NO20070752L - Hydrater og polymorfer av 4-(((7R)-8-cyklopentyl-7-etyl-5,6,7,8-tetrahydro-5-metyl-4-6-okso-2-piperidinyl)-3-metoksy-N-(1-metyl-4-piperidinyl) benzamid, fremgangsmåter for fremstilling derav og anvendelse som medikamenter - Google Patents

Hydrater og polymorfer av 4-(((7R)-8-cyklopentyl-7-etyl-5,6,7,8-tetrahydro-5-metyl-4-6-okso-2-piperidinyl)-3-metoksy-N-(1-metyl-4-piperidinyl) benzamid, fremgangsmåter for fremstilling derav og anvendelse som medikamenter

Info

Publication number
NO20070752L
NO20070752L NO20070752A NO20070752A NO20070752L NO 20070752 L NO20070752 L NO 20070752L NO 20070752 A NO20070752 A NO 20070752A NO 20070752 A NO20070752 A NO 20070752A NO 20070752 L NO20070752 L NO 20070752L
Authority
NO
Norway
Prior art keywords
piperidinyl
methyl
polymorphs
benzamide
hydrates
Prior art date
Application number
NO20070752A
Other languages
English (en)
Norwegian (no)
Inventor
Günter Linz
Rolf Schmid
Rolf Ulrich Wilhelm Herter
Werner Rall
Matthias Hoffmann
Peter Sieger
Gerd F Kraemer
Original Assignee
Boehringer Ingelheim Int
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=35311878&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO20070752(L) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Boehringer Ingelheim Int filed Critical Boehringer Ingelheim Int
Publication of NO20070752L publication Critical patent/NO20070752L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/56—Nitrogen atoms
    • C07D211/58—Nitrogen atoms attached in position 4
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D475/00—Heterocyclic compounds containing pteridine ring systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Immunology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
NO20070752A 2004-08-14 2007-02-08 Hydrater og polymorfer av 4-(((7R)-8-cyklopentyl-7-etyl-5,6,7,8-tetrahydro-5-metyl-4-6-okso-2-piperidinyl)-3-metoksy-N-(1-metyl-4-piperidinyl) benzamid, fremgangsmåter for fremstilling derav og anvendelse som medikamenter NO20070752L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP04019366 2004-08-14
PCT/EP2005/008736 WO2006018222A1 (de) 2004-08-14 2005-08-11 Hydrate und polymorphe des 4-[[(7r)-8-cyclopentyl-7-ethyl-5,6,7,8-tetrahydro-5-methyl-4-6-oxo-2-piperidinyl]amino]-3-methoxy-n-(1-methyl-4-piperidinyl)-benzamid, verfahren zu deren herstellung und deren verwendung als arzneimittel

Publications (1)

Publication Number Publication Date
NO20070752L true NO20070752L (no) 2007-05-10

Family

ID=35311878

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20070752A NO20070752L (no) 2004-08-14 2007-02-08 Hydrater og polymorfer av 4-(((7R)-8-cyklopentyl-7-etyl-5,6,7,8-tetrahydro-5-metyl-4-6-okso-2-piperidinyl)-3-metoksy-N-(1-metyl-4-piperidinyl) benzamid, fremgangsmåter for fremstilling derav og anvendelse som medikamenter

Country Status (19)

Country Link
US (3) US7728134B2 (enExample)
EP (1) EP1778691A1 (enExample)
JP (1) JP2008509953A (enExample)
KR (1) KR101221864B1 (enExample)
CN (1) CN101006090A (enExample)
AR (1) AR052404A1 (enExample)
AU (1) AU2005274340B2 (enExample)
BR (1) BRPI0514351A2 (enExample)
CA (1) CA2578098A1 (enExample)
EA (1) EA011407B1 (enExample)
EC (1) ECSP077249A (enExample)
IL (1) IL181302A0 (enExample)
MX (1) MX2007001854A (enExample)
NO (1) NO20070752L (enExample)
NZ (1) NZ553649A (enExample)
PE (1) PE20060424A1 (enExample)
TW (1) TWI370131B (enExample)
UA (1) UA87865C2 (enExample)
WO (1) WO2006018222A1 (enExample)

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EP3098223A1 (en) 2007-08-03 2016-11-30 Boehringer Ingelheim International GmbH Crystalline form of a dihydropteridione derivative

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Publication number Publication date
US20090318457A1 (en) 2009-12-24
JP2008509953A (ja) 2008-04-03
CA2578098A1 (en) 2006-02-23
US8202867B2 (en) 2012-06-19
AR052404A1 (es) 2007-03-21
EP1778691A1 (de) 2007-05-02
EA011407B1 (ru) 2009-02-27
US20060035902A1 (en) 2006-02-16
KR20070050967A (ko) 2007-05-16
MX2007001854A (es) 2007-03-28
WO2006018222A8 (de) 2006-06-15
BRPI0514351A2 (pt) 2012-10-30
KR101221864B1 (ko) 2013-01-14
PE20060424A1 (es) 2006-06-09
AU2005274340A1 (en) 2006-02-23
US20090298840A1 (en) 2009-12-03
AU2005274340B2 (en) 2012-04-05
IL181302A0 (en) 2007-07-04
US7728134B2 (en) 2010-06-01
US8034816B2 (en) 2011-10-11
CN101006090A (zh) 2007-07-25
WO2006018222A1 (de) 2006-02-23
UA87865C2 (en) 2009-08-25
ECSP077249A (es) 2007-03-29
TWI370131B (en) 2012-08-11
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NZ553649A (en) 2010-11-26
EA200700387A1 (ru) 2007-08-31

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