NO170419C - Analogifremgangsmaate for fremstilling av 1h,3h-pyrrolo-(1,2-c)-tiazolderivater - Google Patents

Analogifremgangsmaate for fremstilling av 1h,3h-pyrrolo-(1,2-c)-tiazolderivater

Info

Publication number
NO170419C
NO170419C NO872779A NO872779A NO170419C NO 170419 C NO170419 C NO 170419C NO 872779 A NO872779 A NO 872779A NO 872779 A NO872779 A NO 872779A NO 170419 C NO170419 C NO 170419C
Authority
NO
Norway
Prior art keywords
group
alkyl
dipyridylcarbamoyl
dialkylsulphamido
alkylsulphamido
Prior art date
Application number
NO872779A
Other languages
English (en)
Norwegian (no)
Other versions
NO872779D0 (no
NO170419B (no
NO872779L (no
Inventor
Jean-Louis Fabre
Claude James
Daniel Lave
Original Assignee
Rhone Poulenc Sante
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Rhone Poulenc Sante filed Critical Rhone Poulenc Sante
Publication of NO872779D0 publication Critical patent/NO872779D0/no
Publication of NO872779L publication Critical patent/NO872779L/no
Publication of NO170419B publication Critical patent/NO170419B/no
Publication of NO170419C publication Critical patent/NO170419C/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D513/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Medicines Containing Plant Substances (AREA)
  • Steroid Compounds (AREA)
  • Pyrrole Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Medicinal Preparation (AREA)
NO872779A 1986-07-04 1987-07-02 Analogifremgangsmaate for fremstilling av 1h,3h-pyrrolo-(1,2-c)-tiazolderivater NO170419C (no)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR8609728A FR2601015B1 (fr) 1986-07-04 1986-07-04 Nouveaux derives du 1h,3h-pyrrolo (1,2-c) thiazole, leur preparation et les compositions pharmaceutiques qui les contiennent

Publications (4)

Publication Number Publication Date
NO872779D0 NO872779D0 (no) 1987-07-02
NO872779L NO872779L (no) 1988-01-05
NO170419B NO170419B (no) 1992-07-06
NO170419C true NO170419C (no) 1992-10-14

Family

ID=9337075

Family Applications (1)

Application Number Title Priority Date Filing Date
NO872779A NO170419C (no) 1986-07-04 1987-07-02 Analogifremgangsmaate for fremstilling av 1h,3h-pyrrolo-(1,2-c)-tiazolderivater

Country Status (28)

Country Link
US (1) US4783472A (fi)
EP (1) EP0253711B1 (fi)
JP (1) JPS6322589A (fi)
KR (1) KR880001681A (fi)
AT (1) ATE53037T1 (fi)
AU (1) AU597996B2 (fi)
BG (2) BG47498A3 (fi)
CA (1) CA1294966C (fi)
CS (1) CS262692B2 (fi)
DD (1) DD263772A5 (fi)
DE (1) DE3762861D1 (fi)
DK (1) DK340087A (fi)
ES (1) ES2015070B3 (fi)
FI (1) FI84727C (fi)
FR (1) FR2601015B1 (fi)
GR (1) GR3000502T3 (fi)
HU (1) HU198727B (fi)
IE (1) IE60743B1 (fi)
IL (1) IL83066A (fi)
MA (1) MA21027A1 (fi)
MX (1) MX173398B (fi)
NO (1) NO170419C (fi)
NZ (1) NZ220929A (fi)
PL (2) PL149903B1 (fi)
PT (1) PT85235B (fi)
SU (2) SU1528323A3 (fi)
TN (1) TNSN87083A1 (fi)
ZA (1) ZA874814B (fi)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2601016B1 (fr) * 1986-07-04 1988-10-07 Rhone Poulenc Sante Nouveaux derives du 1h,3h-pyrrolo (1,2-c) thiazole, leur preparation et les compositions pharmaceutiques qui les contiennent
FR2617484B1 (fr) * 1987-07-02 1989-10-20 Rhone Poulenc Sante Procede de preparation de l'acide (pyridyl-3)-3 1h-3h-pyrrolo (1,2-c) thiazolecarboxylique-7 dextrogyre
FR2644456B1 (fr) * 1989-03-17 1991-07-05 Rhone Poulenc Sante Nouveaux derives du 1h, 3h-pyrrolo(1,2-c)thiazolecarboxamide-7, leur preparation et les compositions pharmaceutiques qui les contiennent
JP3061631B2 (ja) * 1989-10-11 2000-07-10 山之内製薬株式会社 新規なヘテロ環化合物およびその製造法
FR2662606A1 (fr) * 1990-06-01 1991-12-06 Rhone Poulenc Sante Compositions pharmaceutiques pour le traitement de la fibrillation ventriculaire, du syndrome de menace de l'infarctus du myocarde et de l'angine de poitrine contenant le n-(benzoyl-3 phenyl) (pyridyl-3)-3 1h,3h-pyrrolo[1,2-c]thiazolecarboxamide-7.
FR2687574B1 (fr) * 1992-02-25 1995-05-05 Rhone Poulenc Rorer Sa Nouvelle application therapeutique de derives du pyridylpyrrolothiazole carboxamide.
GB9207645D0 (en) * 1992-04-08 1992-05-27 Smithkline Beecham Corp Methods
CA2470427C (en) * 2001-12-21 2012-07-10 Cytokinetics, Incorporated Compositions and methods for treating heart failure
CA2677096A1 (en) * 2007-01-31 2008-08-07 Vertex Pharmaceuticals Incorporated Kinase inhibitors
US8569337B2 (en) 2008-07-23 2013-10-29 Vertex Pharmaceuticals Incorporated Tri-cyclic pyrazolopyridine kinase inhibitors
AU2009274023A1 (en) 2008-07-23 2010-01-28 Vertex Pharmaceuticals Incorporated Tri-cyclic pyrazolopyridine kinase inhibitors
NZ590784A (en) 2008-07-23 2012-12-21 Vertex Pharma Pyrazolopyridine kinase inhibitors
JP2011530527A (ja) 2008-08-06 2011-12-22 バーテックス ファーマシューティカルズ インコーポレイテッド アミノピリジンキナーゼ阻害剤
AU2010245914A1 (en) 2009-05-06 2011-12-15 Vertex Pharmaceuticals Incorporated Pyrazolopyridines
JP5769733B2 (ja) 2010-01-27 2015-08-26 バーテックス ファーマシューティカルズ インコーポレイテッドVertex Pharmaceuticals Incorporated ピラゾロピリジンキナーゼ阻害剤
CN102869664A (zh) 2010-01-27 2013-01-09 沃泰克斯药物股份有限公司 吡唑并嘧啶类激酶抑制剂
EP2550272A1 (en) 2010-01-27 2013-01-30 Vertex Pharmaceuticals Incorporated Pyrazolopyrazine kinase inhibitors
KR102608281B1 (ko) * 2022-07-27 2023-12-01 김규현 감자를 이용한 맥주 제조 방법 및 이에 의해 제조된 감자 맥주

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2541280B1 (fr) * 1983-01-13 1985-06-21 Rhone Poulenc Sante Nouveaux derives du 1h, 3h-pyrrolo (1,2c) thiazolecarboxamide-7, leur preparation et les medicaments qui les contiennent
US4500532A (en) * 1983-03-03 1985-02-19 Usv Pharmaceutical Corporation 1-(Substituted aminoalkyl)-1,4-dihydropyridines
FR2601016B1 (fr) * 1986-07-04 1988-10-07 Rhone Poulenc Sante Nouveaux derives du 1h,3h-pyrrolo (1,2-c) thiazole, leur preparation et les compositions pharmaceutiques qui les contiennent

Also Published As

Publication number Publication date
DK340087D0 (da) 1987-07-02
FI872931A (fi) 1988-01-05
EP0253711A1 (fr) 1988-01-20
CS501387A2 (en) 1988-08-16
DD263772A5 (de) 1989-01-11
ES2015070B3 (es) 1990-08-01
NO872779D0 (no) 1987-07-02
PT85235B (pt) 1990-03-30
IL83066A0 (en) 1987-12-31
KR880001681A (ko) 1988-04-26
FI872931A0 (fi) 1987-07-02
ATE53037T1 (de) 1990-06-15
TNSN87083A1 (fr) 1990-01-01
FR2601015B1 (fr) 1988-08-05
NZ220929A (en) 1989-09-27
ZA874814B (en) 1988-03-30
IE60743B1 (en) 1994-08-10
FI84727B (fi) 1991-09-30
PT85235A (fr) 1987-08-01
EP0253711B1 (fr) 1990-05-23
US4783472A (en) 1988-11-08
PL149434B1 (en) 1990-02-28
JPS6322589A (ja) 1988-01-30
MX173398B (es) 1994-02-28
FI84727C (fi) 1992-01-10
BG47498A3 (en) 1990-07-16
NO170419B (no) 1992-07-06
PL149903B1 (en) 1990-03-31
HUT44791A (en) 1988-04-28
DK340087A (da) 1988-01-05
HU198727B (en) 1989-11-28
AU597996B2 (en) 1990-06-14
CS262692B2 (en) 1989-03-14
CA1294966C (fr) 1992-01-28
DE3762861D1 (de) 1990-06-28
GR3000502T3 (en) 1991-07-31
PL266582A1 (en) 1988-09-01
IL83066A (en) 1991-01-31
IE871767L (en) 1988-01-04
SU1588284A3 (ru) 1990-08-23
MX7191A (es) 1993-10-01
SU1528323A3 (ru) 1989-12-07
AU7504787A (en) 1988-01-07
NO872779L (no) 1988-01-05
BG47038A3 (en) 1990-04-16
MA21027A1 (fr) 1988-04-01
FR2601015A1 (fr) 1988-01-08

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