NO173607C - Analogifremgangsmaate for fremstilling av nye terapeutisk aktive tienotriazolo-diazepin-derivater - Google Patents

Analogifremgangsmaate for fremstilling av nye terapeutisk aktive tienotriazolo-diazepin-derivater

Info

Publication number
NO173607C
NO173607C NO901813A NO901813A NO173607C NO 173607 C NO173607 C NO 173607C NO 901813 A NO901813 A NO 901813A NO 901813 A NO901813 A NO 901813A NO 173607 C NO173607 C NO 173607C
Authority
NO
Norway
Prior art keywords
thienotriazolo
preparation
therapeutically active
analogous procedures
new therapeutically
Prior art date
Application number
NO901813A
Other languages
English (en)
Norwegian (no)
Other versions
NO901813L (no
NO901813D0 (no
NO173607B (no
Inventor
Pierre Braquet
Andr Esanu
Jean-Pierre Laurent
Jacques Pommier
Original Assignee
Sod Conseils Rech Applic
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sod Conseils Rech Applic filed Critical Sod Conseils Rech Applic
Publication of NO901813D0 publication Critical patent/NO901813D0/no
Publication of NO901813L publication Critical patent/NO901813L/no
Publication of NO173607B publication Critical patent/NO173607B/no
Publication of NO173607C publication Critical patent/NO173607C/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/22Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains four or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
NO901813A 1989-05-13 1990-04-24 Analogifremgangsmaate for fremstilling av nye terapeutisk aktive tienotriazolo-diazepin-derivater NO173607C (no)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB898911030A GB8911030D0 (en) 1989-05-13 1989-05-13 Hetrazepine derivatives

Publications (4)

Publication Number Publication Date
NO901813D0 NO901813D0 (no) 1990-04-24
NO901813L NO901813L (no) 1990-11-14
NO173607B NO173607B (no) 1993-09-27
NO173607C true NO173607C (no) 1994-01-05

Family

ID=10656702

Family Applications (1)

Application Number Title Priority Date Filing Date
NO901813A NO173607C (no) 1989-05-13 1990-04-24 Analogifremgangsmaate for fremstilling av nye terapeutisk aktive tienotriazolo-diazepin-derivater

Country Status (32)

Country Link
US (1) US5049559A (fr)
JP (1) JPH06104668B2 (fr)
KR (1) KR900018113A (fr)
AR (1) AR245725A1 (fr)
AT (1) AT399153B (fr)
AU (1) AU628171B2 (fr)
BE (1) BE1004122A3 (fr)
CA (1) CA2016551C (fr)
CH (1) CH681009A5 (fr)
DE (1) DE4015137C2 (fr)
DK (1) DK102990A (fr)
DZ (1) DZ1414A1 (fr)
ES (1) ES2019840A6 (fr)
FI (1) FI93119C (fr)
FR (2) FR2646774B1 (fr)
GB (2) GB8911030D0 (fr)
GR (1) GR1000295B (fr)
HK (1) HK94992A (fr)
IE (1) IE65246B1 (fr)
IN (1) IN174000B (fr)
IT (1) IT1240935B (fr)
LU (1) LU87733A1 (fr)
MA (1) MA21842A1 (fr)
NL (1) NL9001089A (fr)
NO (1) NO173607C (fr)
NZ (1) NZ233574A (fr)
OA (1) OA09209A (fr)
PT (1) PT94008B (fr)
SE (1) SE505407C2 (fr)
SG (1) SG91992G (fr)
TN (1) TNSN90061A1 (fr)
ZA (1) ZA903305B (fr)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5382579A (en) * 1988-10-31 1995-01-17 Eisai Co., Ltd. Triazolo-1,4-diazepine derivatives and their use in pharmaceuticals
US5304553A (en) * 1988-10-31 1994-04-19 Eisai Co., Ltd. 1,4-diazepine derivative and its pharmaceutical use
US5468740A (en) * 1988-10-31 1995-11-21 Eisai Co., Ltd. 1,4-diazepine derivative and its pharmaceutical use
FI95708C (fi) * 1988-10-31 1996-03-11 Eisai Co Ltd Analogiamenetelmä 1,4-diatsepiinijohdannaisen ja sen farmaseuttisesti sopivan suolan valmistamiseksi
US5221671A (en) * 1988-10-31 1993-06-22 Eisai Co., Ltd. Triazolo-1,4-diazepine derivatives and their use in pharmaceuticals
AT394563B (de) * 1990-05-09 1992-05-11 Scras Verfahren zur herstellung von thieno-triazolodiazepinderivaten
GB9207645D0 (en) * 1992-04-08 1992-05-27 Smithkline Beecham Corp Methods
ES2061406B1 (es) * 1993-05-07 1995-06-01 Uriach & Cia Sa J Nuevos derivados de la 2-(quinolina) con actividad farmacologica.
US6262044B1 (en) 1998-03-12 2001-07-17 Novo Nordisk A/S Modulators of protein tyrosine phosphatases (PTPASES)
WO2001083440A2 (fr) * 2000-04-28 2001-11-08 Board Of Supervisors Of Louisiana State University And Agricultural And Mechanical College Synthese et utilisation de thienotriazolodiazepines
JP4901474B2 (ja) 2003-05-30 2012-03-21 ランバクシー ラボラトリーズ リミテッド 置換ピロール誘導体
JP2009514851A (ja) 2005-11-08 2009-04-09 ランバクシー ラボラトリーズ リミテッド (3r,5r)−7−[2−(4−フルオロフェニル)−5−イソプロピル−3−フェニル−4−[(4−ヒドロキシメチルフェニルアミノ)カルボニル]−ピロール−1−イル]−3,5−ジヒドロキシ−ヘプタン酸ヘミカルシウム塩の製法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3435973A1 (de) * 1984-10-01 1986-04-10 Boehringer Ingelheim KG, 6507 Ingelheim Diazepine enthaltende pharmazeutische zusammensetzungen mit paf-antagonistischer wirkung
DE3724031A1 (de) * 1986-07-22 1988-01-28 Boehringer Ingelheim Kg Neue hetrazepine und verfahren zu ihrer herstellung
PH30676A (en) * 1986-07-22 1997-09-16 Boehringer Ingelhein Kg Hetrazepine compounds which have useful pharmaceutical utility
US5028603A (en) * 1987-06-08 1991-07-02 Yoshitomi Pharmaceutical Industries, Ltd. Ester-substituted thienotriazolodiazepine compounds and pharmaceutical uses thereof

Also Published As

Publication number Publication date
GB9010403D0 (en) 1990-06-27
IE65246B1 (en) 1995-10-04
JPH06104668B2 (ja) 1994-12-21
MA21842A1 (fr) 1990-12-31
AU5493190A (en) 1990-11-15
NO901813L (no) 1990-11-14
PT94008B (pt) 1996-12-31
IE901583L (en) 1990-11-13
GR1000295B (el) 1992-05-12
SG91992G (en) 1992-12-04
TNSN90061A1 (fr) 1991-03-05
LU87733A1 (fr) 1990-09-19
OA09209A (fr) 1992-06-30
NL9001089A (nl) 1990-12-03
NO901813D0 (no) 1990-04-24
SE9001670D0 (sv) 1990-05-09
NO173607B (no) 1993-09-27
GB2231330A (en) 1990-11-14
AT399153B (de) 1995-03-27
GB2231330B (en) 1992-04-29
ES2019840A6 (es) 1991-07-01
BE1004122A3 (fr) 1992-09-29
ATA95690A (de) 1994-08-15
GB8911030D0 (en) 1989-06-28
GR900100319A (en) 1991-10-10
DK102990A (da) 1990-11-14
CH681009A5 (en) 1992-12-31
CA2016551A1 (fr) 1990-11-13
KR900018113A (ko) 1990-12-20
IT9020276A0 (it) 1990-05-11
HK94992A (en) 1992-12-04
FR2646774A1 (fr) 1990-11-16
DE4015137A1 (de) 1990-11-15
PT94008A (pt) 1991-01-08
FR2646851B1 (fr) 1992-02-14
FR2646851A1 (fr) 1990-11-16
IT1240935B (it) 1993-12-27
CA2016551C (fr) 1997-09-09
JPH035484A (ja) 1991-01-11
NZ233574A (en) 1991-07-26
SE9001670L (fr)
IN174000B (fr) 1994-08-20
AR245725A1 (es) 1994-02-28
FR2646774B1 (fr) 1992-02-14
DZ1414A1 (fr) 2004-09-13
ZA903305B (en) 1991-02-27
IT9020276A1 (it) 1991-11-11
US5049559A (en) 1991-09-17
DK102990D0 (da) 1990-04-26
FI93119C (fi) 1995-02-27
DE4015137C2 (de) 2003-06-12
AU628171B2 (en) 1992-09-10
SE505407C2 (sv) 1997-08-25
FI93119B (fi) 1994-11-15
FI902355A0 (fi) 1990-05-11

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