FI854862A0 - NYA PTERIDINER, FOERFARANDE FOER DERAS FRAMSTAELLNING OCH DERAS ANVAENDNING SAOSOM MELLANPRODUKTER ELLER SAOSOM LAEKEMEDEL. - Google Patents

NYA PTERIDINER, FOERFARANDE FOER DERAS FRAMSTAELLNING OCH DERAS ANVAENDNING SAOSOM MELLANPRODUKTER ELLER SAOSOM LAEKEMEDEL.

Info

Publication number
FI854862A0
FI854862A0 FI854862A FI854862A FI854862A0 FI 854862 A0 FI854862 A0 FI 854862A0 FI 854862 A FI854862 A FI 854862A FI 854862 A FI854862 A FI 854862A FI 854862 A0 FI854862 A0 FI 854862A0
Authority
FI
Finland
Prior art keywords
saosom
deras
pteridiner
nya
eller
Prior art date
Application number
FI854862A
Other languages
Finnish (fi)
Other versions
FI82696C (en
FI82696B (en
FI854862A (en
Inventor
Josef Roch
Armin Heckel
Josef Nickl
Erich Mueller
Berthold Narr
Rainer Zimmermann
Johannes Weisenberger
Original Assignee
Thomae Gmbh Dr K
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Thomae Gmbh Dr K filed Critical Thomae Gmbh Dr K
Publication of FI854862A0 publication Critical patent/FI854862A0/en
Publication of FI854862A publication Critical patent/FI854862A/en
Application granted granted Critical
Publication of FI82696B publication Critical patent/FI82696B/en
Publication of FI82696C publication Critical patent/FI82696C/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D475/00Heterocyclic compounds containing pteridine ring systems
    • C07D475/06Heterocyclic compounds containing pteridine ring systems with a nitrogen atom directly attached in position 4
    • C07D475/08Heterocyclic compounds containing pteridine ring systems with a nitrogen atom directly attached in position 4 with a nitrogen atom directly attached in position 2
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Hematology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
FI854862A 1984-12-12 1985-12-10 PROCEDURE FOR THE PREPARATION OF PHARMACOLOGICAL PROPERTIES OF PTERIDINER. FI82696C (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE19843445298 DE3445298A1 (en) 1984-12-12 1984-12-12 NEW PTERIDINE, METHOD FOR THE PRODUCTION AND USE THEREOF AS INTERMEDIATE PRODUCTS OR AS A MEDICINAL PRODUCT
DE3445298 1984-12-12

Publications (4)

Publication Number Publication Date
FI854862A0 true FI854862A0 (en) 1985-12-10
FI854862A FI854862A (en) 1986-06-13
FI82696B FI82696B (en) 1990-12-31
FI82696C FI82696C (en) 1991-04-10

Family

ID=6252576

Family Applications (1)

Application Number Title Priority Date Filing Date
FI854862A FI82696C (en) 1984-12-12 1985-12-10 PROCEDURE FOR THE PREPARATION OF PHARMACOLOGICAL PROPERTIES OF PTERIDINER.

Country Status (15)

Country Link
EP (1) EP0185259A3 (en)
JP (1) JPS61140585A (en)
AU (1) AU576924B2 (en)
CA (1) CA1252783A (en)
DE (1) DE3445298A1 (en)
DK (1) DK161327C (en)
ES (1) ES8707238A1 (en)
FI (1) FI82696C (en)
GR (1) GR852996B (en)
IL (1) IL77294A (en)
NO (1) NO161373C (en)
NZ (1) NZ214522A (en)
PH (1) PH24451A (en)
PT (1) PT81650B (en)
ZA (1) ZA859462B (en)

Families Citing this family (23)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7276506B2 (en) 1998-12-28 2007-10-02 4 Aza Bioscience Nv Immunosuppressive effects of pteridine derivatives
IL159538A0 (en) * 2001-06-28 2004-06-01 Pliva D D 8/17 heterocyclic compounds and uses thereof as d-alanyl-d-alanine ligase inhibitors
DE10202468A1 (en) * 2002-01-23 2004-09-30 Faustus Forschungs Cie. Translational Cancer Research Gmbh Pteridine derivatives, process for their preparation and their use
ATE376421T1 (en) * 2003-08-29 2007-11-15 4 Aza Ip Nv IMMUNOSUPPRESSIVE EFFECTS OF PTERIDINE DERIVATIVES
PT1673092E (en) * 2003-10-17 2007-11-23 4 Aza Ip Nv Heterocycle-substituted pteridine derivatives and their use in therapy
GB2407089A (en) * 2003-10-17 2005-04-20 4 Aza Bioscience Nv Pteridine derivatives
JP2007526323A (en) * 2004-03-04 2007-09-13 ニューロジェン・コーポレーション Arylalkylamino substituted quinazoline analogs
DE102004057645A1 (en) * 2004-11-29 2006-06-01 Boehringer Ingelheim Pharma Gmbh & Co. Kg New substituted pteridine compounds, useful as phosphodiesterase 4 inhibitors for treating e.g. inflammatory diseases, cancer, asthma, ulcerative colitis, depression and schizophrenia
DE102004057595A1 (en) 2004-11-29 2006-06-08 Boehringer Ingelheim Pharma Gmbh & Co. Kg Substituted pteridines for the treatment of inflammatory diseases
DE102004057618A1 (en) 2004-11-29 2006-06-01 Boehringer Ingelheim Pharma Gmbh & Co. Kg Substituted pteridines for the treatment of inflammatory diseases
DE102004057594A1 (en) 2004-11-29 2006-06-08 Boehringer Ingelheim Pharma Gmbh & Co. Kg Substitute pteridine for the treatment of inflammatory diseases
RU2445315C2 (en) * 2005-11-22 2012-03-20 Кудос Фармасьютиклз Лимитед PYRIDO-, PYRAZO- AND PYRIMIDO-PYRIMIDINE DERIVATIVES AND USE THEREOF AS mTOR INHIBITORS
AU2006318948B2 (en) * 2005-11-22 2011-02-24 Kudos Pharmaceuticals Limited Pyrido-,pyrazo- and pyrimido-pyrimidine derivatives as mTOR inhibitors
WO2007135026A2 (en) 2006-05-24 2007-11-29 Boehringer Ingelheim International Gmbh Substituted pteridines as therapeutic agents
US10144736B2 (en) 2006-07-20 2018-12-04 Gilead Sciences, Inc. Substituted pteridines useful for the treatment and prevention of viral infections
KR101438245B1 (en) 2006-08-23 2014-09-04 쿠도스 파마슈티칼스 리미티드 2-methylmorpholine pyrido-, pyrazo- and pyrimido-pyrimidine derivatives as mtor inhibitors
ES2398423T3 (en) 2008-06-20 2013-03-19 Astrazeneca Ab Compositions with and procedure for methylmorpholine substituted pyrimidines [2,3-D] pyrimidines
EP3097102B1 (en) 2015-03-04 2017-10-18 Gilead Sciences, Inc. Toll-like receptor modulating 4,6-diamino-pyrido[3,2-d]pyrimidine compounds
EP3507276B1 (en) 2016-09-02 2021-11-03 Gilead Sciences, Inc. Toll like receptor modulator compounds
US10640499B2 (en) 2016-09-02 2020-05-05 Gilead Sciences, Inc. Toll like receptor modulator compounds
TWI751517B (en) 2019-04-17 2022-01-01 美商基利科學股份有限公司 Solid forms of a toll-like receptor modulator
TWI751516B (en) 2019-04-17 2022-01-01 美商基利科學股份有限公司 Solid forms of a toll-like receptor modulator
TW202115056A (en) 2019-06-28 2021-04-16 美商基利科學股份有限公司 Processes for preparing toll-like receptor modulator compounds

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3159628A (en) * 1962-05-28 1964-12-01 Smith Kline French Lab Pteridine-5-oxide derivatives
DE3323932A1 (en) * 1983-07-02 1985-01-10 Dr. Karl Thomae Gmbh, 7950 Biberach NEW 2-PIPERAZINO-PTERIDINE, METHOD FOR THE PRODUCTION THEREOF AND MEDICINAL PRODUCTS CONTAINING THIS COMPOUND

Also Published As

Publication number Publication date
EP0185259A3 (en) 1989-03-01
PT81650A (en) 1986-01-01
FI82696C (en) 1991-04-10
IL77294A (en) 1989-02-28
NO161373C (en) 1989-08-09
AU576924B2 (en) 1988-09-08
CA1252783A (en) 1989-04-18
DE3445298A1 (en) 1986-06-12
GR852996B (en) 1986-04-16
NZ214522A (en) 1988-07-28
NO854965L (en) 1986-06-13
FI82696B (en) 1990-12-31
FI854862A (en) 1986-06-13
DK161327C (en) 1991-12-09
AU5123285A (en) 1986-06-19
PH24451A (en) 1990-06-25
JPS61140585A (en) 1986-06-27
PT81650B (en) 1988-04-21
EP0185259A2 (en) 1986-06-25
DK572685D0 (en) 1985-12-11
ES549806A0 (en) 1987-07-16
NO161373B (en) 1989-05-02
ES8707238A1 (en) 1987-07-16
DK572685A (en) 1986-06-13
DK161327B (en) 1991-06-24
ZA859462B (en) 1987-07-29

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Owner name: DR. KARL THOMAE GESELLSCHAFT MIT