NO20091058L - Sulfonamidforbindelse eller salt derav - Google Patents

Sulfonamidforbindelse eller salt derav

Info

Publication number
NO20091058L
NO20091058L NO20091058A NO20091058A NO20091058L NO 20091058 L NO20091058 L NO 20091058L NO 20091058 A NO20091058 A NO 20091058A NO 20091058 A NO20091058 A NO 20091058A NO 20091058 L NO20091058 L NO 20091058L
Authority
NO
Norway
Prior art keywords
salt
sulfonamide compound
receptor
compound
sulfonamide
Prior art date
Application number
NO20091058A
Other languages
English (en)
Norwegian (no)
Inventor
Issei Tsukamoto
Susumu Toda
Hideki Kubota
Yuta Fukuda
Ryutaro Wakayama
Kazuki Ono
Toru Watanabe
Hidenori Azami
Original Assignee
Astellas Pharma Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astellas Pharma Inc filed Critical Astellas Pharma Inc
Publication of NO20091058L publication Critical patent/NO20091058L/no

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    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C311/00—Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
    • C07C311/22—Sulfonamides, the carbon skeleton of the acid part being further substituted by singly-bound oxygen atoms
    • C07C311/29—Sulfonamides, the carbon skeleton of the acid part being further substituted by singly-bound oxygen atoms having the sulfur atom of at least one of the sulfonamide groups bound to a carbon atom of a six-membered aromatic ring
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    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/16—Amides, e.g. hydroxamic acids
    • A61K31/18—Sulfonamides
    • A—HUMAN NECESSITIES
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    • A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19—Carboxylic acids, e.g. valproic acid
    • A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
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    • A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
    • A61K31/197—Carboxylic acids, e.g. valproic acid having an amino group the amino and the carboxyl groups being attached to the same acyclic carbon chain, e.g. gamma-aminobutyric acid [GABA], beta-alanine, epsilon-aminocaproic acid or pantothenic acid
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    • A61K31/197—Carboxylic acids, e.g. valproic acid having an amino group the amino and the carboxyl groups being attached to the same acyclic carbon chain, e.g. gamma-aminobutyric acid [GABA], beta-alanine, epsilon-aminocaproic acid or pantothenic acid
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    • A61K31/4015—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil having oxo groups directly attached to the heterocyclic ring, e.g. piracetam, ethosuximide
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EP2563761A1 (en) 2010-04-29 2013-03-06 The U.S.A. As Represented By The Secretary, Department Of Health And Human Services Activators of human pyruvate kinase
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RU2015113746A (ru) 2012-09-27 2016-11-20 Ф. Хоффманн-Ля Рош Аг Замещенные сульфонамиды
CN104902894A (zh) * 2012-10-26 2015-09-09 默沙东公司 具有电压门控性钠通道选择性活性的苯并噁唑啉酮化合物
EP2774919A1 (en) * 2013-03-06 2014-09-10 Pharmeste S.R.L. In Liquidazione Novel sulfonamide TRPA1 receptor antagonists
CN109843855B (zh) * 2016-11-08 2021-06-25 正大天晴药业集团股份有限公司 作为cccDNA抑制剂的磺酰胺类化合物
WO2020199683A1 (zh) * 2019-04-04 2020-10-08 上海海雁医药科技有限公司 氮杂环取代的磺酰基苯甲酰胺衍生物、其制法与医药上的用途
CN110698420B (zh) * 2019-10-25 2022-10-14 上海阿拉丁生化科技股份有限公司 一种2-噁唑甲胺杂环化合物的制备方法

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US7973078B2 (en) 2011-07-05
IL196656A0 (en) 2009-11-18
TW200817319A (en) 2008-04-16
KR101352217B1 (ko) 2014-01-15
KR20090048401A (ko) 2009-05-13
ES2467097T3 (es) 2014-06-11
AU2007282465C1 (en) 2012-05-10
US20090312328A1 (en) 2009-12-17
WO2008018544A1 (fr) 2008-02-14
CA2660424A1 (en) 2008-02-14
RU2425029C2 (ru) 2011-07-27
EP2050446B1 (en) 2014-05-07
JP5029970B2 (ja) 2012-09-19
MX2009001512A (es) 2009-02-18
AU2007282465B2 (en) 2011-12-01
PL2050446T3 (pl) 2014-10-31
CN101500554B (zh) 2012-06-27
RU2009108275A (ru) 2010-09-20
JPWO2008018544A1 (ja) 2010-01-07
PT2050446E (pt) 2014-07-18
IL196656A (en) 2013-11-28
ZA200900549B (en) 2010-03-31
EP2050446A1 (en) 2009-04-22
AU2007282465A1 (en) 2008-02-14
CN101500554A (zh) 2009-08-05
BRPI0716491A2 (pt) 2014-03-11
EP2050446A4 (en) 2011-02-16

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