HUP0301917A3 - Proved process for water soluble azole compounds - Google Patents
Proved process for water soluble azole compoundsInfo
- Publication number
- HUP0301917A3 HUP0301917A3 HU0301917A HUP0301917A HUP0301917A3 HU P0301917 A3 HUP0301917 A3 HU P0301917A3 HU 0301917 A HU0301917 A HU 0301917A HU P0301917 A HUP0301917 A HU P0301917A HU P0301917 A3 HUP0301917 A3 HU P0301917A3
- Authority
- HU
- Hungary
- Prior art keywords
- water soluble
- azole compounds
- soluble azole
- proved process
- proved
- Prior art date
Links
- 150000003851 azoles Chemical class 0.000 title 1
- XLYOFNOQVPJJNP-UHFFFAOYSA-N water Substances O XLYOFNOQVPJJNP-UHFFFAOYSA-N 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/06—Phosphorus compounds without P—C bonds
- C07F9/08—Esters of oxyacids of phosphorus
- C07F9/09—Esters of phosphoric acids
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/6558—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing at least two different or differently substituted hetero rings neither condensed among themselves nor condensed with a common carbocyclic ring or ring system
- C07F9/65583—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing at least two different or differently substituted hetero rings neither condensed among themselves nor condensed with a common carbocyclic ring or ring system each of the hetero rings containing nitrogen as ring hetero atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/6515—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having three nitrogen atoms as the only ring hetero atoms
- C07F9/6518—Five-membered rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Biochemistry (AREA)
- General Health & Medical Sciences (AREA)
- Molecular Biology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Preventing Corrosion Or Incrustation Of Metals (AREA)
- Plural Heterocyclic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US25200100P | 2000-11-20 | 2000-11-20 | |
| PCT/US2001/032382 WO2002042283A1 (en) | 2000-11-20 | 2001-10-18 | Improved process for water soluble azole compounds |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| HUP0301917A2 HUP0301917A2 (en) | 2003-09-29 |
| HUP0301917A3 true HUP0301917A3 (en) | 2005-11-28 |
Family
ID=22954236
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| HU0301917A HUP0301917A3 (en) | 2000-11-20 | 2001-10-18 | Proved process for water soluble azole compounds |
Country Status (18)
| Country | Link |
|---|---|
| US (1) | US6448401B1 (en) |
| EP (1) | EP1345915B1 (en) |
| JP (1) | JP4579496B2 (en) |
| KR (1) | KR100734456B1 (en) |
| CN (1) | CN1279033C (en) |
| AT (1) | ATE353079T1 (en) |
| AU (2) | AU2002213317B2 (en) |
| BR (1) | BR0115448A (en) |
| CA (1) | CA2429378C (en) |
| CZ (1) | CZ20031388A3 (en) |
| DE (1) | DE60126425T2 (en) |
| ES (1) | ES2280405T3 (en) |
| HU (1) | HUP0301917A3 (en) |
| IL (2) | IL155612A0 (en) |
| MX (1) | MXPA03004332A (en) |
| NO (1) | NO20032241D0 (en) |
| PL (1) | PL361003A1 (en) |
| WO (1) | WO2002042283A1 (en) |
Families Citing this family (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6362172B2 (en) * | 2000-01-20 | 2002-03-26 | Bristol-Myers Squibb Company | Water soluble prodrugs of azole compounds |
| TWI329105B (en) | 2002-02-01 | 2010-08-21 | Rigel Pharmaceuticals Inc | 2,4-pyrimidinediamine compounds and their uses |
| US8178671B2 (en) | 2003-07-30 | 2012-05-15 | Rigel Pharmaceuticals, Inc. | Methods of treating or preventing autoimmune diseases with 2, 4-pyrimidinediamine compounds |
| US20060047135A1 (en) * | 2004-08-30 | 2006-03-02 | Chadwick Scott T | Process for preparing chloromethyl di-tert-butylphosphate |
| DE602006010979D1 (en) | 2005-01-19 | 2010-01-21 | Rigel Pharmaceuticals Inc | PRODRUGS FROM 2,4-PYRIMIDIN DIAMIN COMPOUNDS AND THEIR USES |
| JO2691B1 (en) * | 2005-05-03 | 2013-03-03 | ايساي آر آند دي مانجمنت كو.، ليمتد | Mono-lysine salts of azole compounds |
| JP4981673B2 (en) * | 2005-09-13 | 2012-07-25 | エーザイ・アール・アンド・ディー・マネジメント株式会社 | Composition comprising chloromethyl phosphate derivative with improved stability and method for producing the same |
| EP1964843B1 (en) * | 2005-12-20 | 2013-08-28 | Eisai R&D Management Co., Ltd. | Process for production of water-soluble azole prodrug |
| DE602007009489D1 (en) * | 2006-02-22 | 2010-11-11 | Eisai R&D Man Co Ltd | STABILIZED PHARMACEUTICAL COMPOSITION |
| CN101622263B (en) | 2007-03-06 | 2013-05-29 | 卫材R&D管理有限公司 | Composition containing chloromethyl phosphate derivative with improved stability and method for producing the same |
| FI20070574A0 (en) * | 2007-07-30 | 2007-07-30 | Kuopion Yliopisto | Water-soluble ethylene phosphate prodrug of propofol |
| EA032840B8 (en) | 2011-06-22 | 2020-06-18 | Вайоми Терапеутикс Лимитед | Conjugate-based antifungal prodrugs and use thereof |
| EP3525759A1 (en) * | 2016-10-14 | 2019-08-21 | Pulmatrix Operating Company, Inc. | Antifungal dry powders |
Family Cites Families (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA2111527C (en) | 1992-12-24 | 2000-07-18 | Jerzy Golik | Phosphonooxymethyl ethers of taxane derivatives |
| CA2129288C (en) | 1993-08-17 | 2000-05-16 | Jerzy Golik | Phosphonooxymethyl esters of taxane derivatives |
| DK0736030T3 (en) | 1993-12-21 | 2001-10-29 | Schering Corp | Fungicidal tetrahydrofurans |
| PL181947B1 (en) * | 1994-01-24 | 2001-10-31 | Janssen Pharmaceutica Nv | Water-soluble azole-type antimycotic agents |
| NZ270418A (en) * | 1994-02-07 | 1997-09-22 | Eisai Co Ltd | Polycyclic triazole & imidazole derivatives, antifungal compositions |
| WO1996038443A1 (en) | 1995-06-02 | 1996-12-05 | Schering Corporation | Tetrahydrofuran antifungals |
| GB9602080D0 (en) * | 1996-02-02 | 1996-04-03 | Pfizer Ltd | Pharmaceutical compounds |
| EP0829478A3 (en) | 1996-09-09 | 1998-03-25 | F. Hoffmann-La Roche Ag | N-Benzylimidazolium and N-benzyltriazolium derivatives, their preparation and their use as antifungal and antimycotic agents |
| DE69912250T2 (en) | 1998-01-29 | 2004-07-29 | Bristol-Myers Squibb Co., Wallingford | PHOSPHORYLATED DERIVATIVES OF DIARYL 1,3,4 OXADIAZOLONE |
| US5883097A (en) | 1998-04-16 | 1999-03-16 | Schering Corporation | Soluble azole antifungal salt |
| US6265584B1 (en) | 1998-05-22 | 2001-07-24 | Bristol-Myers Squibb Company | Water soluble prodrugs of azole compounds |
| US6204257B1 (en) * | 1998-08-07 | 2001-03-20 | Universtiy Of Kansas | Water soluble prodrugs of hindered alcohols |
| WO2000030655A1 (en) * | 1998-11-20 | 2000-06-02 | Bristol-Myers Squibb Company | Water soluble prodrugs of azole compounds |
| US6362172B2 (en) * | 2000-01-20 | 2002-03-26 | Bristol-Myers Squibb Company | Water soluble prodrugs of azole compounds |
-
2001
- 2001-10-16 US US09/982,199 patent/US6448401B1/en not_active Expired - Lifetime
- 2001-10-18 HU HU0301917A patent/HUP0301917A3/en unknown
- 2001-10-18 KR KR1020037006747A patent/KR100734456B1/en active IP Right Grant
- 2001-10-18 CN CNB018191665A patent/CN1279033C/en not_active Expired - Fee Related
- 2001-10-18 AT AT01981688T patent/ATE353079T1/en not_active IP Right Cessation
- 2001-10-18 ES ES01981688T patent/ES2280405T3/en not_active Expired - Lifetime
- 2001-10-18 PL PL01361003A patent/PL361003A1/en not_active Application Discontinuation
- 2001-10-18 CA CA002429378A patent/CA2429378C/en not_active Expired - Lifetime
- 2001-10-18 AU AU2002213317A patent/AU2002213317B2/en not_active Ceased
- 2001-10-18 EP EP01981688A patent/EP1345915B1/en not_active Expired - Lifetime
- 2001-10-18 BR BR0115448-6A patent/BR0115448A/en not_active IP Right Cessation
- 2001-10-18 IL IL15561201A patent/IL155612A0/en unknown
- 2001-10-18 WO PCT/US2001/032382 patent/WO2002042283A1/en active IP Right Grant
- 2001-10-18 MX MXPA03004332A patent/MXPA03004332A/en unknown
- 2001-10-18 AU AU1331702A patent/AU1331702A/en active Pending
- 2001-10-18 DE DE60126425T patent/DE60126425T2/en not_active Expired - Lifetime
- 2001-10-18 CZ CZ20031388A patent/CZ20031388A3/en unknown
- 2001-10-18 JP JP2002544418A patent/JP4579496B2/en not_active Expired - Lifetime
-
2003
- 2003-04-28 IL IL155612A patent/IL155612A/en not_active IP Right Cessation
- 2003-05-19 NO NO20032241A patent/NO20032241D0/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| ES2280405T3 (en) | 2007-09-16 |
| JP4579496B2 (en) | 2010-11-10 |
| IL155612A (en) | 2010-05-31 |
| NO20032241D0 (en) | 2003-05-19 |
| EP1345915A4 (en) | 2005-08-03 |
| US20020062028A1 (en) | 2002-05-23 |
| DE60126425D1 (en) | 2007-03-22 |
| CN1279033C (en) | 2006-10-11 |
| EP1345915A1 (en) | 2003-09-24 |
| CA2429378C (en) | 2008-03-18 |
| JP2004518640A (en) | 2004-06-24 |
| US6448401B1 (en) | 2002-09-10 |
| MXPA03004332A (en) | 2004-05-04 |
| AU1331702A (en) | 2002-06-03 |
| ATE353079T1 (en) | 2007-02-15 |
| CZ20031388A3 (en) | 2003-08-13 |
| HUP0301917A2 (en) | 2003-09-29 |
| PL361003A1 (en) | 2004-09-20 |
| CA2429378A1 (en) | 2002-05-30 |
| WO2002042283A1 (en) | 2002-05-30 |
| EP1345915B1 (en) | 2007-01-31 |
| BR0115448A (en) | 2004-02-17 |
| CN1474817A (en) | 2004-02-11 |
| DE60126425T2 (en) | 2007-10-18 |
| KR20040020865A (en) | 2004-03-09 |
| KR100734456B1 (en) | 2007-07-03 |
| IL155612A0 (en) | 2003-11-23 |
| AU2002213317B2 (en) | 2007-03-15 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FA9A | Lapse of provisional patent protection due to relinquishment or protection considered relinquished |