NO20055316L - Nye heterocykliske forbindelser som er nyttige ved behandling av inflammatoriske og allergiske forstyrrelser, fremgangsmate for fremstilling derav og farmasoytiske sammensetninger som inneholder slike - Google Patents

Nye heterocykliske forbindelser som er nyttige ved behandling av inflammatoriske og allergiske forstyrrelser, fremgangsmate for fremstilling derav og farmasoytiske sammensetninger som inneholder slike

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Publication number
NO20055316L
NO20055316L NO20055316A NO20055316A NO20055316L NO 20055316 L NO20055316 L NO 20055316L NO 20055316 A NO20055316 A NO 20055316A NO 20055316 A NO20055316 A NO 20055316A NO 20055316 L NO20055316 L NO 20055316L
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pharmaceutical compositions
compositions containing
heterocyclic compounds
inflammatory
processes
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NO20055316A
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English (en)
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NO20055316D0 (no
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Aftab Dawoodbhai Lakdawala
Balasubramanian Gopalan
Laxmikant Atmaram Gharat
Usha Karaunakaran
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Glenmark Pharmaceuticals Sa
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Publication of NO20055316D0 publication Critical patent/NO20055316D0/no
Publication of NO20055316L publication Critical patent/NO20055316L/no

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/91—Dibenzofurans; Hydrogenated dibenzofurans
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    • A61P27/16—Otologicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A61P9/00—Drugs for disorders of the cardiovascular system
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    • A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links

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  • Chemical Kinetics & Catalysis (AREA)
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  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Cardiology (AREA)
  • Diabetes (AREA)
  • Hospice & Palliative Care (AREA)
  • Dermatology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
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  • Hematology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Urology & Nephrology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

Det beskrives nye, heterosykliske forbindelser samt deres analoger, tautomerer, regioisomerer, stereoisomerer, enantiomerer, diastereomerer, polymorfer, deres farmasøytisk akseptable salter, deres egnede N-oksider og deres farmasøytisk akseptable solvater. Videre beskrives det farmasøytiske preparater irmeholdende forbindelsene. Nærmere bestemt beskrives det nye fosfodiesterase type 4 (PDE4)-inhibitorer med formel (1) samt deres analoger, tautomerer, regioisomerer, stereoisomerer, enantiomerer, diastereomerer, polymorfer, deres farmasøytisk akseptable salter, deres egnede N-oksider og deres farmasøytisk akseptable solvater og også farmasøytiske preparater irmeholdende forbindelsene. Betydningen av gruppene X, Ar, Y, P og R' - R'' er definert i krav 1.
NO20055316A 2003-04-11 2005-11-10 Nye heterocykliske forbindelser som er nyttige ved behandling av inflammatoriske og allergiske forstyrrelser, fremgangsmate for fremstilling derav og farmasoytiske sammensetninger som inneholder slike NO20055316L (no)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
IN363MU2003 2003-04-11
US51996703P 2003-11-13 2003-11-13
PCT/IB2004/000355 WO2004089940A1 (en) 2003-04-11 2004-02-11 Novel heterocyclic compounds useful for the treatment of inflammatory and allergic disorders: process for their preparation and pharmaceutical compositions containing them

Publications (2)

Publication Number Publication Date
NO20055316D0 NO20055316D0 (no) 2005-11-10
NO20055316L true NO20055316L (no) 2006-01-11

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NO20055316A NO20055316L (no) 2003-04-11 2005-11-10 Nye heterocykliske forbindelser som er nyttige ved behandling av inflammatoriske og allergiske forstyrrelser, fremgangsmate for fremstilling derav og farmasoytiske sammensetninger som inneholder slike

Country Status (34)

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US (4) US7223789B2 (no)
EP (1) EP1620429B1 (no)
JP (1) JP2006522789A (no)
KR (1) KR20060017494A (no)
CN (1) CN1829711B (no)
AP (1) AP2008A (no)
AR (1) AR043199A1 (no)
AT (1) ATE427308T1 (no)
AU (1) AU2004228453B2 (no)
BR (1) BRPI0409747A (no)
CA (1) CA2522023A1 (no)
CL (1) CL2004000526A1 (no)
CO (1) CO5700824A2 (no)
DE (1) DE602004020332D1 (no)
DK (1) DK1620429T3 (no)
EA (1) EA010634B1 (no)
ES (1) ES2320888T3 (no)
GE (1) GEP20084526B (no)
HR (1) HRP20050944A2 (no)
IS (1) IS8123A (no)
MA (1) MA27801A1 (no)
MX (1) MXPA05010948A (no)
MY (1) MY136516A (no)
NO (1) NO20055316L (no)
NZ (1) NZ542882A (no)
OA (1) OA13154A (no)
PL (1) PL378813A1 (no)
PT (1) PT1620429E (no)
SI (1) SI1620429T1 (no)
TN (1) TNSN05252A1 (no)
TW (1) TW200508212A (no)
UA (1) UA79558C2 (no)
WO (1) WO2004089940A1 (no)
ZA (1) ZA200508240B (no)

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CN114163417B (zh) * 2021-12-06 2023-08-04 郑州海阔光电材料有限公司 一种3-溴硫芴的合成方法

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