NO20061322L - Kinazolinderivater som tyrosin kinase inhibitorer - Google Patents

Kinazolinderivater som tyrosin kinase inhibitorer

Info

Publication number
NO20061322L
NO20061322L NO20061322A NO20061322A NO20061322L NO 20061322 L NO20061322 L NO 20061322L NO 20061322 A NO20061322 A NO 20061322A NO 20061322 A NO20061322 A NO 20061322A NO 20061322 L NO20061322 L NO 20061322L
Authority
NO
Norway
Prior art keywords
quinazoline derivatives
tyrosine kinase
kinase inhibitors
manufacture
formula
Prior art date
Application number
NO20061322A
Other languages
English (en)
Norwegian (no)
Inventor
Laurent Francois And Hennequin
Christopher Thomas Halsall
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=34315440&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO20061322(L) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from GBGB0321620.7A external-priority patent/GB0321620D0/en
Priority claimed from GB0406163A external-priority patent/GB0406163D0/en
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of NO20061322L publication Critical patent/NO20061322L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C04—CEMENTS; CONCRETE; ARTIFICIAL STONE; CERAMICS; REFRACTORIES
    • C04B—LIME, MAGNESIA; SLAG; CEMENTS; COMPOSITIONS THEREOF, e.g. MORTARS, CONCRETE OR LIKE BUILDING MATERIALS; ARTIFICIAL STONE; CERAMICS; REFRACTORIES; TREATMENT OF NATURAL STONE
    • C04B35/00—Shaped ceramic products characterised by their composition; Ceramics compositions; Processing powders of inorganic compounds preparatory to the manufacturing of ceramic products
    • C04B35/622—Forming processes; Processing powders of inorganic compounds preparatory to the manufacturing of ceramic products
    • C04B35/626—Preparing or treating the powders individually or as batches ; preparing or treating macroscopic reinforcing agents for ceramic products, e.g. fibres; mechanical aspects section B
    • C04B35/63—Preparing or treating the powders individually or as batches ; preparing or treating macroscopic reinforcing agents for ceramic products, e.g. fibres; mechanical aspects section B using additives specially adapted for forming the products, e.g.. binder binders
    • C04B35/632—Organic additives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Ceramic Engineering (AREA)
  • Health & Medical Sciences (AREA)
  • Manufacturing & Machinery (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Inorganic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Structural Engineering (AREA)
  • Materials Engineering (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
NO20061322A 2003-09-16 2006-03-23 Kinazolinderivater som tyrosin kinase inhibitorer NO20061322L (no)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GBGB0321620.7A GB0321620D0 (en) 2003-09-16 2003-09-16 Quinazoline derivatives
GB0406163A GB0406163D0 (en) 2004-03-19 2004-03-19 Quinazoline derivatives
PCT/GB2004/003923 WO2005026150A1 (fr) 2003-09-16 2004-09-13 Derives de quinazoline utilises comme inhibiteurs de la tyrosine kinase

Publications (1)

Publication Number Publication Date
NO20061322L true NO20061322L (no) 2006-06-15

Family

ID=34315440

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20061322A NO20061322L (no) 2003-09-16 2006-03-23 Kinazolinderivater som tyrosin kinase inhibitorer

Country Status (25)

Country Link
US (2) US7569577B2 (fr)
EP (1) EP1667991B1 (fr)
JP (1) JP4795952B2 (fr)
AR (1) AR045663A1 (fr)
AT (1) ATE395346T1 (fr)
AU (1) AU2004272348B2 (fr)
BR (1) BRPI0414489A8 (fr)
CA (1) CA2538884C (fr)
CO (1) CO5690594A2 (fr)
CY (1) CY1108186T1 (fr)
DE (1) DE602004013806D1 (fr)
DK (1) DK1667991T3 (fr)
ES (1) ES2305844T3 (fr)
HK (1) HK1091480A1 (fr)
HR (1) HRP20080329T3 (fr)
IL (1) IL174261A0 (fr)
MX (1) MXPA06002964A (fr)
NO (1) NO20061322L (fr)
PL (1) PL1667991T3 (fr)
PT (1) PT1667991E (fr)
RU (1) RU2378268C2 (fr)
SI (1) SI1667991T1 (fr)
TW (1) TW200519104A (fr)
UA (1) UA84167C2 (fr)
WO (1) WO2005026150A1 (fr)

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US20080113874A1 (en) * 2004-01-23 2008-05-15 The Regents Of The University Of Colorado Gefitinib sensitivity-related gene expression and products and methods related thereto
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CA2723989C (fr) 2008-05-13 2017-04-25 Astrazeneca Ab Sel de fumarate de 4-(3-chloro-2-fluoroanilino)-7-methoxy-6-{[1-(n-methylcarbamoylmethyl)piperidin-4-yl]oxy}quinazoline
CN102452988B (zh) 2010-10-27 2016-01-27 中国科学院化学研究所 一种喹唑啉衍生物及其制备方法
JP6026441B2 (ja) 2011-03-04 2016-11-16 グラクソスミスクライン、インテレクチュアル、プロパティー、ディベロップメント、リミテッドＧｌａｘｏｓｍｉｔｈｋｌｉｎｅ Ｉｎｔｅｌｌｅｃｔｕａｌ Ｐｒｏｐｅｒｔｙ Ｄｅｖｅｌｏｐｍｅｎｔ Ｌｉｍｉｔｅｄ キナーゼ阻害剤としてのアミノキノリン
TWI547494B (zh) 2011-08-18 2016-09-01 葛蘭素史克智慧財產發展有限公司 作為激酶抑制劑之胺基喹唑啉類
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CA3044432A1 (fr) 2016-11-17 2018-05-24 Board Of Regents, The University Of Texas System Composes a activite antitumorale contre des cellules cancereuses porteuses de mutations egfr ou her2 exon 20

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JP2007505873A (ja) * 2003-09-16 2007-03-15 アストラゼネカ アクチボラグ チロシンキナーゼ阻害剤としてのキナゾリン誘導体
KR20070027487A (ko) * 2003-09-16 2007-03-09 아스트라제네카 아베 퀴나졸린 유도체
JP2007505878A (ja) * 2003-09-19 2007-03-15 アストラゼネカ アクチボラグ キナゾリン誘導体
GB0322409D0 (en) * 2003-09-25 2003-10-29 Astrazeneca Ab Quinazoline derivatives
BRPI0414735A (pt) * 2003-09-25 2006-11-21 Astrazeneca Ab derivado de quinazolina, composto, composição farmacêutica, uso de derivado de quinazolina, método para produzir um efeito anti-proliferativo em um animal de sangue quente, e, processo para a preparação de um derivado de quinazolina
GB0326459D0 (en) * 2003-11-13 2003-12-17 Astrazeneca Ab Quinazoline derivatives
WO2005075439A1 (fr) * 2004-02-03 2005-08-18 Astrazeneca Ab Derives de quinazoline
WO2005114576A1 (fr) * 2004-05-21 2005-12-01 Asahi Kasei Kabushiki Kaisha Dispositif d'évaluation du contenu d'opération
US20070232607A1 (en) * 2004-06-04 2007-10-04 Bradbury Robert H Quinazoline Derivatives as Erbb Receptor Tyrosine kinases

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US20090312343A1 (en) 2009-12-17
TW200519104A (en) 2005-06-16
CA2538884C (fr) 2010-09-21
PT1667991E (pt) 2008-07-14
JP4795952B2 (ja) 2011-10-19
EP1667991B1 (fr) 2008-05-14
EP1667991A1 (fr) 2006-06-14
DK1667991T3 (da) 2008-08-18
DE602004013806D1 (en) 2008-06-26
IL174261A0 (en) 2006-08-01
US20070043009A1 (en) 2007-02-22
AU2004272348A1 (en) 2005-03-24
BRPI0414489A (pt) 2006-11-14
ATE395346T1 (de) 2008-05-15
BRPI0414489A8 (pt) 2019-01-15
CY1108186T1 (el) 2014-02-12
JP2007505872A (ja) 2007-03-15
RU2378268C2 (ru) 2010-01-10
PL1667991T3 (pl) 2008-12-31
HRP20080329T3 (en) 2008-08-31
CO5690594A2 (es) 2006-10-31
RU2006112599A (ru) 2007-11-10
AU2004272348B2 (en) 2008-09-04
ES2305844T3 (es) 2008-11-01
CA2538884A1 (fr) 2005-03-24
SI1667991T1 (sl) 2008-10-31
US7569577B2 (en) 2009-08-04
AR045663A1 (es) 2005-11-02
WO2005026150A1 (fr) 2005-03-24
MXPA06002964A (es) 2006-06-14
HK1091480A1 (en) 2007-01-19
UA84167C2 (ru) 2008-09-25

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