HUP0301917A3 - Proved process for water soluble azole compounds - Google Patents
Proved process for water soluble azole compoundsInfo
- Publication number
- HUP0301917A3 HUP0301917A3 HU0301917A HUP0301917A HUP0301917A3 HU P0301917 A3 HUP0301917 A3 HU P0301917A3 HU 0301917 A HU0301917 A HU 0301917A HU P0301917 A HUP0301917 A HU P0301917A HU P0301917 A3 HUP0301917 A3 HU P0301917A3
- Authority
- HU
- Hungary
- Prior art keywords
- water soluble
- azole compounds
- soluble azole
- proved process
- proved
- Prior art date
Links
- 150000003851 azoles Chemical class 0.000 title 1
- XLYOFNOQVPJJNP-UHFFFAOYSA-N water Substances O XLYOFNOQVPJJNP-UHFFFAOYSA-N 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/06—Phosphorus compounds without P—C bonds
- C07F9/08—Esters of oxyacids of phosphorus
- C07F9/09—Esters of phosphoric acids
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/6558—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing at least two different or differently substituted hetero rings neither condensed among themselves nor condensed with a common carbocyclic ring or ring system
- C07F9/65583—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing at least two different or differently substituted hetero rings neither condensed among themselves nor condensed with a common carbocyclic ring or ring system each of the hetero rings containing nitrogen as ring hetero atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/6515—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having three nitrogen atoms as the only ring hetero atoms
- C07F9/6518—Five-membered rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Biochemistry (AREA)
- General Health & Medical Sciences (AREA)
- Molecular Biology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Preventing Corrosion Or Incrustation Of Metals (AREA)
- Plural Heterocyclic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US25200100P | 2000-11-20 | 2000-11-20 | |
PCT/US2001/032382 WO2002042283A1 (en) | 2000-11-20 | 2001-10-18 | Improved process for water soluble azole compounds |
Publications (2)
Publication Number | Publication Date |
---|---|
HUP0301917A2 HUP0301917A2 (hu) | 2003-09-29 |
HUP0301917A3 true HUP0301917A3 (en) | 2005-11-28 |
Family
ID=22954236
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
HU0301917A HUP0301917A3 (en) | 2000-11-20 | 2001-10-18 | Proved process for water soluble azole compounds |
Country Status (18)
Country | Link |
---|---|
US (1) | US6448401B1 (hu) |
EP (1) | EP1345915B1 (hu) |
JP (1) | JP4579496B2 (hu) |
KR (1) | KR100734456B1 (hu) |
CN (1) | CN1279033C (hu) |
AT (1) | ATE353079T1 (hu) |
AU (2) | AU2002213317B2 (hu) |
BR (1) | BR0115448A (hu) |
CA (1) | CA2429378C (hu) |
CZ (1) | CZ20031388A3 (hu) |
DE (1) | DE60126425T2 (hu) |
ES (1) | ES2280405T3 (hu) |
HU (1) | HUP0301917A3 (hu) |
IL (2) | IL155612A0 (hu) |
MX (1) | MXPA03004332A (hu) |
NO (1) | NO20032241D0 (hu) |
PL (1) | PL361003A1 (hu) |
WO (1) | WO2002042283A1 (hu) |
Families Citing this family (13)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6362172B2 (en) * | 2000-01-20 | 2002-03-26 | Bristol-Myers Squibb Company | Water soluble prodrugs of azole compounds |
TWI329105B (en) | 2002-02-01 | 2010-08-21 | Rigel Pharmaceuticals Inc | 2,4-pyrimidinediamine compounds and their uses |
PT1656372E (pt) | 2003-07-30 | 2013-06-27 | Rigel Pharmaceuticals Inc | Métodos para o tratamento ou prevenção de doenças autoimunes com compostos de 2,4-pirimidinadiamina |
US20060047135A1 (en) * | 2004-08-30 | 2006-03-02 | Chadwick Scott T | Process for preparing chloromethyl di-tert-butylphosphate |
EP1856135B1 (en) | 2005-01-19 | 2009-12-09 | Rigel Pharmaceuticals, Inc. | Prodrugs of 2,4-pyrimidinediamine compounds and their uses |
JO2691B1 (en) * | 2005-05-03 | 2013-03-03 | ايساي آر آند دي مانجمنت كو.، ليمتد | Monolysine salts for azole compounds |
JP4981673B2 (ja) * | 2005-09-13 | 2012-07-25 | エーザイ・アール・アンド・ディー・マネジメント株式会社 | 安定性が改善されたクロロメチルフォスフェイト誘導体を含む組成物およびその製造方法 |
EP1964843B1 (en) * | 2005-12-20 | 2013-08-28 | Eisai R&D Management Co., Ltd. | Process for production of water-soluble azole prodrug |
CA2640331C (en) | 2006-02-22 | 2013-07-09 | Eisai R&D Management Co., Ltd. | Stabilized pharmaceutical composition |
WO2008108384A1 (ja) | 2007-03-06 | 2008-09-12 | Eisai R & D Management Co., Ltd. | 安定性が改善されたクロロメチルフォスフェイト誘導体を含む組成物及びその製造方法 |
FI20070574A0 (fi) * | 2007-07-30 | 2007-07-30 | Kuopion Yliopisto | Vesiliukoinen propofolin etylideenifosfaatti-aihiolääke |
KR20140057414A (ko) | 2011-06-22 | 2014-05-12 | 바이옴 바이오사이언스 피브이티. 엘티디. | 컨쥬게이트계 항진균 및 항세균 프로드러그 |
WO2018071757A1 (en) * | 2016-10-14 | 2018-04-19 | Pulmatrix Operating Company, Inc. | Antifungal dry powders |
Family Cites Families (14)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
NO310238B1 (no) | 1992-12-24 | 2001-06-11 | Bristol Myers Squibb Co | Kjemiske forbindelser og farmasöytisk preparat samt anvendelse av slike preparater |
CA2129288C (en) | 1993-08-17 | 2000-05-16 | Jerzy Golik | Phosphonooxymethyl esters of taxane derivatives |
CA2179396C (en) | 1993-12-21 | 2001-04-17 | Anil K. Saksena | Tetrahydrofuran antifungals |
KR100352147B1 (ko) | 1994-01-24 | 2002-11-11 | 얀센 파마슈티카 엔.브이. | 수용성아졸항진균제 |
NZ270418A (en) * | 1994-02-07 | 1997-09-22 | Eisai Co Ltd | Polycyclic triazole & imidazole derivatives, antifungal compositions |
NZ309281A (en) | 1995-06-02 | 1998-07-28 | Schering Corp | (2r-cis)-4-[4-[4-[4-[[(5-(2,4-dihalophenyl)-tetrahydro-5-(1h-1,2,4-tr iazol-1-ylmethyl)-tetrahydrofuran-3-yl]methoxy]phenyl]2,4-dihydro-2-[ esters and ethers of mono- or dihydroxy-substituted (c4-c5) alkyl]-3h-1,2,4-triazol-3-one |
GB9602080D0 (en) * | 1996-02-02 | 1996-04-03 | Pfizer Ltd | Pharmaceutical compounds |
EP0829478A3 (en) | 1996-09-09 | 1998-03-25 | F. Hoffmann-La Roche Ag | N-Benzylimidazolium and N-benzyltriazolium derivatives, their preparation and their use as antifungal and antimycotic agents |
DE69912250T2 (de) | 1998-01-29 | 2004-07-29 | Bristol-Myers Squibb Co., Wallingford | Phosphorylierte derivate des diaryl 1,3,4 oxadiazolon |
US5883097A (en) | 1998-04-16 | 1999-03-16 | Schering Corporation | Soluble azole antifungal salt |
US6265584B1 (en) | 1998-05-22 | 2001-07-24 | Bristol-Myers Squibb Company | Water soluble prodrugs of azole compounds |
US6204257B1 (en) * | 1998-08-07 | 2001-03-20 | Universtiy Of Kansas | Water soluble prodrugs of hindered alcohols |
WO2000030655A1 (en) * | 1998-11-20 | 2000-06-02 | Bristol-Myers Squibb Company | Water soluble prodrugs of azole compounds |
US6362172B2 (en) * | 2000-01-20 | 2002-03-26 | Bristol-Myers Squibb Company | Water soluble prodrugs of azole compounds |
-
2001
- 2001-10-16 US US09/982,199 patent/US6448401B1/en not_active Expired - Lifetime
- 2001-10-18 AU AU2002213317A patent/AU2002213317B2/en not_active Ceased
- 2001-10-18 CZ CZ20031388A patent/CZ20031388A3/cs unknown
- 2001-10-18 ES ES01981688T patent/ES2280405T3/es not_active Expired - Lifetime
- 2001-10-18 WO PCT/US2001/032382 patent/WO2002042283A1/en active IP Right Grant
- 2001-10-18 AU AU1331702A patent/AU1331702A/xx active Pending
- 2001-10-18 IL IL15561201A patent/IL155612A0/xx unknown
- 2001-10-18 DE DE60126425T patent/DE60126425T2/de not_active Expired - Lifetime
- 2001-10-18 CN CNB018191665A patent/CN1279033C/zh not_active Expired - Fee Related
- 2001-10-18 PL PL01361003A patent/PL361003A1/xx not_active Application Discontinuation
- 2001-10-18 HU HU0301917A patent/HUP0301917A3/hu unknown
- 2001-10-18 CA CA002429378A patent/CA2429378C/en not_active Expired - Lifetime
- 2001-10-18 KR KR1020037006747A patent/KR100734456B1/ko active IP Right Grant
- 2001-10-18 JP JP2002544418A patent/JP4579496B2/ja not_active Expired - Lifetime
- 2001-10-18 BR BR0115448-6A patent/BR0115448A/pt not_active IP Right Cessation
- 2001-10-18 AT AT01981688T patent/ATE353079T1/de not_active IP Right Cessation
- 2001-10-18 EP EP01981688A patent/EP1345915B1/en not_active Expired - Lifetime
- 2001-10-18 MX MXPA03004332A patent/MXPA03004332A/es unknown
-
2003
- 2003-04-28 IL IL155612A patent/IL155612A/en not_active IP Right Cessation
- 2003-05-19 NO NO20032241A patent/NO20032241D0/no unknown
Also Published As
Publication number | Publication date |
---|---|
HUP0301917A2 (hu) | 2003-09-29 |
AU2002213317B2 (en) | 2007-03-15 |
AU1331702A (en) | 2002-06-03 |
PL361003A1 (en) | 2004-09-20 |
CN1279033C (zh) | 2006-10-11 |
CA2429378A1 (en) | 2002-05-30 |
CN1474817A (zh) | 2004-02-11 |
CZ20031388A3 (cs) | 2003-08-13 |
BR0115448A (pt) | 2004-02-17 |
IL155612A (en) | 2010-05-31 |
KR20040020865A (ko) | 2004-03-09 |
WO2002042283A1 (en) | 2002-05-30 |
ATE353079T1 (de) | 2007-02-15 |
JP4579496B2 (ja) | 2010-11-10 |
EP1345915A4 (en) | 2005-08-03 |
US6448401B1 (en) | 2002-09-10 |
EP1345915A1 (en) | 2003-09-24 |
ES2280405T3 (es) | 2007-09-16 |
CA2429378C (en) | 2008-03-18 |
DE60126425T2 (de) | 2007-10-18 |
DE60126425D1 (de) | 2007-03-22 |
JP2004518640A (ja) | 2004-06-24 |
NO20032241D0 (no) | 2003-05-19 |
EP1345915B1 (en) | 2007-01-31 |
US20020062028A1 (en) | 2002-05-23 |
KR100734456B1 (ko) | 2007-07-03 |
IL155612A0 (en) | 2003-11-23 |
MXPA03004332A (es) | 2004-05-04 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FA9A | Lapse of provisional patent protection due to relinquishment or protection considered relinquished |