NO20083462L - Nye tiofenderivater som S1P1/EDG1-reseptoragonister - Google Patents
Nye tiofenderivater som S1P1/EDG1-reseptoragonisterInfo
- Publication number
- NO20083462L NO20083462L NO20083462A NO20083462A NO20083462L NO 20083462 L NO20083462 L NO 20083462L NO 20083462 A NO20083462 A NO 20083462A NO 20083462 A NO20083462 A NO 20083462A NO 20083462 L NO20083462 L NO 20083462L
- Authority
- NO
- Norway
- Prior art keywords
- thiophene derivatives
- receptor agonists
- edg1 receptor
- new thiophene
- new
- Prior art date
Links
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/06—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
- C07D333/22—Radicals substituted by doubly bound hetero atoms, or by two hetero atoms other than halogen singly bound to the same carbon atom
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4245—Oxadiazoles
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Diabetes (AREA)
- Immunology (AREA)
- Dermatology (AREA)
- Physical Education & Sports Medicine (AREA)
- Endocrinology (AREA)
- Hematology (AREA)
- Pulmonology (AREA)
- Neurology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Cardiology (AREA)
- Ophthalmology & Optometry (AREA)
- Oncology (AREA)
- Heart & Thoracic Surgery (AREA)
- Rheumatology (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Urology & Nephrology (AREA)
- Communicable Diseases (AREA)
- Obesity (AREA)
- Hospice & Palliative Care (AREA)
- Otolaryngology (AREA)
- Pain & Pain Management (AREA)
- Psychology (AREA)
- Emergency Medicine (AREA)
- Toxicology (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IB2006050103 | 2006-01-11 | ||
PCT/IB2007/050070 WO2007080542A1 (en) | 2006-01-11 | 2007-01-10 | Novel thiophene derivatives as s1p1/edg1 receptor agonists |
Publications (1)
Publication Number | Publication Date |
---|---|
NO20083462L true NO20083462L (no) | 2008-10-09 |
Family
ID=37908151
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO20083462A NO20083462L (no) | 2006-01-11 | 2008-08-08 | Nye tiofenderivater som S1P1/EDG1-reseptoragonister |
Country Status (17)
Country | Link |
---|---|
US (1) | US8003800B2 (ja) |
EP (1) | EP1976512B1 (ja) |
JP (1) | JP5114430B2 (ja) |
KR (1) | KR101382710B1 (ja) |
CN (1) | CN101370496B (ja) |
AR (1) | AR058956A1 (ja) |
AU (1) | AU2007204121B2 (ja) |
BR (1) | BRPI0706476A2 (ja) |
CA (1) | CA2635047C (ja) |
ES (1) | ES2553345T3 (ja) |
IL (1) | IL192657A (ja) |
MY (1) | MY154909A (ja) |
NO (1) | NO20083462L (ja) |
NZ (1) | NZ570258A (ja) |
RU (1) | RU2437877C2 (ja) |
TW (1) | TWI404706B (ja) |
WO (1) | WO2007080542A1 (ja) |
Families Citing this family (39)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JP5063615B2 (ja) | 2006-01-24 | 2012-10-31 | アクテリオン ファーマシューティカルズ リミテッド | 新規ピリジン誘導体 |
TWI408139B (zh) * | 2006-09-07 | 2013-09-11 | Actelion Pharmaceuticals Ltd | 新穎噻吩衍生物 |
SI2069336T1 (sl) * | 2006-09-07 | 2013-03-29 | Actelion Pharmaceuticals Ltd. | Derivati piridin-4-ila kot imunomodulirna sredstva |
MX2009002234A (es) * | 2006-09-08 | 2009-03-16 | Actelion Pharmaceuticals Ltd | Derivados de piridin-3-il como agentes inmunomoduladores. |
NZ577111A (en) | 2006-12-15 | 2012-05-25 | Abbott Lab | Novel oxadiazole compounds |
CN101627034B (zh) * | 2007-03-16 | 2013-05-15 | 埃科特莱茵药品有限公司 | 氨基-吡啶衍生物作为s1p1/edg1受体激动剂 |
MX2009012587A (es) * | 2007-05-22 | 2010-05-14 | Wyeth Llc | Proceso mejorado para la elaboracion de hidrazidas. |
JP5451614B2 (ja) * | 2007-08-17 | 2014-03-26 | アクテリオン ファーマシューティカルズ リミテッド | S1p1/edg1受容体調節剤としてのピリジン誘導体 |
BRPI0817597A2 (pt) * | 2007-10-04 | 2015-04-07 | Merck Serono Sa | Compostos de diarila de oxadiazol, processo para sua preparação, composições farmacêuticas e kit compreendendo os mesmos, bem como seus usos |
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IL192657A0 (en) | 2009-02-11 |
TW200804298A (en) | 2008-01-16 |
CA2635047C (en) | 2014-07-29 |
NZ570258A (en) | 2011-07-29 |
ES2553345T3 (es) | 2015-12-07 |
AU2007204121B2 (en) | 2012-06-07 |
JP2009523165A (ja) | 2009-06-18 |
WO2007080542A1 (en) | 2007-07-19 |
JP5114430B2 (ja) | 2013-01-09 |
EP1976512A1 (en) | 2008-10-08 |
CA2635047A1 (en) | 2007-07-19 |
US20100240717A1 (en) | 2010-09-23 |
KR101382710B1 (ko) | 2014-04-08 |
MY154909A (en) | 2015-08-28 |
TWI404706B (zh) | 2013-08-11 |
IL192657A (en) | 2015-09-24 |
AU2007204121A1 (en) | 2007-07-19 |
AR058956A1 (es) | 2008-03-05 |
CN101370496B (zh) | 2012-07-04 |
RU2437877C2 (ru) | 2011-12-27 |
US8003800B2 (en) | 2011-08-23 |
EP1976512B1 (en) | 2015-09-30 |
BRPI0706476A2 (pt) | 2011-04-05 |
RU2008132802A (ru) | 2010-02-20 |
CN101370496A (zh) | 2009-02-18 |
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