NO161373C - Analogifremgangsmaate for fremstilling av terapeutisk aktive pteridin-derivater. - Google Patents

Analogifremgangsmaate for fremstilling av terapeutisk aktive pteridin-derivater.

Info

Publication number
NO161373C
NO161373C NO854965A NO854965A NO161373C NO 161373 C NO161373 C NO 161373C NO 854965 A NO854965 A NO 854965A NO 854965 A NO854965 A NO 854965A NO 161373 C NO161373 C NO 161373C
Authority
NO
Norway
Prior art keywords
preparation
therapeutic active
pteridine derivatives
analogue procedure
active pteridine
Prior art date
Application number
NO854965A
Other languages
English (en)
Norwegian (no)
Other versions
NO854965L (no
NO161373B (no
Inventor
Josef Roch
Armin Heckel
Josef Nickl
Erich Mueller
Berthold Narr
Rainer Zimmermann
Hans Weisenberger
Original Assignee
Thomae Gmbh Dr K
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Thomae Gmbh Dr K filed Critical Thomae Gmbh Dr K
Publication of NO854965L publication Critical patent/NO854965L/no
Publication of NO161373B publication Critical patent/NO161373B/no
Publication of NO161373C publication Critical patent/NO161373C/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D475/00—Heterocyclic compounds containing pteridine ring systems
    • C07D475/06—Heterocyclic compounds containing pteridine ring systems with a nitrogen atom directly attached in position 4
    • C07D475/08—Heterocyclic compounds containing pteridine ring systems with a nitrogen atom directly attached in position 4 with a nitrogen atom directly attached in position 2
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
NO854965A 1984-12-12 1985-12-11 Analogifremgangsmaate for fremstilling av terapeutisk aktive pteridin-derivater. NO161373C (no)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19843445298 DE3445298A1 (de) 1984-12-12 1984-12-12 Neue pteridine, verfahren zu ihrer herstellung und deren verwendung als zwischenprodukte oder als arzneimittel

Publications (3)

Publication Number Publication Date
NO854965L NO854965L (no) 1986-06-13
NO161373B NO161373B (no) 1989-05-02
NO161373C true NO161373C (no) 1989-08-09

Family

ID=6252576

Family Applications (1)

Application Number Title Priority Date Filing Date
NO854965A NO161373C (no) 1984-12-12 1985-12-11 Analogifremgangsmaate for fremstilling av terapeutisk aktive pteridin-derivater.

Country Status (15)

Country Link
EP (1) EP0185259A3 (forum.php)
JP (1) JPS61140585A (forum.php)
AU (1) AU576924B2 (forum.php)
CA (1) CA1252783A (forum.php)
DE (1) DE3445298A1 (forum.php)
DK (1) DK161327C (forum.php)
ES (1) ES8707238A1 (forum.php)
FI (1) FI82696C (forum.php)
GR (1) GR852996B (forum.php)
IL (1) IL77294A (forum.php)
NO (1) NO161373C (forum.php)
NZ (1) NZ214522A (forum.php)
PH (1) PH24451A (forum.php)
PT (1) PT81650B (forum.php)
ZA (1) ZA859462B (forum.php)

Families Citing this family (24)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7276506B2 (en) 1998-12-28 2007-10-02 4 Aza Bioscience Nv Immunosuppressive effects of pteridine derivatives
CN1543465A (zh) * 2001-06-28 2004-11-03 ��������ҽѧ���޹�˾ 用作选择性细菌dhfr抑制剂的新的杂环化合物及其应用
DE10202468A1 (de) * 2002-01-23 2004-09-30 Faustus Forschungs Cie. Translational Cancer Research Gmbh Pteridinderivate, Verfahren zu deren Herstellung und ihre Verwendung
DK1658081T3 (da) * 2003-08-29 2008-02-25 4 Aza Ip Nv Immunsuppressive virkninger af pteridinderivater
PT1673092E (pt) * 2003-10-17 2007-11-23 4 Aza Ip Nv ''derivados de pteridina substituídos com heterociclos e sua utilização em terapia''
GB2407089A (en) * 2003-10-17 2005-04-20 4 Aza Bioscience Nv Pteridine derivatives
EP1720542A4 (en) * 2004-03-04 2007-11-28 Neurogen Corp ARYL ALKYLAMINO-SUBSTITUTED CHINAZOLINE ANALOGUE
DE102004057595A1 (de) 2004-11-29 2006-06-08 Boehringer Ingelheim Pharma Gmbh & Co. Kg Substituierte Pteridine zur Behandlung von entzündlichen Erkrankungen
DE102004057594A1 (de) 2004-11-29 2006-06-08 Boehringer Ingelheim Pharma Gmbh & Co. Kg Substitueirte Pteridine zur Behandlung von entzündlichen Erkrankungen
DE102004057645A1 (de) 2004-11-29 2006-06-01 Boehringer Ingelheim Pharma Gmbh & Co. Kg Substituierte Pteridine zur Behandlung von entzündlichen Erkrankungen
DE102004057618A1 (de) 2004-11-29 2006-06-01 Boehringer Ingelheim Pharma Gmbh & Co. Kg Substituierte Pteridine zur Behandlung von entzündlichen Erkrankungen
JP5161102B2 (ja) * 2005-11-22 2013-03-13 クドス ファーマシューティカルズ リミテッド ｍＴＯＲ阻害剤としてのピリドピリミジン、ピラゾピリミジンおよびピリミドピリミジン誘導体
RU2445315C2 (ru) * 2005-11-22 2012-03-20 Кудос Фармасьютиклз Лимитед ПРОИЗВОДНЫЕ ПИРИДО-, ПИРАЗО- И ПИРИМИДО-ПИРИМИДИНА И ИХ ПРИМЕНЕНИЕ В КАЧЕСТВЕ ИНГИБИТОРОВ mTOR
JP5440934B2 (ja) 2006-05-24 2014-03-12 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング 置換プテリジン
WO2008009078A2 (en) 2006-07-20 2008-01-24 Gilead Sciences, Inc. 4,6-dl- and 2,4,6-trisubstituted quinazoline derivatives useful for treating viral infections
US10144736B2 (en) 2006-07-20 2018-12-04 Gilead Sciences, Inc. Substituted pteridines useful for the treatment and prevention of viral infections
MX2009001946A (es) 2006-08-23 2009-03-05 Kudos Pharm Ltd Derivados de 2-metilmorfolin-pirido-, pirazo- y pirimido- pirimidina como inhibidores de mtor.
EP2303875B1 (en) 2008-06-20 2012-11-28 AstraZeneca AB Compositions with and process for methylmorpholin-subsituted pyrido[2,3-d]pyrimidines
KR102335970B1 (ko) 2015-03-04 2021-12-07 길리애드 사이언시즈, 인코포레이티드 톨 유사 수용체 조정제 화합물
US10370342B2 (en) 2016-09-02 2019-08-06 Gilead Sciences, Inc. Toll like receptor modulator compounds
ES2826748T3 (es) 2016-09-02 2021-05-19 Gilead Sciences Inc Derivados de 4,6-diamino-pirido[3,2-d]pirimidina como moduladores de receptores de tipo Toll
TWI751517B (zh) 2019-04-17 2022-01-01 美商基利科學股份有限公司 類鐸受體調節劑之固體形式
TW202210480A (zh) 2019-04-17 2022-03-16 美商基利科學股份有限公司 類鐸受體調節劑之固體形式
TWI879779B (zh) 2019-06-28 2025-04-11 美商基利科學股份有限公司 類鐸受體調節劑化合物的製備方法

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3159628A (en) * 1962-05-28 1964-12-01 Smith Kline French Lab Pteridine-5-oxide derivatives
DE3323932A1 (de) * 1983-07-02 1985-01-10 Dr. Karl Thomae Gmbh, 7950 Biberach Neue 2-piperazino-pteridine, verfahren zu ihrer herstellung und diese verbindung enthaltende arzneimittel

Also Published As

Publication number Publication date
AU5123285A (en) 1986-06-19
DK572685A (da) 1986-06-13
CA1252783A (en) 1989-04-18
PT81650B (pt) 1988-04-21
PH24451A (en) 1990-06-25
ZA859462B (en) 1987-07-29
FI854862A0 (fi) 1985-12-10
DE3445298A1 (de) 1986-06-12
PT81650A (de) 1986-01-01
EP0185259A3 (de) 1989-03-01
NO854965L (no) 1986-06-13
GR852996B (forum.php) 1986-04-16
ES8707238A1 (es) 1987-07-16
FI854862A7 (fi) 1986-06-13
FI82696B (fi) 1990-12-31
DK161327C (da) 1991-12-09
JPS61140585A (ja) 1986-06-27
DK572685D0 (da) 1985-12-11
DK161327B (da) 1991-06-24
ES549806A0 (es) 1987-07-16
EP0185259A2 (de) 1986-06-25
AU576924B2 (en) 1988-09-08
IL77294A (en) 1989-02-28
NO161373B (no) 1989-05-02
FI82696C (fi) 1991-04-10
NZ214522A (en) 1988-07-28

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