NO20021781L - Heteroalkylamino-substituerte bicykliske nitrogenheterocykler som inhibitorer for P38-proteinkinase - Google Patents

Heteroalkylamino-substituerte bicykliske nitrogenheterocykler som inhibitorer for P38-proteinkinase

Info

Publication number
NO20021781L
NO20021781L NO20021781A NO20021781A NO20021781L NO 20021781 L NO20021781 L NO 20021781L NO 20021781 A NO20021781 A NO 20021781A NO 20021781 A NO20021781 A NO 20021781A NO 20021781 L NO20021781 L NO 20021781L
Authority
NO
Norway
Prior art keywords
inhibitors
heteroalkylamino
protein kinase
substituted bicyclic
nitrogen heterocycles
Prior art date
Application number
NO20021781A
Other languages
English (en)
Norwegian (no)
Other versions
NO20021781D0 (no
Inventor
James Patrick Dunn
Lawrence Emerson Fisher
David Michael Goldstein
William Harris
Christopher Huw Hill
Ian Edward David Smith
Teresa Rosanne Welch
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of NO20021781D0 publication Critical patent/NO20021781D0/no
Publication of NO20021781L publication Critical patent/NO20021781L/no

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
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    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
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  • Health & Medical Sciences (AREA)
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  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Medicinal Chemistry (AREA)
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  • Diabetes (AREA)
  • Rheumatology (AREA)
  • Virology (AREA)
  • Pulmonology (AREA)
  • Oncology (AREA)
  • Biomedical Technology (AREA)
  • Dermatology (AREA)
  • Cardiology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Hematology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Communicable Diseases (AREA)
  • Ophthalmology & Optometry (AREA)
  • Pain & Pain Management (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Hospice & Palliative Care (AREA)
  • Molecular Biology (AREA)
  • Reproductive Health (AREA)
  • Urology & Nephrology (AREA)
  • Endocrinology (AREA)
  • Transplantation (AREA)
NO20021781A 1999-10-21 2002-04-16 Heteroalkylamino-substituerte bicykliske nitrogenheterocykler som inhibitorer for P38-proteinkinase NO20021781L (no)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US16080399P 1999-10-21 1999-10-21
US21374300P 2000-06-22 2000-06-22
PCT/EP2000/010088 WO2001029042A1 (en) 1999-10-21 2000-10-13 Heteroalkylamino-substituted bicyclic nitrogen heterocycles as inhibitors of p38 protein kinase

Publications (2)

Publication Number Publication Date
NO20021781D0 NO20021781D0 (no) 2002-04-16
NO20021781L true NO20021781L (no) 2002-04-18

Family

ID=26857240

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20021781A NO20021781L (no) 1999-10-21 2002-04-16 Heteroalkylamino-substituerte bicykliske nitrogenheterocykler som inhibitorer for P38-proteinkinase

Country Status (27)

Country Link
US (1) US6451804B1 (sh)
EP (1) EP1228070B1 (sh)
JP (1) JP3961830B2 (sh)
KR (1) KR100523120B1 (sh)
CN (1) CN1171889C (sh)
AR (1) AR026084A1 (sh)
AT (1) ATE353329T1 (sh)
AU (1) AU776250B2 (sh)
BR (1) BR0015243A (sh)
CA (1) CA2388142C (sh)
CZ (1) CZ20021744A3 (sh)
DE (1) DE60033307T2 (sh)
ES (1) ES2280247T3 (sh)
HK (1) HK1051039A1 (sh)
HR (1) HRP20020328A2 (sh)
HU (1) HUP0203564A3 (sh)
IL (1) IL149100A0 (sh)
MA (1) MA26837A1 (sh)
MX (1) MXPA02003950A (sh)
NO (1) NO20021781L (sh)
NZ (1) NZ518119A (sh)
PE (1) PE20010758A1 (sh)
PL (1) PL357502A1 (sh)
RU (1) RU2265606C2 (sh)
TR (1) TR200201057T2 (sh)
WO (1) WO2001029042A1 (sh)
YU (1) YU29102A (sh)

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RU2310657C2 (ru) * 2002-04-03 2007-11-20 Ф.Хоффманн-Ля Рош Аг Имидазоконденсированные соединения и фармацевтическая композиция, содержащая их
BR0309053A (pt) * 2002-04-19 2005-02-22 Smithkline Beecham Corp Compostos
DE60310730T2 (de) 2002-07-09 2007-05-16 Boehringer Ingelheim Pharma Gmbh & Co. Kg Pharmazeutische zusammensetzungen aus anticholinergica und p38 kinase hemmern zur behandlung von erkrankungen der atemwege
PA8577501A1 (es) 2002-07-25 2004-02-07 Warner Lambert Co Inhibidores de quinasas
JP4252534B2 (ja) * 2002-08-06 2009-04-08 エフ．ホフマン−ラ ロシュ アーゲー ｐ−３８ＭＡＰキナーゼインヒビターとしての６−アルコキシ−ピリド−ピリミジン類
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EP2108641A1 (en) * 2008-04-11 2009-10-14 Laboratorios Almirall, S.A. New substituted spiro[cycloalkyl-1,3'-indo]-2'(1'H)-one derivatives and their use as p38 mitogen-activated kinase inhibitors
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