NO20062591L - Difenylazetidinonderivater med kolesterolabsorpsjonsinhiberende aktivitet - Google Patents
Difenylazetidinonderivater med kolesterolabsorpsjonsinhiberende aktivitetInfo
- Publication number
- NO20062591L NO20062591L NO20062591A NO20062591A NO20062591L NO 20062591 L NO20062591 L NO 20062591L NO 20062591 A NO20062591 A NO 20062591A NO 20062591 A NO20062591 A NO 20062591A NO 20062591 L NO20062591 L NO 20062591L
- Authority
- NO
- Norway
- Prior art keywords
- cholesterol absorption
- diphenyllazetidinone
- derivatives
- inhibitory activity
- absorption inhibitory
- Prior art date
Links
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
- C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
- C07D205/06—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D205/08—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/10—Antimycotics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06008—Dipeptides with the first amino acid being neutral
- C07K5/06017—Dipeptides with the first amino acid being neutral and aliphatic
- C07K5/06026—Dipeptides with the first amino acid being neutral and aliphatic the side chain containing 0 or 1 carbon atom, i.e. Gly or Ala
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06008—Dipeptides with the first amino acid being neutral
- C07K5/06078—Dipeptides with the first amino acid being neutral and aromatic or cycloaliphatic
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
Abstract
Forbindelser med formel (I):. (hvor variable grupper er som definert i beskrivelsen), farmasøytisk akseptable salter, solvater, solvater av slike salter og promedikamenter derav, og anvendelse av dem som kolesterolabsorpsjonshemmere for behandling av hyperlipidemi, er beskrevet. Fremgangsmåter for fremstilling av dem, og farmasøytiske preparater inneholdende dem, er også beskrevet.
Applications Claiming Priority (4)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB0329780A GB0329780D0 (en) | 2003-12-23 | 2003-12-23 | Chemical compounds |
SE0401907A SE0401907D0 (sv) | 2004-07-21 | 2004-07-21 | Chemical compounds |
SE0402785A SE0402785D0 (sv) | 2004-11-15 | 2004-11-15 | Chemical compunds |
PCT/SE2004/001960 WO2005061452A1 (en) | 2003-12-23 | 2004-12-21 | Diphenylazetidinone derivates possessing cholesterol absorption inhibitory activity |
Publications (1)
Publication Number | Publication Date |
---|---|
NO20062591L true NO20062591L (no) | 2006-09-20 |
Family
ID=34714057
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO20062591A NO20062591L (no) | 2003-12-23 | 2006-06-06 | Difenylazetidinonderivater med kolesterolabsorpsjonsinhiberende aktivitet |
Country Status (15)
Country | Link |
---|---|
US (1) | US7871998B2 (no) |
EP (1) | EP1699759B1 (no) |
JP (1) | JP4688819B2 (no) |
AR (1) | AR047070A1 (no) |
AT (1) | ATE485267T1 (no) |
AU (1) | AU2004303742B2 (no) |
BR (1) | BRPI0418004A (no) |
CA (1) | CA2550215A1 (no) |
DE (1) | DE602004029715D1 (no) |
IL (1) | IL176158A0 (no) |
NO (1) | NO20062591L (no) |
SA (1) | SA04250427A (no) |
TW (1) | TW200526572A (no) |
UY (1) | UY28695A1 (no) |
WO (1) | WO2005061452A1 (no) |
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DE102007005045B4 (de) | 2007-01-26 | 2008-12-18 | Sanofi-Aventis | Phenothiazin Derivate, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel |
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-
2004
- 2004-12-21 AU AU2004303742A patent/AU2004303742B2/en not_active Ceased
- 2004-12-21 CA CA002550215A patent/CA2550215A1/en not_active Abandoned
- 2004-12-21 WO PCT/SE2004/001960 patent/WO2005061452A1/en active Application Filing
- 2004-12-21 JP JP2006546914A patent/JP4688819B2/ja not_active Expired - Fee Related
- 2004-12-21 SA SA04250427A patent/SA04250427A/ar unknown
- 2004-12-21 BR BRPI0418004-6A patent/BRPI0418004A/pt not_active IP Right Cessation
- 2004-12-21 DE DE602004029715T patent/DE602004029715D1/de active Active
- 2004-12-21 EP EP04809133A patent/EP1699759B1/en active Active
- 2004-12-21 AT AT04809133T patent/ATE485267T1/de not_active IP Right Cessation
- 2004-12-21 US US10/596,731 patent/US7871998B2/en not_active Expired - Fee Related
- 2004-12-22 AR ARP040104864A patent/AR047070A1/es not_active Application Discontinuation
- 2004-12-22 UY UY28695A patent/UY28695A1/es unknown
- 2004-12-23 TW TW093140329A patent/TW200526572A/zh unknown
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2006
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Also Published As
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TW200526572A (en) | 2005-08-16 |
DE602004029715D1 (de) | 2010-12-02 |
AU2004303742A1 (en) | 2005-07-07 |
BRPI0418004A (pt) | 2007-04-17 |
ATE485267T1 (de) | 2010-11-15 |
WO2005061452A1 (en) | 2005-07-07 |
EP1699759B1 (en) | 2010-10-20 |
AR047070A1 (es) | 2006-01-04 |
CA2550215A1 (en) | 2005-07-07 |
JP4688819B2 (ja) | 2011-05-25 |
IL176158A0 (en) | 2006-10-05 |
US20100099657A2 (en) | 2010-04-22 |
JP2007516280A (ja) | 2007-06-21 |
AU2004303742B2 (en) | 2008-06-19 |
UY28695A1 (es) | 2005-07-29 |
SA04250427A (ar) | 2005-12-03 |
EP1699759A1 (en) | 2006-09-13 |
US7871998B2 (en) | 2011-01-18 |
US20080064676A1 (en) | 2008-03-13 |
WO2005061452A8 (en) | 2006-04-06 |
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