NO20061700L - 2-pyridonderivater som neutrofil elastase inhibitorer og deres anvendelse - Google Patents

2-pyridonderivater som neutrofil elastase inhibitorer og deres anvendelse

Info

Publication number
NO20061700L
NO20061700L NO20061700A NO20061700A NO20061700L NO 20061700 L NO20061700 L NO 20061700L NO 20061700 A NO20061700 A NO 20061700A NO 20061700 A NO20061700 A NO 20061700A NO 20061700 L NO20061700 L NO 20061700L
Authority
NO
Norway
Prior art keywords
neutrophil elastase
elastase inhibitors
pyridone derivatives
inhibitors
pyridone
Prior art date
Application number
NO20061700A
Other languages
English (en)
Norwegian (no)
Inventor
Peter Hansen
Hans Lonn
Karolina Lawitz
Antonios Nikitidis
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=29212489&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO20061700(L) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of NO20061700L publication Critical patent/NO20061700L/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D213/00Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/78Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D213/81Amides; Imides
    • C07D213/82Amides; Imides in position 3
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D213/00Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/78Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D213/84Nitriles
    • C07D213/85Nitriles in position 3
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
NO20061700A 2003-09-18 2006-04-18 2-pyridonderivater som neutrofil elastase inhibitorer og deres anvendelse NO20061700L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
SE0302487A SE0302487D0 (sv) 2003-09-18 2003-09-18 Novel compounds
PCT/SE2004/001336 WO2005026124A1 (en) 2003-09-18 2004-09-15 2-pyridone derivatives as netrophil elastase inhibitors and their use

Publications (1)

Publication Number Publication Date
NO20061700L true NO20061700L (no) 2006-04-18

Family

ID=29212489

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20061700A NO20061700L (no) 2003-09-18 2006-04-18 2-pyridonderivater som neutrofil elastase inhibitorer og deres anvendelse

Country Status (25)

Country Link
US (1) US20070043036A1 (ref)
EP (1) EP1663974B1 (ref)
JP (1) JP2007505902A (ref)
KR (1) KR20060096995A (ref)
CN (1) CN100439339C (ref)
AR (1) AR046083A1 (ref)
AT (1) ATE420861T1 (ref)
AU (1) AU2004272485B2 (ref)
BR (1) BRPI0414570A (ref)
CA (1) CA2538410A1 (ref)
CO (1) CO5670357A2 (ref)
DE (1) DE602004019110D1 (ref)
ES (1) ES2319300T3 (ref)
IL (1) IL173986A0 (ref)
IS (1) IS8394A (ref)
MX (1) MXPA06002723A (ref)
NO (1) NO20061700L (ref)
RU (1) RU2348617C2 (ref)
SA (1) SA04250300B1 (ref)
SE (1) SE0302487D0 (ref)
TW (1) TW200526579A (ref)
UA (1) UA84878C2 (ref)
UY (1) UY28513A1 (ref)
WO (1) WO2005026124A1 (ref)
ZA (1) ZA200602262B (ref)

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Also Published As

Publication number Publication date
AR046083A1 (es) 2005-11-23
BRPI0414570A (pt) 2006-11-07
UA84878C2 (ru) 2008-12-10
CO5670357A2 (es) 2006-08-31
ATE420861T1 (de) 2009-01-15
EP1663974A1 (en) 2006-06-07
DE602004019110D1 (de) 2009-03-05
SA04250300B1 (ar) 2008-09-07
UY28513A1 (es) 2005-04-29
AU2004272485A1 (en) 2005-03-24
KR20060096995A (ko) 2006-09-13
JP2007505902A (ja) 2007-03-15
TW200526579A (en) 2005-08-16
SE0302487D0 (sv) 2003-09-18
CN1856467A (zh) 2006-11-01
RU2348617C2 (ru) 2009-03-10
IS8394A (is) 2006-03-31
AU2004272485B2 (en) 2008-03-13
WO2005026124A1 (en) 2005-03-24
CN100439339C (zh) 2008-12-03
ES2319300T3 (es) 2009-05-06
HK1089167A1 (en) 2006-11-24
CA2538410A1 (en) 2005-03-24
US20070043036A1 (en) 2007-02-22
IL173986A0 (en) 2006-07-05
ZA200602262B (en) 2007-07-25
EP1663974B1 (en) 2009-01-14
RU2006112427A (ru) 2007-11-10
MXPA06002723A (es) 2006-06-06

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