NO161373C - ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE PTERIDINE DERIVATIVES. - Google Patents

ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE PTERIDINE DERIVATIVES.

Info

Publication number
NO161373C
NO161373C NO854965A NO854965A NO161373C NO 161373 C NO161373 C NO 161373C NO 854965 A NO854965 A NO 854965A NO 854965 A NO854965 A NO 854965A NO 161373 C NO161373 C NO 161373C
Authority
NO
Norway
Prior art keywords
preparation
therapeutic active
pteridine derivatives
analogue procedure
active pteridine
Prior art date
Application number
NO854965A
Other languages
Norwegian (no)
Other versions
NO161373B (en
NO854965L (en
Inventor
Josef Roch
Armin Heckel
Josef Nickl
Erich Mueller
Berthold Narr
Rainer Zimmermann
Hans Weisenberger
Original Assignee
Thomae Gmbh Dr K
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Thomae Gmbh Dr K filed Critical Thomae Gmbh Dr K
Publication of NO854965L publication Critical patent/NO854965L/en
Publication of NO161373B publication Critical patent/NO161373B/en
Publication of NO161373C publication Critical patent/NO161373C/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D475/00Heterocyclic compounds containing pteridine ring systems
    • C07D475/06Heterocyclic compounds containing pteridine ring systems with a nitrogen atom directly attached in position 4
    • C07D475/08Heterocyclic compounds containing pteridine ring systems with a nitrogen atom directly attached in position 4 with a nitrogen atom directly attached in position 2
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
NO854965A 1984-12-12 1985-12-11 ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE PTERIDINE DERIVATIVES. NO161373C (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19843445298 DE3445298A1 (en) 1984-12-12 1984-12-12 NEW PTERIDINE, METHOD FOR THE PRODUCTION AND USE THEREOF AS INTERMEDIATE PRODUCTS OR AS A MEDICINAL PRODUCT

Publications (3)

Publication Number Publication Date
NO854965L NO854965L (en) 1986-06-13
NO161373B NO161373B (en) 1989-05-02
NO161373C true NO161373C (en) 1989-08-09

Family

ID=6252576

Family Applications (1)

Application Number Title Priority Date Filing Date
NO854965A NO161373C (en) 1984-12-12 1985-12-11 ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE PTERIDINE DERIVATIVES.

Country Status (15)

Country Link
EP (1) EP0185259A3 (en)
JP (1) JPS61140585A (en)
AU (1) AU576924B2 (en)
CA (1) CA1252783A (en)
DE (1) DE3445298A1 (en)
DK (1) DK161327C (en)
ES (1) ES8707238A1 (en)
FI (1) FI82696C (en)
GR (1) GR852996B (en)
IL (1) IL77294A (en)
NO (1) NO161373C (en)
NZ (1) NZ214522A (en)
PH (1) PH24451A (en)
PT (1) PT81650B (en)
ZA (1) ZA859462B (en)

Families Citing this family (23)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7276506B2 (en) 1998-12-28 2007-10-02 4 Aza Bioscience Nv Immunosuppressive effects of pteridine derivatives
SK302004A3 (en) * 2001-06-28 2005-07-01 Pliva, D.D. Heterocyclic compounds and use thereof as D-alanyl-D-alanine ligase inhibitors
DE10202468A1 (en) * 2002-01-23 2004-09-30 Faustus Forschungs Cie. Translational Cancer Research Gmbh Pteridine derivatives, process for their preparation and their use
ATE376421T1 (en) * 2003-08-29 2007-11-15 4 Aza Ip Nv IMMUNOSUPPRESSIVE EFFECTS OF PTERIDINE DERIVATIVES
GB2407089A (en) * 2003-10-17 2005-04-20 4 Aza Bioscience Nv Pteridine derivatives
AU2004283479A1 (en) * 2003-10-17 2005-05-06 4 Aza Bioscience Nv Heterocycle-substituted pteridine derivatives and their use in therapy
WO2005087227A1 (en) * 2004-03-04 2005-09-22 Neurogen Corporation Arylalkylamino-substituted quinazoline analogues
DE102004057594A1 (en) 2004-11-29 2006-06-08 Boehringer Ingelheim Pharma Gmbh & Co. Kg Substitute pteridine for the treatment of inflammatory diseases
DE102004057595A1 (en) 2004-11-29 2006-06-08 Boehringer Ingelheim Pharma Gmbh & Co. Kg Substituted pteridines for the treatment of inflammatory diseases
DE102004057645A1 (en) * 2004-11-29 2006-06-01 Boehringer Ingelheim Pharma Gmbh & Co. Kg New substituted pteridine compounds, useful as phosphodiesterase 4 inhibitors for treating e.g. inflammatory diseases, cancer, asthma, ulcerative colitis, depression and schizophrenia
DE102004057618A1 (en) 2004-11-29 2006-06-01 Boehringer Ingelheim Pharma Gmbh & Co. Kg Substituted pteridines for the treatment of inflammatory diseases
EP1954699B1 (en) * 2005-11-22 2012-09-19 Kudos Pharmaceuticals Ltd PYRIDO-, PYRAZO- AND PYRIMIDOPYRIMIDINE DERIVATIVES AS mTOR INHIBITORS
RU2445315C2 (en) * 2005-11-22 2012-03-20 Кудос Фармасьютиклз Лимитед PYRIDO-, PYRAZO- AND PYRIMIDO-PYRIMIDINE DERIVATIVES AND USE THEREOF AS mTOR INHIBITORS
EP2032585B1 (en) 2006-05-24 2014-07-23 Boehringer Ingelheim International GmbH Substituted pteridines as therapeutic agents
WO2008009079A2 (en) 2006-07-20 2008-01-24 Gilead Sciences, Inc. Substituted pteridines useful for the treatment and prevention of viral infections
MX2009001946A (en) 2006-08-23 2009-03-05 Kudos Pharm Ltd 2-methylmorpholine pyrido-, pyrazo- and pyrimido-pyrimidine derivatives as mtor inhibitors.
WO2009153597A2 (en) 2008-06-20 2009-12-23 Astrazeneca Ab Composition and process - 356
PL3097102T3 (en) 2015-03-04 2018-04-30 Gilead Sciences Inc Toll-like receptor modulating 4,6-diamino-pyrido[3,2-d]pyrimidine compounds
EP3507276B1 (en) 2016-09-02 2021-11-03 Gilead Sciences, Inc. Toll like receptor modulator compounds
EP3507288B1 (en) 2016-09-02 2020-08-26 Gilead Sciences, Inc. 4,6-diamino-pyrido[3,2-d]pyrimidine derivaties as toll like receptor modulators
TW202210480A (en) 2019-04-17 2022-03-16 美商基利科學股份有限公司 Solid forms of a toll-like receptor modulator
TW202212339A (en) 2019-04-17 2022-04-01 美商基利科學股份有限公司 Solid forms of a toll-like receptor modulator
TW202115056A (en) 2019-06-28 2021-04-16 美商基利科學股份有限公司 Processes for preparing toll-like receptor modulator compounds

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3159628A (en) * 1962-05-28 1964-12-01 Smith Kline French Lab Pteridine-5-oxide derivatives
DE3323932A1 (en) * 1983-07-02 1985-01-10 Dr. Karl Thomae Gmbh, 7950 Biberach NEW 2-PIPERAZINO-PTERIDINE, METHOD FOR THE PRODUCTION THEREOF AND MEDICINAL PRODUCTS CONTAINING THIS COMPOUND

Also Published As

Publication number Publication date
FI82696B (en) 1990-12-31
JPS61140585A (en) 1986-06-27
EP0185259A2 (en) 1986-06-25
EP0185259A3 (en) 1989-03-01
ES549806A0 (en) 1987-07-16
NZ214522A (en) 1988-07-28
AU5123285A (en) 1986-06-19
ZA859462B (en) 1987-07-29
DK161327B (en) 1991-06-24
IL77294A (en) 1989-02-28
NO161373B (en) 1989-05-02
FI854862A0 (en) 1985-12-10
DK572685D0 (en) 1985-12-11
PT81650A (en) 1986-01-01
CA1252783A (en) 1989-04-18
ES8707238A1 (en) 1987-07-16
FI854862A (en) 1986-06-13
AU576924B2 (en) 1988-09-08
PH24451A (en) 1990-06-25
DE3445298A1 (en) 1986-06-12
PT81650B (en) 1988-04-21
FI82696C (en) 1991-04-10
DK572685A (en) 1986-06-13
NO854965L (en) 1986-06-13
DK161327C (en) 1991-12-09
GR852996B (en) 1986-04-16

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