NO171365C - Analogifremgangsmaate for fremstilling av terapeutisk aktive benzimidazolderivater - Google Patents
Analogifremgangsmaate for fremstilling av terapeutisk aktive benzimidazolderivaterInfo
- Publication number
- NO171365C NO171365C NO872686A NO872686A NO171365C NO 171365 C NO171365 C NO 171365C NO 872686 A NO872686 A NO 872686A NO 872686 A NO872686 A NO 872686A NO 171365 C NO171365 C NO 171365C
- Authority
- NO
- Norway
- Prior art keywords
- preparation
- therapeutic active
- analogy procedure
- benzimidazold
- derivatives
- Prior art date
Links
- 230000001225 therapeutic effect Effects 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 3
- 239000004480 active ingredient Substances 0.000 abstract 1
- 239000003814 drug Substances 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Medicines Containing Material From Animals Or Micro-Organisms (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicinal Preparation (AREA)
- Indole Compounds (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
SE8505112A SE8505112D0 (sv) | 1985-10-29 | 1985-10-29 | Novel pharmacological compounds |
PCT/SE1986/000493 WO1987002668A1 (en) | 1985-10-29 | 1986-10-28 | Novel pharmacological compounds |
Publications (4)
Publication Number | Publication Date |
---|---|
NO872686D0 NO872686D0 (no) | 1987-06-26 |
NO872686L NO872686L (no) | 1987-06-26 |
NO171365B NO171365B (no) | 1992-11-23 |
NO171365C true NO171365C (no) | 1993-03-03 |
Family
ID=20361960
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO872686A NO171365C (no) | 1985-10-29 | 1987-06-26 | Analogifremgangsmaate for fremstilling av terapeutisk aktive benzimidazolderivater |
Country Status (31)
Country | Link |
---|---|
US (1) | US5021433A (no) |
EP (2) | EP0221041A3 (no) |
JP (2) | JPH0780874B2 (no) |
KR (1) | KR950009858B1 (no) |
CN (1) | CN1022487C (no) |
AT (1) | ATE79619T1 (no) |
AU (1) | AU598491B2 (no) |
CS (1) | CS272767B2 (no) |
DD (1) | DD252375A5 (no) |
DE (1) | DE3686483T2 (no) |
DK (1) | DK320587D0 (no) |
EG (1) | EG17753A (no) |
ES (1) | ES2051696T3 (no) |
FI (1) | FI91151C (no) |
GR (1) | GR3006177T3 (no) |
HU (1) | HU198474B (no) |
IE (1) | IE59167B1 (no) |
IL (1) | IL80437A0 (no) |
IS (1) | IS1564B (no) |
JO (1) | JO1502B1 (no) |
LT (1) | LTIP1681A (no) |
LV (1) | LV10270B (no) |
MY (1) | MY101791A (no) |
NO (1) | NO171365C (no) |
NZ (1) | NZ218028A (no) |
PH (1) | PH25319A (no) |
PL (1) | PL150240B1 (no) |
PT (1) | PT83647B (no) |
SE (1) | SE8505112D0 (no) |
WO (1) | WO1987002668A1 (no) |
ZA (1) | ZA867716B (no) |
Families Citing this family (39)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
NZ234564A (en) * | 1986-11-21 | 1991-04-26 | Haessle Ab | 1-substituted benzimidazoles and pharmaceutical compositions |
EP0436025A4 (en) * | 1988-09-20 | 1991-09-11 | Hisamitsu Pharmaceutical Co. Inc. | Novel dibenz b,e)oxepin derivatives |
SE8804629D0 (sv) * | 1988-12-22 | 1988-12-22 | Ab Haessle | New therapeutically active compounds |
EG19302A (en) * | 1988-12-22 | 1994-11-30 | Haessle Ab | Compound with gastric acid inhibitory effect and process for its preparation |
US5274099A (en) * | 1989-12-20 | 1993-12-28 | Aktiebolaget Hassle | Therapeutically active fluoro substituted benzimidazoles |
US4965269A (en) * | 1989-12-20 | 1990-10-23 | Ab Hassle | Therapeutically active chloro substituted benzimidazoles |
US5049674A (en) * | 1989-12-20 | 1991-09-17 | Aktiebolaget Hassle | Therapeutically active fluoro substituted benzimidazoles |
SE9002206D0 (sv) * | 1990-06-20 | 1990-06-20 | Haessle Ab | New compounds |
PL166209B1 (pl) * | 1990-06-20 | 1995-04-28 | Astra Ab | Sposób wytwarzania nowych pochodnych benzimidazolu PL |
ES2048109B1 (es) * | 1992-07-20 | 1994-12-16 | Espanola Prod Quimicos | Procedimiento de preparacion de nuevos derivados piperidicos del bencimidazol. |
WO1995032957A1 (en) * | 1994-05-27 | 1995-12-07 | Astra Aktiebolag | Novel ethoxycarbonyloxymethyl derivatives of substituted benzimidazoles |
ATE231857T1 (de) | 1998-08-10 | 2003-02-15 | Winston Pharmateuticals Llc | Prodrugs für proton-pump-inhibitoren |
US6093734A (en) * | 1998-08-10 | 2000-07-25 | Partnership Of Michael E. Garst, George Sachs, And Jai Moo Shin | Prodrugs of proton pump inhibitors |
US6852739B1 (en) | 1999-02-26 | 2005-02-08 | Nitromed Inc. | Methods using proton pump inhibitors and nitric oxide donors |
US6369087B1 (en) * | 1999-08-26 | 2002-04-09 | Robert R. Whittle | Alkoxy substituted benzimidazole compounds, pharmaceutical preparations containing the same, and methods of using the same |
AU2001294228A1 (en) * | 2000-10-12 | 2002-04-22 | Takeda Chemical Industries Ltd. | Benzimidazole compounds, process for producing the same and use thereof |
WO2003027098A1 (fr) * | 2001-09-25 | 2003-04-03 | Takeda Chemical Industries, Ltd. | Compose de benzymidazole, procede de production et d'utilisation de celui-ci |
AU2003242390A1 (en) * | 2002-06-14 | 2003-12-31 | Takeda Pharmaceutical Company Limited | Prodrugs of imidazole derivatives, for use as proton pump inhibitors in the treatment of e.g. peptic ulcers |
KR100822981B1 (ko) * | 2002-07-19 | 2008-04-16 | 윈스턴 파마슈티컬즈, 엘엘씨 | 벤즈이미다졸 유도체 및 이들의 프로톤 펌프 억제제의프로드럭으로서의 이용 |
EP1534278A4 (en) | 2002-08-01 | 2006-09-06 | Nitromed Inc | NITROSED PROTONATE PUMP INHIBITORS, COMPOSITIONS AND USE METHOD |
MY148805A (en) | 2002-10-16 | 2013-05-31 | Takeda Pharmaceutical | Controlled release preparation |
EP2112920B1 (en) * | 2003-06-26 | 2018-07-25 | Intellipharmaceutics Corp. | Proton pump-inhibitor-containing capsules which comprise subunits differently structured for a delayed release of the active ingredient |
US20050075371A1 (en) * | 2003-10-03 | 2005-04-07 | Allergan, Inc. | Methods and compositions for the oral administration of prodrugs of proton pump inhibitors |
WO2005039640A1 (en) * | 2003-10-03 | 2005-05-06 | Allergan Inc. | Compositions comprising trefoil factor family peptides and/or mucoadhesives and proton pump inhibitor prodrugs |
US20070161679A1 (en) * | 2004-02-18 | 2007-07-12 | Allergan, Inc. | Method and compositions for the intravenous administration of compounds related to proton pump inhibitors |
EP1715861A2 (en) * | 2004-02-18 | 2006-11-02 | Allergan, Inc. | Compositions comprising prodrugs of proton pump inhibitors |
WO2005117870A2 (en) * | 2004-04-16 | 2005-12-15 | Santarus, Inc. | Combination of proton pump inhibitor, buffering agent, and prokinetic agent |
US7176319B2 (en) | 2004-04-28 | 2007-02-13 | Hetero Drugs Limited | Process for substituted sulfoxides |
WO2005116011A1 (en) * | 2004-05-28 | 2005-12-08 | Hetero Drugs Limited | A novel stereoselective synthesis of benzimidazole sulfoxides |
US8394409B2 (en) * | 2004-07-01 | 2013-03-12 | Intellipharmaceutics Corp. | Controlled extended drug release technology |
US10624858B2 (en) | 2004-08-23 | 2020-04-21 | Intellipharmaceutics Corp | Controlled release composition using transition coating, and method of preparing same |
US10064828B1 (en) | 2005-12-23 | 2018-09-04 | Intellipharmaceutics Corp. | Pulsed extended-pulsed and extended-pulsed pulsed drug delivery systems |
US9561188B2 (en) * | 2006-04-03 | 2017-02-07 | Intellipharmaceutics Corporation | Controlled release delivery device comprising an organosol coat |
US10960077B2 (en) | 2006-05-12 | 2021-03-30 | Intellipharmaceutics Corp. | Abuse and alcohol resistant drug composition |
WO2008036201A1 (en) * | 2006-09-19 | 2008-03-27 | Alevium Pharmaceuticals, Inc. | Prodrugs of proton pump inhibitors including the 1h-imidazo[4,5-b] pyridine moiety |
US20080103169A1 (en) | 2006-10-27 | 2008-05-01 | The Curators Of The University Of Missouri | Compositions comprising acid labile proton pump inhibiting agents, at least one other pharmaceutically active agent and methods of using same |
US20080194307A1 (en) * | 2007-02-13 | 2008-08-14 | Jeff Sanger | Sports-based game of chance |
WO2009105568A1 (en) | 2008-02-20 | 2009-08-27 | The Curators Of The University Of Missouri | Composition comprising a combination of omeprazole and lansoprazole, and a buffering agent, and methods of using same |
ES2768295T3 (es) * | 2010-01-07 | 2020-06-22 | Alkermes Pharma Ireland Ltd | Profármacos de compuestos heteroaromáticos |
Family Cites Families (23)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR320097A (fr) * | 1902-04-01 | 1902-12-01 | Betts | Perfectionnements dans et relatifs au raffinage électrolytique du plomb et des alliages de plomb |
FR1474663A (fr) * | 1966-04-06 | 1967-03-24 | Electrolyt Zinc Australasia | Procédé d'extraction de métaux |
US4026776A (en) * | 1970-12-02 | 1977-05-31 | Mitsui Mining & Smelting Co., Ltd. | Method for producing high purity lead |
SE418966B (sv) * | 1974-02-18 | 1981-07-06 | Haessle Ab | Analogiforfarande for framstellning av foreningar med magsyrasekretionsinhiberande verkan |
US4045564A (en) * | 1974-02-18 | 1977-08-30 | Ab Hassle | Benzimidazole derivatives useful as gastric acid secretion inhibitors |
US3960681A (en) * | 1974-02-21 | 1976-06-01 | Mitsui Mining & Smelting Co., Ltd. | Method for producing electrolytic high purity lead using large-sized electrodes |
SE416649B (sv) * | 1974-05-16 | 1981-01-26 | Haessle Ab | Forfarande for framstellning av foreningar som paverkar magsyrasekretionen |
NZ181123A (en) * | 1975-06-30 | 1979-12-11 | Univ Melbourne | Treatment of mineralcontaining materials with an acid in the presence of fluoride ion |
US3972790A (en) * | 1975-09-26 | 1976-08-03 | Uop Inc. | Production of metallic lead |
IN148930B (no) * | 1977-09-19 | 1981-07-25 | Hoffmann La Roche | |
US4189461A (en) * | 1977-11-30 | 1980-02-19 | Kennecott Copper Corporation | Metal leaching from concentrates using nitrogen dioxide in acids |
SE7804231L (sv) * | 1978-04-14 | 1979-10-15 | Haessle Ab | Magsyrasekretionsmedel |
FR2446863A1 (fr) * | 1979-01-22 | 1980-08-14 | Uop Inc | Procede perfectionne de recuperation de plomb |
FR2453906A1 (fr) * | 1979-04-12 | 1980-11-07 | Uop Inc | Procede de preparation hydrometallurgique de plomb a l'aide d'une extraction par voie electrochimique |
US4229271A (en) * | 1979-05-24 | 1980-10-21 | Rsr Corporation | Method of recovering lead values from battery sludge |
US4359465A (en) * | 1980-07-28 | 1982-11-16 | The Upjohn Company | Methods for treating gastrointestinal inflammation |
CH644116A5 (de) * | 1980-08-21 | 1984-07-13 | Hoffmann La Roche | Imidazolderivate. |
FR2505876A1 (en) * | 1981-05-12 | 1982-11-19 | Noual Patrick | Selective winning of lead from sulphide ores - by leaching with hot aq. hydro:fluorosilicic acid soln. contg. hydrogen peroxide and air so only lead is dissolved |
SE8300736D0 (sv) * | 1983-02-11 | 1983-02-11 | Haessle Ab | Novel pharmacologically active compounds |
IL75400A (en) * | 1984-06-16 | 1988-10-31 | Byk Gulden Lomberg Chem Fab | Dialkoxypyridine methyl(sulfinyl or sulfonyl)benzimidazoles,processes for the preparation thereof and pharmaceutical compositions containing the same |
US4500398A (en) * | 1984-06-20 | 1985-02-19 | The United States Of America As Represented By The Secretary Of The Interior | Production of lead from sulfides |
ZA856671B (en) * | 1984-09-24 | 1986-04-30 | Upjohn Co | N-substituted derivatives of 2-(pyridylaklenesulfinyl)benzimidazoles as gastric antisecretory agents |
AU568441B2 (en) * | 1984-09-24 | 1987-12-24 | Upjohn Company, The | 2-(pyridylalkenesulfinyl) benzimidazole derivatives |
-
1985
- 1985-10-29 SE SE8505112A patent/SE8505112D0/xx unknown
-
1986
- 1986-10-09 ZA ZA867716A patent/ZA867716B/xx unknown
- 1986-10-22 NZ NZ218028A patent/NZ218028A/xx unknown
- 1986-10-22 EG EG661/86A patent/EG17753A/xx active
- 1986-10-23 IE IE280586A patent/IE59167B1/en not_active IP Right Cessation
- 1986-10-24 PH PH34408A patent/PH25319A/en unknown
- 1986-10-27 DD DD86295633A patent/DD252375A5/de not_active IP Right Cessation
- 1986-10-27 JO JO19861502A patent/JO1502B1/en active
- 1986-10-27 MY MYPI86000038A patent/MY101791A/en unknown
- 1986-10-28 EP EP86850378A patent/EP0221041A3/en active Pending
- 1986-10-28 IS IS3156A patent/IS1564B/is unknown
- 1986-10-28 JP JP61505700A patent/JPH0780874B2/ja not_active Expired - Lifetime
- 1986-10-28 WO PCT/SE1986/000493 patent/WO1987002668A1/en active IP Right Grant
- 1986-10-28 EP EP86906498A patent/EP0233284B1/en not_active Expired - Lifetime
- 1986-10-28 AU AU65429/86A patent/AU598491B2/en not_active Ceased
- 1986-10-28 IL IL80437A patent/IL80437A0/xx not_active IP Right Cessation
- 1986-10-28 HU HU865443A patent/HU198474B/hu not_active IP Right Cessation
- 1986-10-28 AT AT86906498T patent/ATE79619T1/de not_active IP Right Cessation
- 1986-10-28 KR KR1019870700555A patent/KR950009858B1/ko active IP Right Grant
- 1986-10-28 DE DE8686906498T patent/DE3686483T2/de not_active Expired - Fee Related
- 1986-10-28 ES ES86906498T patent/ES2051696T3/es not_active Expired - Lifetime
- 1986-10-29 PL PL1986262105A patent/PL150240B1/pl unknown
- 1986-10-29 PT PT83647A patent/PT83647B/pt not_active IP Right Cessation
- 1986-10-29 CN CN86107595A patent/CN1022487C/zh not_active Expired - Lifetime
- 1986-10-29 CS CS782686A patent/CS272767B2/cs unknown
-
1987
- 1987-06-24 DK DK320587A patent/DK320587D0/da not_active Application Discontinuation
- 1987-06-26 NO NO872686A patent/NO171365C/no unknown
- 1987-06-29 FI FI872864A patent/FI91151C/sv not_active IP Right Cessation
-
1988
- 1988-05-12 US US07/195,343 patent/US5021433A/en not_active Expired - Fee Related
-
1992
- 1992-11-05 GR GR920402498T patent/GR3006177T3/el unknown
-
1993
- 1993-06-30 LV LVP-93-856A patent/LV10270B/xx unknown
- 1993-12-28 LT LTIP1681A patent/LTIP1681A/xx not_active Application Discontinuation
-
1994
- 1994-12-21 JP JP6318132A patent/JPH0826014B2/ja not_active Expired - Lifetime
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