NO20032241D0 - Forbedret prosess for vannlöselige azolforbindelser - Google Patents

Forbedret prosess for vannlöselige azolforbindelser

Info

Publication number
NO20032241D0
NO20032241D0 NO20032241A NO20032241A NO20032241D0 NO 20032241 D0 NO20032241 D0 NO 20032241D0 NO 20032241 A NO20032241 A NO 20032241A NO 20032241 A NO20032241 A NO 20032241A NO 20032241 D0 NO20032241 D0 NO 20032241D0
Authority
NO
Norway
Prior art keywords
improved process
water
azole compounds
soluble
triazole antifungal
Prior art date
Application number
NO20032241A
Other languages
English (en)
Norwegian (no)
Inventor
Chung-Pin Chen
Timothy Paul Connolly
Laxma Reddy Kolla
John D Matiskella
Richard H Mueller
Yadagiri Rendri
Dejah T Petsch
Original Assignee
Bristol Myers Squibb Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol Myers Squibb Co filed Critical Bristol Myers Squibb Co
Publication of NO20032241D0 publication Critical patent/NO20032241D0/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/06—Phosphorus compounds without P—C bonds
    • C07F9/08—Esters of oxyacids of phosphorus
    • C07F9/09—Esters of phosphoric acids
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6558—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing at least two different or differently substituted hetero rings neither condensed among themselves nor condensed with a common carbocyclic ring or ring system
    • C07F9/65583—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing at least two different or differently substituted hetero rings neither condensed among themselves nor condensed with a common carbocyclic ring or ring system each of the hetero rings containing nitrogen as ring hetero atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6515—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having three nitrogen atoms as the only ring hetero atoms
    • C07F9/6518—Five-membered rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Preventing Corrosion Or Incrustation Of Metals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
NO20032241A 2000-11-20 2003-05-19 Forbedret prosess for vannlöselige azolforbindelser NO20032241D0 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US25200100P 2000-11-20 2000-11-20
PCT/US2001/032382 WO2002042283A1 (en) 2000-11-20 2001-10-18 Improved process for water soluble azole compounds

Publications (1)

Publication Number Publication Date
NO20032241D0 true NO20032241D0 (no) 2003-05-19

Family

ID=22954236

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20032241A NO20032241D0 (no) 2000-11-20 2003-05-19 Forbedret prosess for vannlöselige azolforbindelser

Country Status (18)

Country Link
US (1) US6448401B1 (ko)
EP (1) EP1345915B1 (ko)
JP (1) JP4579496B2 (ko)
KR (1) KR100734456B1 (ko)
CN (1) CN1279033C (ko)
AT (1) ATE353079T1 (ko)
AU (2) AU1331702A (ko)
BR (1) BR0115448A (ko)
CA (1) CA2429378C (ko)
CZ (1) CZ20031388A3 (ko)
DE (1) DE60126425T2 (ko)
ES (1) ES2280405T3 (ko)
HU (1) HUP0301917A3 (ko)
IL (2) IL155612A0 (ko)
MX (1) MXPA03004332A (ko)
NO (1) NO20032241D0 (ko)
PL (1) PL361003A1 (ko)
WO (1) WO2002042283A1 (ko)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6362172B2 (en) * 2000-01-20 2002-03-26 Bristol-Myers Squibb Company Water soluble prodrugs of azole compounds
TWI329105B (en) 2002-02-01 2010-08-21 Rigel Pharmaceuticals Inc 2,4-pyrimidinediamine compounds and their uses
ES2421139T3 (es) 2003-07-30 2013-08-29 Rigel Pharmaceuticals, Inc. Compuestos de 2,4-pirimidindiamina para su uso en el tratamiento o la prevención de enfermedades autoinmunitarias
US20060047135A1 (en) * 2004-08-30 2006-03-02 Chadwick Scott T Process for preparing chloromethyl di-tert-butylphosphate
MX2007007189A (es) 2005-01-19 2010-09-28 Rigel Pharmaceuticals Inc Prodrogas de compuestos de 2,4-pirimidindiamina y sus usos.
JO2691B1 (en) * 2005-05-03 2013-03-03 ايساي آر آند دي مانجمنت كو.، ليمتد Monolysine salts for azole compounds
JP4981673B2 (ja) * 2005-09-13 2012-07-25 エーザイ・アール・アンド・ディー・マネジメント株式会社 安定性が改善されたクロロメチルフォスフェイト誘導体を含む組成物およびその製造方法
WO2007072851A1 (ja) * 2005-12-20 2007-06-28 Eisai R & D Management Co., Ltd. 水溶性アゾールプロドラッグの製造方法
AU2007218596C1 (en) 2006-02-22 2012-07-26 Eisai R & D Management Co., Ltd. Stabilized pharmaceutical composition
JP5221514B2 (ja) 2007-03-06 2013-06-26 エーザイ・アール・アンド・ディー・マネジメント株式会社 安定性が改善されたクロロメチルフォスフェイト誘導体を含む組成物及びその製造方法
FI20070574A0 (fi) * 2007-07-30 2007-07-30 Kuopion Yliopisto Vesiliukoinen propofolin etylideenifosfaatti-aihiolääke
KR20140057414A (ko) 2011-06-22 2014-05-12 바이옴 바이오사이언스 피브이티. 엘티디. 컨쥬게이트계 항진균 및 항세균 프로드러그
EP3525759A1 (en) * 2016-10-14 2019-08-21 Pulmatrix Operating Company, Inc. Antifungal dry powders

Family Cites Families (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2111527C (en) 1992-12-24 2000-07-18 Jerzy Golik Phosphonooxymethyl ethers of taxane derivatives
CA2129288C (en) 1993-08-17 2000-05-16 Jerzy Golik Phosphonooxymethyl esters of taxane derivatives
AU681753B2 (en) 1993-12-21 1997-09-04 Merck Sharp & Dohme Corp. Tetrahydrofuran antifungals
PT741737E (pt) 1994-01-24 2000-04-28 Janssen Pharmaceutica Nv Antifungicos do tipo azole soluveis em agua
NZ270418A (en) * 1994-02-07 1997-09-22 Eisai Co Ltd Polycyclic triazole & imidazole derivatives, antifungal compositions
ATE240319T1 (de) 1995-06-02 2003-05-15 Schering Corp Antifungale tetrahydrofurane
GB9602080D0 (en) * 1996-02-02 1996-04-03 Pfizer Ltd Pharmaceutical compounds
EP0829478A3 (en) 1996-09-09 1998-03-25 F. Hoffmann-La Roche Ag N-Benzylimidazolium and N-benzyltriazolium derivatives, their preparation and their use as antifungal and antimycotic agents
PT1056754E (pt) 1998-01-29 2004-03-31 Bristol Myers Squibb Co Derivados fosfatados de 1,3,4-oxadiazolona de diarilo
US5883097A (en) 1998-04-16 1999-03-16 Schering Corporation Soluble azole antifungal salt
US6265584B1 (en) 1998-05-22 2001-07-24 Bristol-Myers Squibb Company Water soluble prodrugs of azole compounds
US6204257B1 (en) * 1998-08-07 2001-03-20 Universtiy Of Kansas Water soluble prodrugs of hindered alcohols
WO2000030655A1 (en) * 1998-11-20 2000-06-02 Bristol-Myers Squibb Company Water soluble prodrugs of azole compounds
US6362172B2 (en) * 2000-01-20 2002-03-26 Bristol-Myers Squibb Company Water soluble prodrugs of azole compounds

Also Published As

Publication number Publication date
HUP0301917A2 (hu) 2003-09-29
EP1345915A1 (en) 2003-09-24
CN1279033C (zh) 2006-10-11
CN1474817A (zh) 2004-02-11
JP4579496B2 (ja) 2010-11-10
AU2002213317B2 (en) 2007-03-15
US20020062028A1 (en) 2002-05-23
DE60126425D1 (de) 2007-03-22
KR20040020865A (ko) 2004-03-09
ATE353079T1 (de) 2007-02-15
HUP0301917A3 (en) 2005-11-28
KR100734456B1 (ko) 2007-07-03
JP2004518640A (ja) 2004-06-24
AU1331702A (en) 2002-06-03
IL155612A (en) 2010-05-31
MXPA03004332A (es) 2004-05-04
WO2002042283A1 (en) 2002-05-30
CZ20031388A3 (cs) 2003-08-13
BR0115448A (pt) 2004-02-17
DE60126425T2 (de) 2007-10-18
ES2280405T3 (es) 2007-09-16
IL155612A0 (en) 2003-11-23
CA2429378A1 (en) 2002-05-30
EP1345915B1 (en) 2007-01-31
EP1345915A4 (en) 2005-08-03
US6448401B1 (en) 2002-09-10
CA2429378C (en) 2008-03-18
PL361003A1 (en) 2004-09-20

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