PL2857404T3 - POCHODNE IMIDAZO[1,2-b]PIRYDAZYNY JAKO INHIBITORY KINAZY - Google Patents

POCHODNE IMIDAZO[1,2-b]PIRYDAZYNY JAKO INHIBITORY KINAZY

Info

Publication number
PL2857404T3
PL2857404T3 PL13801320T PL13801320T PL2857404T3 PL 2857404 T3 PL2857404 T3 PL 2857404T3 PL 13801320 T PL13801320 T PL 13801320T PL 13801320 T PL13801320 T PL 13801320T PL 2857404 T3 PL2857404 T3 PL 2857404T3
Authority
PL
Poland
Prior art keywords
imidazo
kinase inhibitors
pyridazine derivatives
pyridazine
derivatives
Prior art date
Application number
PL13801320T
Other languages
English (en)
Inventor
Yasuyuki Takeda
Kenji Yoshikawa
Yoshiko Kagoshima
Yuko Yamamoto
Ryoichi Tanaka
Yuichi Tominaga
Masaki Kiga
Yoshito HAMADA
Original Assignee
Daiichi Sankyo Co., Ltd.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Daiichi Sankyo Co., Ltd. filed Critical Daiichi Sankyo Co., Ltd.
Publication of PL2857404T3 publication Critical patent/PL2857404T3/pl

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/50—Pyridazines; Hydrogenated pyridazines
    • A61K31/5025—Pyridazines; Hydrogenated pyridazines ortho- or peri-condensed with heterocyclic ring systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Hematology (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
PL13801320T 2012-06-04 2013-06-03 POCHODNE IMIDAZO[1,2-b]PIRYDAZYNY JAKO INHIBITORY KINAZY PL2857404T3 (pl)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP2012127079 2012-06-04
EP13801320.6A EP2857404B1 (en) 2012-06-04 2013-06-03 IMIDAZO[1,2-b]PYRIDAZINE DERIVATIVES AS KINASE INHIBITORS
PCT/JP2013/065328 WO2013183578A1 (ja) 2012-06-04 2013-06-03 キナーゼ阻害剤としてのイミダゾ[１，２－ｂ]ピリダジン誘導体

Publications (1)

Publication Number Publication Date
PL2857404T3 true PL2857404T3 (pl) 2018-04-30

Family

ID=49711970

Family Applications (1)

Application Number Title Priority Date Filing Date
PL13801320T PL2857404T3 (pl) 2012-06-04 2013-06-03 POCHODNE IMIDAZO[1,2-b]PIRYDAZYNY JAKO INHIBITORY KINAZY

Country Status (32)

Country Link
US (2) US9187489B2 (pl)
EP (1) EP2857404B1 (pl)
JP (1) JP5814467B2 (pl)
KR (1) KR101781255B1 (pl)
CN (1) CN104520300B (pl)
AU (1) AU2013272701B2 (pl)
BR (1) BR112014029851B1 (pl)
CA (1) CA2874819C (pl)
CO (1) CO7160119A2 (pl)
CY (1) CY1119607T1 (pl)
DK (1) DK2857404T3 (pl)
ES (1) ES2648228T3 (pl)
HR (1) HRP20171724T1 (pl)
HU (1) HUE037221T2 (pl)
IL (1) IL236075A (pl)
IN (1) IN2014MN02497A (pl)
LT (1) LT2857404T (pl)
MX (1) MX357021B (pl)
MY (1) MY170326A (pl)
NO (1) NO2857404T3 (pl)
NZ (1) NZ702574A (pl)
PH (1) PH12014502721A1 (pl)
PL (1) PL2857404T3 (pl)
PT (1) PT2857404T (pl)
RS (1) RS56625B1 (pl)
RU (1) RU2635917C2 (pl)
SG (1) SG11201408052WA (pl)
SI (1) SI2857404T1 (pl)
SM (1) SMT201700539T1 (pl)
TW (1) TWI585088B (pl)
WO (1) WO2013183578A1 (pl)
ZA (1) ZA201408843B (pl)

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Also Published As

Publication number Publication date
ES2648228T3 (es) 2017-12-29
CA2874819C (en) 2017-06-20
DK2857404T3 (en) 2017-12-04
MY170326A (en) 2019-07-17
KR20150014942A (ko) 2015-02-09
PH12014502721B1 (en) 2015-02-02
SI2857404T1 (sl) 2017-11-30
IL236075A0 (en) 2015-02-01
HUE037221T2 (hu) 2018-08-28
TWI585088B (zh) 2017-06-01
BR112014029851A2 (pt) 2017-06-27
CN104520300A (zh) 2015-04-15
BR112014029851B1 (pt) 2023-01-03
CY1119607T1 (el) 2018-04-04
CA2874819A1 (en) 2013-12-12
MX357021B (es) 2018-06-25
EP2857404A1 (en) 2015-04-08
IL236075A (en) 2017-10-31
NO2857404T3 (pl) 2018-01-20
US20150051190A1 (en) 2015-02-19
SG11201408052WA (en) 2015-01-29
EP2857404A4 (en) 2016-01-20
SMT201700539T1 (it) 2018-01-11
EP2857404B1 (en) 2017-08-23
US20160046639A1 (en) 2016-02-18
CN104520300B (zh) 2016-12-21
JP5814467B2 (ja) 2015-11-17
CO7160119A2 (es) 2015-01-15
PT2857404T (pt) 2017-11-23
JPWO2013183578A1 (ja) 2016-01-28
HRP20171724T1 (hr) 2018-01-12
US9187489B2 (en) 2015-11-17
AU2013272701A1 (en) 2015-01-15
US9751887B2 (en) 2017-09-05
PH12014502721A1 (en) 2015-02-02
RS56625B1 (sr) 2018-03-30
TW201400486A (zh) 2014-01-01
AU2013272701A2 (en) 2015-01-22
ZA201408843B (en) 2016-01-27
RU2014153627A (ru) 2016-08-10
NZ702574A (en) 2016-07-29
MX2014014803A (es) 2015-02-12
HK1207374A1 (en) 2016-01-29
WO2013183578A1 (ja) 2013-12-12
AU2013272701B2 (en) 2017-12-21
RU2635917C2 (ru) 2017-11-17
LT2857404T (lt) 2017-11-10
KR101781255B1 (ko) 2017-09-22
IN2014MN02497A (pl) 2015-07-17

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