU (1) HU214337B (pl)
MX (1) MX9206042A (pl)
NO (1) NO303013B1 (pl)
PL (1) PL171273B1 (pl)
TW (1) TW309518B (pl)
ZA (1) ZA928236B (pl)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW309520B (pl) * 1994-04-26 1997-07-01 Mitsubishi Chem Corp
DE19500558A1 (de) * 1995-01-11 1996-07-18 Merck Patent Gmbh 3-Alkoxycarbonyl-thiadiazinone
DE19502699A1 (de) * 1995-01-28 1996-08-01 Merck Patent Gmbh Arylalkyl-thiadiazinone
DE19533975A1 (de) * 1995-09-14 1997-03-20 Merck Patent Gmbh Arylalkyl-diazinone
DE10150517A1 (de) * 2001-10-12 2003-04-17 Merck Patent Gmbh Verwendung von Phosphodiesterase IV-Inhibitoren
CZ2004516A3 (cs) * 2001-10-31 2004-08-18 Merckápatentágmbh Inhibitor fosfodiesterázy typu @Ź jeho kombinace s jinými drogami a jeho použití
US7494990B2 (en) 2004-02-04 2009-02-24 Nycomed Gmbh 2-(piperidin-4-yl)-4,5-dihydro-2H-pyridazin-3-one derivatives as PDE4 inhibitors
CN101602687A (zh) * 2008-06-13 2009-12-16 上海特化医药科技有限公司 6-硝基苯乙酮类化合物、其制备方法及用途

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4495185A (en) * 1981-11-12 1985-01-22 Imperial Chemical Industries, Plc 1,2,4-Triazin-3(2H) ones
AU614965B2 (en) * 1987-06-06 1991-09-19 Merck Patent Gesellschaft Mit Beschrankter Haftung Thiadiazinones
EP0478195B1 (en) * 1990-09-21 1999-05-26 Rohm And Haas Company Dihydropyridazinones and pyridazinones as fungicides

Also Published As

Publication number Publication date
US5276027A (en) 1994-01-04
AU2723192A (en) 1993-04-29
JPH05222017A (ja) 1993-08-31
MX9206042A (es) 1993-04-01
DE59201148D1 (de) 1995-02-16
HUT67938A (en) 1995-05-29
TW309518B (pl) 1997-07-01
DK0539806T3 (da) 1995-03-13
ZA928236B (en) 1993-05-06
CZ281377B6 (cs) 1996-09-11
ES2066540T3 (es) 1995-03-01
EP0539806A1 (de) 1993-05-05
NO924098D0 (no) 1992-10-22
JP3193789B2 (ja) 2001-07-30
EP0539806B1 (de) 1995-01-04
DE4134893A1 (de) 1993-04-29
CA2081049A1 (en) 1993-04-24
PL296314A2 (en) 1993-05-04
HU9203332D0 (en) 1992-12-28
PL171273B1 (pl) 1997-03-28
NO924098L (no) 1993-04-26
ATE116644T1 (de) 1995-01-15
AU653444B2 (en) 1994-09-29
HU214337B (hu) 1998-03-02
CZ263692A3 (en) 1993-05-12

Similar Documents

Publication Publication Date Title
KR0130976B1 (ko) 3-[4-(1-치환된-4-피페라지닐)부틸]-4-티아졸리디논, 이의 제조방법 및 이를 포함하는 약제학적 조성물
KR0165131B1 (ko) 1,4-벤조티아제핀 유도체
JP5218737B2 (ja) スフィンゴシン−1−リン酸結合阻害物質
TW200813003A (en) Benzoazepin-oxy-acetic acid derivatives as PPAR-delta agonists used for the increase of HDL-C, lower LDL-C and lower cholesterol
NL8501856A (nl) Farmacologisch actieve gesubstitueerde benzamiden.
NO303013B1 (no) Tiadiazinonderivater, farmas÷ytiske preparater som inneholder minst ett av derivatene, samt anvendelse av derivater til fremstilling av legemidler
NO851950L (no) Analogifremgangsmaate for fremstilling av terapeutisk aktive benzazepinderivater.
DK168010B1 (da) Tetrahydroisoquinolinforbindelser og farmaceutisk middel indeholdende en saadan forbindelse
HUT70543A (en) Thiadiazinone derivatives, pharmaceutical compositions containing them and process for producing them
US20110269744A1 (en) Benzazepine Compound
US4683312A (en) Imidazolium hypoglycemic agents
US4089861A (en) (+)-(S)-Enantiomer of 3-{2-[4-(8-fluoro-10,11-dihydro-2-methyl-dibenzo[b,f]thiepin-10-yl)-1-piperazinyl]-ethyl}-2-oxazolidinone
US4110472A (en) Derivatives of 1-(disubstituted phenoxy)-3-amino-2-hydroxypropanes
US5401762A (en) Aminoalkyl-substituted thiazolin-2-ones, the preparation and use thereof
US3954776A (en) 1-[Methylated piperidino(and pyrrolidin-1-yl)]-3-(substituted phenoxy)-2propanols
JP4025377B2 (ja) 3−アルコキシカルボニル−チアジアジノン化合物
US3850947A (en) 3-thiazol-4'-oxy-aminopropanol cardiovascular agents
US3047571A (en) Derivatives of oxopiperidinyl phenthiazines
DK158979B (da) Aminopropanol-derivater af substituerede 2-hydroxypropiophenoner og terapeutiske praeparater med indhold deraf
HU186488B (en) Process for producing pyridine derivatives and pharmaceutival compositions containing them as active agents
EP0668276A1 (en) 2-alkoxy-5,6,7,8-tetrahydroquinoxaline derivative, process for producing the same, and use thereof
FI64353B (fi) Foerfarande foer framstaellning av e-3-(4-bromfenyl)-n-metyl-3-(3-pyridyl)-allylamin till anvaendning som laekemedel
ES2198947T3 (es) Derivados de azabicicloheptano n-substituidos, su obtencion y empleo.
JPS6245866B2 (pl)
CS268837B2 (en) Method of new 1-aryloxy-dihydrobenzothiadiazinyl alkylamino-alkanes production