FI20070574A0 - Vesiliukoinen propofolin etylideenifosfaatti-aihiolääke - Google Patents

Vesiliukoinen propofolin etylideenifosfaatti-aihiolääke

Info

Publication number
FI20070574A0
FI20070574A0 FI20070574A FI20070574A FI20070574A0 FI 20070574 A0 FI20070574 A0 FI 20070574A0 FI 20070574 A FI20070574 A FI 20070574A FI 20070574 A FI20070574 A FI 20070574A FI 20070574 A0 FI20070574 A0 FI 20070574A0
Authority
FI
Finland
Prior art keywords
propofol
water
phosphate prodrug
soluble ethylene
ethylene phosphate
Prior art date
Application number
FI20070574A
Other languages
English (en)
Swedish (sv)
Inventor
Hanna Kumpulainen
Tomi Jaervinen
Jarkko Rautio
Original Assignee
Kuopion Yliopisto
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Kuopion Yliopisto filed Critical Kuopion Yliopisto
Priority to FI20070574A priority Critical patent/FI20070574A0/fi
Publication of FI20070574A0 publication Critical patent/FI20070574A0/fi
Priority to PCT/FI2008/050446 priority patent/WO2009016269A1/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/06Phosphorus compounds without P—C bonds
    • C07F9/08Esters of oxyacids of phosphorus
    • C07F9/09Esters of phosphoric acids
    • C07F9/12Esters of phosphoric acids with hydroxyaryl compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P23/00Anaesthetics

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Anesthesiology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
FI20070574A 2007-07-30 2007-07-30 Vesiliukoinen propofolin etylideenifosfaatti-aihiolääke FI20070574A0 (fi)

Priority Applications (2)

Application Number Priority Date Filing Date Title
FI20070574A FI20070574A0 (fi) 2007-07-30 2007-07-30 Vesiliukoinen propofolin etylideenifosfaatti-aihiolääke
PCT/FI2008/050446 WO2009016269A1 (en) 2007-07-30 2008-07-30 Water-soluble ethylidene phosphate prodrug of propofol

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FI20070574A FI20070574A0 (fi) 2007-07-30 2007-07-30 Vesiliukoinen propofolin etylideenifosfaatti-aihiolääke

Publications (1)

Publication Number Publication Date
FI20070574A0 true FI20070574A0 (fi) 2007-07-30

Family

ID=38331586

Family Applications (1)

Application Number Title Priority Date Filing Date
FI20070574A FI20070574A0 (fi) 2007-07-30 2007-07-30 Vesiliukoinen propofolin etylideenifosfaatti-aihiolääke

Country Status (2)

Country Link
FI (1) FI20070574A0 (fi)
WO (1) WO2009016269A1 (fi)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US9150600B2 (en) 2009-05-07 2015-10-06 Regents Of The University Of Minnesota Triptolide prodrugs
DK2427467T3 (en) * 2009-05-07 2015-11-09 Univ Minnesota Triptolid prodrugs
CN102784099A (zh) * 2012-06-11 2012-11-21 陕西合成药业有限公司 一种含有磷丙泊酚钠的组合制剂及其制备方法和用途
CN103588810B (zh) * 2013-11-29 2016-03-30 成都理工大学 丙泊酚水溶性环烷基磷酸酯衍生物
US11331271B2 (en) 2016-05-27 2022-05-17 The Johns Hopkins University Buccal, sublingual and intranasal delivery of fospropofol
US11478490B1 (en) 2021-03-30 2022-10-25 Epalex Corporation Fospropofol formulations
US11547714B2 (en) 2020-02-05 2023-01-10 Epalex Corporation Fospropofol salts, methods and compositions
US11628178B2 (en) 2019-03-26 2023-04-18 Epalex Corporation Fospropofol methods and compositions
US11439653B1 (en) 2021-03-30 2022-09-13 Epalex Corporation Fospropofol formulations

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2318817A1 (en) * 1998-01-29 1999-08-05 Bristol-Myers Squibb Company Phosphate derivatives of diaryl 1,3,4-oxadiazolone
US6204257B1 (en) * 1998-08-07 2001-03-20 Universtiy Of Kansas Water soluble prodrugs of hindered alcohols
US6448401B1 (en) * 2000-11-20 2002-09-10 Bristol-Myers Squibb Company Process for water soluble azole compounds
WO2006014282A2 (en) * 2004-07-06 2006-02-09 Abbott Laboratories Prodrugs of hiv protease inhibitors

Also Published As

Publication number Publication date
WO2009016269A1 (en) 2009-02-05

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Owner name: FENNOPHARMA OY

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