NO2857404T3 - - Google Patents

Info

Publication number
NO2857404T3
NO2857404T3 NO13801320A NO13801320A NO2857404T3 NO 2857404 T3 NO2857404 T3 NO 2857404T3 NO 13801320 A NO13801320 A NO 13801320A NO 13801320 A NO13801320 A NO 13801320A NO 2857404 T3 NO2857404 T3 NO 2857404T3
Authority
NO
Norway
Application number
NO13801320A
Other languages
Norwegian (no)
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Publication of NO2857404T3 publication Critical patent/NO2857404T3/no

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/02Antineoplastic agents specific for leukemia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/50Pyridazines; Hydrogenated pyridazines
    • A61K31/5025Pyridazines; Hydrogenated pyridazines ortho- or peri-condensed with heterocyclic ring systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Hematology (AREA)
  • Oncology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
NO13801320A 2012-06-04 2013-06-03 NO2857404T3 (https=)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2012127079 2012-06-04
PCT/JP2013/065328 WO2013183578A1 (ja) 2012-06-04 2013-06-03 キナーゼ阻害剤としてのイミダゾ[1,2-b]ピリダジン誘導体

Publications (1)

Publication Number Publication Date
NO2857404T3 true NO2857404T3 (https=) 2018-01-20

Family

ID=49711970

Family Applications (1)

Application Number Title Priority Date Filing Date
NO13801320A NO2857404T3 (https=) 2012-06-04 2013-06-03

Country Status (32)

Country Link
US (2) US9187489B2 (https=)
EP (1) EP2857404B1 (https=)
JP (1) JP5814467B2 (https=)
KR (1) KR101781255B1 (https=)
CN (1) CN104520300B (https=)
AU (1) AU2013272701B2 (https=)
BR (1) BR112014029851B1 (https=)
CA (1) CA2874819C (https=)
CO (1) CO7160119A2 (https=)
CY (1) CY1119607T1 (https=)
DK (1) DK2857404T3 (https=)
ES (1) ES2648228T3 (https=)
HR (1) HRP20171724T1 (https=)
HU (1) HUE037221T2 (https=)
IL (1) IL236075A (https=)
IN (1) IN2014MN02497A (https=)
LT (1) LT2857404T (https=)
MX (1) MX357021B (https=)
MY (1) MY170326A (https=)
NO (1) NO2857404T3 (https=)
NZ (1) NZ702574A (https=)
PH (1) PH12014502721A1 (https=)
PL (1) PL2857404T3 (https=)
PT (1) PT2857404T (https=)
RS (1) RS56625B1 (https=)
RU (1) RU2635917C2 (https=)
SG (1) SG11201408052WA (https=)
SI (1) SI2857404T1 (https=)
SM (1) SMT201700539T1 (https=)
TW (1) TWI585088B (https=)
WO (1) WO2013183578A1 (https=)
ZA (1) ZA201408843B (https=)

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CN113354649B (zh) 2014-11-16 2024-12-10 阵列生物制药公司 一种新的晶型
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TWI752098B (zh) 2016-10-10 2022-01-11 美商亞雷生物製藥股份有限公司 作為ret激酶抑制劑之經取代吡唑并[1,5-a]吡啶化合物
TWI704148B (zh) 2016-10-10 2020-09-11 美商亞雷生物製藥股份有限公司 作為ret激酶抑制劑之經取代吡唑并[1,5-a]吡啶化合物
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WO2019084285A1 (en) 2017-10-26 2019-05-02 Qian Zhao FORMULATIONS OF A MACROCYCLIC TRK KINASE INHIBITOR
CN109748902B (zh) * 2017-11-02 2020-11-06 杭州科巢生物科技有限公司 一种盐酸安罗替尼的制备方法
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CN108129288B (zh) * 2017-12-27 2021-01-22 上海毕得医药科技股份有限公司 一种反式-3-羟基环丁基甲酸的合成方法
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CN112996794A (zh) 2018-09-10 2021-06-18 阿雷生物药品公司 作为ret激酶抑制剂的稠合杂环化合物
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Also Published As

Publication number Publication date
CN104520300B (zh) 2016-12-21
SMT201700539T1 (it) 2018-01-11
DK2857404T3 (en) 2017-12-04
SG11201408052WA (en) 2015-01-29
MY170326A (en) 2019-07-17
RS56625B1 (sr) 2018-03-30
RU2014153627A (ru) 2016-08-10
JPWO2013183578A1 (ja) 2016-01-28
ES2648228T3 (es) 2017-12-29
HRP20171724T1 (hr) 2018-01-12
MX357021B (es) 2018-06-25
US20160046639A1 (en) 2016-02-18
PT2857404T (pt) 2017-11-23
LT2857404T (lt) 2017-11-10
EP2857404A1 (en) 2015-04-08
IN2014MN02497A (https=) 2015-07-17
IL236075A (en) 2017-10-31
CN104520300A (zh) 2015-04-15
HK1207374A1 (en) 2016-01-29
AU2013272701B2 (en) 2017-12-21
US9751887B2 (en) 2017-09-05
NZ702574A (en) 2016-07-29
SI2857404T1 (sl) 2017-11-30
BR112014029851B1 (pt) 2023-01-03
CA2874819A1 (en) 2013-12-12
CO7160119A2 (es) 2015-01-15
KR20150014942A (ko) 2015-02-09
JP5814467B2 (ja) 2015-11-17
AU2013272701A1 (en) 2015-01-15
IL236075A0 (en) 2015-02-01
WO2013183578A1 (ja) 2013-12-12
PL2857404T3 (pl) 2018-04-30
HUE037221T2 (hu) 2018-08-28
US9187489B2 (en) 2015-11-17
PH12014502721B1 (en) 2015-02-02
BR112014029851A2 (pt) 2017-06-27
MX2014014803A (es) 2015-02-12
RU2635917C2 (ru) 2017-11-17
KR101781255B1 (ko) 2017-09-22
ZA201408843B (en) 2016-01-27
CA2874819C (en) 2017-06-20
TWI585088B (zh) 2017-06-01
PH12014502721A1 (en) 2015-02-02
AU2013272701A2 (en) 2015-01-22
CY1119607T1 (el) 2018-04-04
EP2857404B1 (en) 2017-08-23
EP2857404A4 (en) 2016-01-20
TW201400486A (zh) 2014-01-01
US20150051190A1 (en) 2015-02-19

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