NO20011638L - Imidazo[4,5-c]pyridin-4-on-derivater med faktor Xa- inhiberende virkning - Google Patents
Imidazo[4,5-c]pyridin-4-on-derivater med faktor Xa- inhiberende virkningInfo
- Publication number
- NO20011638L NO20011638L NO20011638A NO20011638A NO20011638L NO 20011638 L NO20011638 L NO 20011638L NO 20011638 A NO20011638 A NO 20011638A NO 20011638 A NO20011638 A NO 20011638A NO 20011638 L NO20011638 L NO 20011638L
- Authority
- NO
- Norway
- Prior art keywords
- imidazo
- pyridin
- derivatives
- factor
- inhibitory effect
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
- A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE19845153A DE19845153A1 (de) | 1998-10-01 | 1998-10-01 | Imidazo[4,5]-pyridin-4-on-derivate |
| PCT/EP1999/006655 WO2000020416A1 (de) | 1998-10-01 | 1999-09-09 | Imidazo[4,5-c-]-pyridin-4-on-derivate mit faktor xa hemmender wirkung |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| NO20011638L true NO20011638L (no) | 2001-03-30 |
| NO20011638D0 NO20011638D0 (no) | 2001-03-30 |
Family
ID=7883005
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO20011638A NO20011638D0 (no) | 1998-10-01 | 2001-03-30 | Imidazo[4,5-c]pyridin-4-on-derivater med faktor Xa- inhiberende virkning |
Country Status (18)
| Country | Link |
|---|---|
| US (1) | US6492384B1 (de) |
| EP (1) | EP1117664A1 (de) |
| JP (1) | JP2002526542A (de) |
| KR (1) | KR20010074980A (de) |
| CN (1) | CN1324358A (de) |
| AR (1) | AR020688A1 (de) |
| AU (1) | AU752574B2 (de) |
| BR (1) | BR9914213A (de) |
| CA (1) | CA2346033A1 (de) |
| DE (1) | DE19845153A1 (de) |
| HU (1) | HUP0104164A3 (de) |
| ID (1) | ID29466A (de) |
| MY (1) | MY130736A (de) |
| NO (1) | NO20011638D0 (de) |
| PL (1) | PL346542A1 (de) |
| SK (1) | SK4282001A3 (de) |
| WO (1) | WO2000020416A1 (de) |
| ZA (1) | ZA200103498B (de) |
Families Citing this family (19)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DK1140941T3 (da) | 1998-12-23 | 2005-02-14 | Bristol Myers Squibb Pharma Co | Nitrogenholdige heterobicykliske forbindelser som faktor Xa-inhibitorer |
| US6858616B2 (en) | 1998-12-23 | 2005-02-22 | Bristol-Myers Squibb Pharma Company | Nitrogen containing heterobicycles as factor Xa inhibitors |
| AU2001268712A1 (en) | 2000-06-23 | 2002-01-08 | Bristol-Myers Squibb Company | 1 - (heteroaryl-phenyl) - condensed pyrazol derivatives as factor Xa inhibitors |
| AU2002310070A1 (en) | 2001-05-22 | 2002-12-03 | Bristol-Myers Squibb Company | Bicyclic inhibitors of factor xa |
| AU2003210958A1 (en) * | 2002-02-08 | 2003-09-02 | Glsynthesis Inc. | Purine and isosteric antibacterial compounds |
| GB0215293D0 (en) * | 2002-07-03 | 2002-08-14 | Rega Foundation | Viral inhibitors |
| DK1569912T3 (en) | 2002-12-03 | 2015-06-29 | Pharmacyclics Inc | 2- (2-hydroxybiphenyl-3-yl) -1h-benzoimidazole-5-carboxamidine derivatives as factor VIIa inhibitors. |
| US7135469B2 (en) * | 2003-03-18 | 2006-11-14 | Bristol Myers Squibb, Co. | Linear chain substituted monocyclic and bicyclic derivatives as factor Xa inhibitors |
| ATE544765T1 (de) * | 2003-12-22 | 2012-02-15 | Leuven K U Res & Dev | Imidazoä4,5-cüpyridinverbindungen und verfahren zur antiviralen behandlung |
| US7381732B2 (en) | 2004-10-26 | 2008-06-03 | Bristol-Myers Squibb Company | Pyrazolobenzamides and derivatives as factor Xa inhibitors |
| CA2592388C (en) * | 2004-12-21 | 2013-04-02 | Steven S. Bondy | Imidazo[4,5-c]pyridine compound and method of antiviral treatment |
| NZ566799A (en) | 2005-09-14 | 2011-04-29 | Takeda Pharmaceutical | Dipeptidyl peptidase inhibitors for treating diabetes |
| CN101360723A (zh) | 2005-09-16 | 2009-02-04 | 武田药品工业株式会社 | 制备嘧啶二酮衍生物的方法 |
| TW200734338A (en) * | 2006-01-16 | 2007-09-16 | Organon Nv | 6-Phenyl-1H-imidazo [4,5-c] pyridine-4-carbonitrile derivatives |
| WO2007112347A1 (en) | 2006-03-28 | 2007-10-04 | Takeda Pharmaceutical Company Limited | Dipeptidyl peptidase inhibitors |
| ES2339298T3 (es) * | 2006-07-07 | 2010-05-18 | Gilead Sciences, Inc. | Compuesto de piridazina novedoso y uso del mismo. |
| TW200838536A (en) | 2006-11-29 | 2008-10-01 | Takeda Pharmaceutical | Polymorphs of succinate salt of 2-[6-(3-amino-piperidin-1-yl)-3-methyl-2,4-dioxo-3,4-dihydro-2H-pyrimidin-1-ylmethy]-4-fluor-benzonitrile and methods of use therefor |
| UA99466C2 (en) | 2007-07-06 | 2012-08-27 | Гилиад Сайенсиз, Инк. | Crystalline pyridazine compound |
| CA2772907C (en) | 2009-09-11 | 2018-01-09 | Glsynthesis Inc. | Selective antibacterials for clostridium difficile infections |
Family Cites Families (18)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE602521C (de) * | 1934-09-10 | Wilhelm Stoeckicht Dipl Ing | Umlaufraederwechselgetriebe, insbesondere fuer Kraftfahrzeuge | |
| DE546449C (de) * | 1932-03-12 | Mueller Paul | Verbindung von Belagblechen | |
| DE574846C (de) * | 1933-04-21 | Wilhelm Germann | Schienenbefestigung unter Verwendung von Schienenfuehrungsleisten | |
| DE595151C (de) * | 1934-04-04 | Buderus Eisenwerk | Verfahren und Vorrichtung zum Regeln des Gewichts von in Schleudergussmaschinen herzustellenden Rohren | |
| DE505893C (de) * | 1926-08-07 | 1930-08-26 | Medizinische Produkte Ag F | Verfahren zur Herstellung von Eiweiss-Halogen-Schwefelverbindungen |
| DE564960C (de) * | 1931-05-13 | 1932-11-24 | Siemens Schuckertwerke Akt Ges | Einrichtung zur Anpassung der Drehzahlregelung, insbesondere von Dampfturbinen, an veraenderte Betriebsverhaeltnisse |
| DE628556C (de) * | 1932-12-07 | 1936-04-08 | Wolf Johannes Mueller Dr | Verfahren zur Herstellung von insbesondere hochkonzentrierten Wasserglasloesungen |
| DE702013C (de) * | 1933-07-17 | 1941-01-29 | Union Oil Co | Verfahren zur Abscheidung von Paraffin aus paraffinhaltigen OElen |
| US5798364A (en) * | 1992-03-26 | 1998-08-25 | Merck Patent Gesellschaft Mit Beschrankter Haftung | Imidazopyridines |
| DE4110019C2 (de) | 1991-03-27 | 2000-04-13 | Merck Patent Gmbh | Imidazopyridine, Verfahren zu ihrer Herstellung und diese enthaltende pharmazeutische Zubereitungen |
| DE4140519A1 (de) * | 1991-12-09 | 1993-06-17 | Merck Patent Gmbh | Benzofurane |
| DE4211474A1 (de) * | 1992-04-06 | 1993-10-07 | Merck Patent Gmbh | Imidazopyridine |
| DE4305602A1 (de) * | 1992-06-17 | 1993-12-23 | Merck Patent Gmbh | Imidazopyridine |
| DE4236026A1 (de) * | 1992-10-24 | 1994-04-28 | Merck Patent Gmbh | Imidazopyridine |
| DE4242459A1 (de) | 1992-12-16 | 1994-06-23 | Merck Patent Gmbh | Imidazopyridine |
| DE4318813A1 (de) | 1993-06-07 | 1994-12-08 | Merck Patent Gmbh | Imidazopyridine |
| DE4432860A1 (de) | 1994-09-15 | 1996-03-21 | Merck Patent Gmbh | Imidazopyridine |
| EP0960102A1 (de) | 1996-07-08 | 1999-12-01 | Du Pont Pharmaceuticals Company | Amidinoindole, amidinoazole und analoge davon als inhibitoren von thrombin und von faktor xa |
-
1998
- 1998-10-01 DE DE19845153A patent/DE19845153A1/de not_active Withdrawn
-
1999
- 1999-09-09 CN CN99811601A patent/CN1324358A/zh active Pending
- 1999-09-09 KR KR1020017002922A patent/KR20010074980A/ko not_active Application Discontinuation
- 1999-09-09 BR BR9914213-9A patent/BR9914213A/pt not_active IP Right Cessation
- 1999-09-09 US US09/806,418 patent/US6492384B1/en not_active Expired - Fee Related
- 1999-09-09 CA CA002346033A patent/CA2346033A1/en not_active Abandoned
- 1999-09-09 PL PL99346542A patent/PL346542A1/xx unknown
- 1999-09-09 EP EP99946151A patent/EP1117664A1/de not_active Withdrawn
- 1999-09-09 SK SK428-2001A patent/SK4282001A3/sk unknown
- 1999-09-09 HU HU0104164A patent/HUP0104164A3/hu unknown
- 1999-09-09 ID IDW20010909A patent/ID29466A/id unknown
- 1999-09-09 AU AU58618/99A patent/AU752574B2/en not_active Ceased
- 1999-09-09 WO PCT/EP1999/006655 patent/WO2000020416A1/de not_active Application Discontinuation
- 1999-09-09 JP JP2000574528A patent/JP2002526542A/ja active Pending
- 1999-09-28 MY MYPI99004187A patent/MY130736A/en unknown
- 1999-10-01 AR ARP990104991A patent/AR020688A1/es not_active Application Discontinuation
-
2001
- 2001-03-30 NO NO20011638A patent/NO20011638D0/no not_active Application Discontinuation
- 2001-04-30 ZA ZA200103498A patent/ZA200103498B/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| EP1117664A1 (de) | 2001-07-25 |
| WO2000020416A1 (de) | 2000-04-13 |
| JP2002526542A (ja) | 2002-08-20 |
| SK4282001A3 (en) | 2002-10-08 |
| HUP0104164A3 (en) | 2002-08-28 |
| AR020688A1 (es) | 2002-05-22 |
| MY130736A (en) | 2007-07-31 |
| CA2346033A1 (en) | 2000-04-13 |
| US6492384B1 (en) | 2002-12-10 |
| CN1324358A (zh) | 2001-11-28 |
| HUP0104164A2 (hu) | 2002-04-29 |
| ZA200103498B (en) | 2002-08-13 |
| PL346542A1 (en) | 2002-02-11 |
| BR9914213A (pt) | 2001-06-26 |
| KR20010074980A (ko) | 2001-08-09 |
| AU752574B2 (en) | 2002-09-26 |
| ID29466A (id) | 2001-08-30 |
| AU5861899A (en) | 2000-04-26 |
| NO20011638D0 (no) | 2001-03-30 |
| DE19845153A1 (de) | 2000-04-06 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FC2A | Withdrawal, rejection or dismissal of laid open patent application |