FI854862A - NYA PTERIDINER, FOERFARANDE FOER DERAS FRAMSTAELLNING OCH DERAS ANVAENDNING SAOSOM MELLANPRODUKTER ELLER SAOSOM LAEKEMEDEL. - Google Patents
NYA PTERIDINER, FOERFARANDE FOER DERAS FRAMSTAELLNING OCH DERAS ANVAENDNING SAOSOM MELLANPRODUKTER ELLER SAOSOM LAEKEMEDEL. Download PDFInfo
- Publication number
- FI854862A FI854862A FI854862A FI854862A FI854862A FI 854862 A FI854862 A FI 854862A FI 854862 A FI854862 A FI 854862A FI 854862 A FI854862 A FI 854862A FI 854862 A FI854862 A FI 854862A
- Authority
- FI
- Finland
- Prior art keywords
- saosom
- deras
- pteridiner
- nya
- eller
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D475/00—Heterocyclic compounds containing pteridine ring systems
- C07D475/06—Heterocyclic compounds containing pteridine ring systems with a nitrogen atom directly attached in position 4
- C07D475/08—Heterocyclic compounds containing pteridine ring systems with a nitrogen atom directly attached in position 4 with a nitrogen atom directly attached in position 2
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE19843445298 DE3445298A1 (en) | 1984-12-12 | 1984-12-12 | NEW PTERIDINE, METHOD FOR THE PRODUCTION AND USE THEREOF AS INTERMEDIATE PRODUCTS OR AS A MEDICINAL PRODUCT |
DE3445298 | 1984-12-12 |
Publications (4)
Publication Number | Publication Date |
---|---|
FI854862A0 FI854862A0 (en) | 1985-12-10 |
FI854862A true FI854862A (en) | 1986-06-13 |
FI82696B FI82696B (en) | 1990-12-31 |
FI82696C FI82696C (en) | 1991-04-10 |
Family
ID=6252576
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FI854862A FI82696C (en) | 1984-12-12 | 1985-12-10 | PROCEDURE FOR THE PREPARATION OF PHARMACOLOGICAL PROPERTIES OF PTERIDINER. |
Country Status (15)
Country | Link |
---|---|
EP (1) | EP0185259A3 (en) |
JP (1) | JPS61140585A (en) |
AU (1) | AU576924B2 (en) |
CA (1) | CA1252783A (en) |
DE (1) | DE3445298A1 (en) |
DK (1) | DK161327C (en) |
ES (1) | ES8707238A1 (en) |
FI (1) | FI82696C (en) |
GR (1) | GR852996B (en) |
IL (1) | IL77294A (en) |
NO (1) | NO161373C (en) |
NZ (1) | NZ214522A (en) |
PH (1) | PH24451A (en) |
PT (1) | PT81650B (en) |
ZA (1) | ZA859462B (en) |
Families Citing this family (23)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US7276506B2 (en) | 1998-12-28 | 2007-10-02 | 4 Aza Bioscience Nv | Immunosuppressive effects of pteridine derivatives |
HUP0700061A2 (en) | 2001-06-28 | 2007-05-02 | Pliva D D | Pyridopyrimidine and pyrimidinopyrimidine derivatives, process for their preparation and pharmaceutical compositions therof as antibacterials having dhfr inhibitor activity |
DE10202468A1 (en) * | 2002-01-23 | 2004-09-30 | Faustus Forschungs Cie. Translational Cancer Research Gmbh | Pteridine derivatives, process for their preparation and their use |
AU2004267885A1 (en) * | 2003-08-29 | 2005-03-10 | 4 Aza Bioscience Nv | Immunosuppressive effects of pteridine derivatives |
GB2407089A (en) * | 2003-10-17 | 2005-04-20 | 4 Aza Bioscience Nv | Pteridine derivatives |
DK1673092T3 (en) * | 2003-10-17 | 2007-12-17 | 4 Aza Ip Nv | Heterocyclyl-substituted pteridine derivatives and their use in therapy |
CA2555867A1 (en) * | 2004-03-04 | 2005-09-22 | Neurogen Corporation | Arylalkylamino-substituted quinazoline analogues |
DE102004057645A1 (en) | 2004-11-29 | 2006-06-01 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | New substituted pteridine compounds, useful as phosphodiesterase 4 inhibitors for treating e.g. inflammatory diseases, cancer, asthma, ulcerative colitis, depression and schizophrenia |
DE102004057595A1 (en) | 2004-11-29 | 2006-06-08 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Substituted pteridines for the treatment of inflammatory diseases |
DE102004057618A1 (en) | 2004-11-29 | 2006-06-01 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Substituted pteridines for the treatment of inflammatory diseases |
DE102004057594A1 (en) * | 2004-11-29 | 2006-06-08 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Substitute pteridine for the treatment of inflammatory diseases |
PL1954699T3 (en) * | 2005-11-22 | 2013-01-31 | Kudos Pharm Ltd | PYRIDO-, PYRAZO- AND PYRIMIDOPYRIMIDINE DERIVATIVES AS mTOR INHIBITORS |
RU2445315C2 (en) * | 2005-11-22 | 2012-03-20 | Кудос Фармасьютиклз Лимитед | PYRIDO-, PYRAZO- AND PYRIMIDO-PYRIMIDINE DERIVATIVES AND USE THEREOF AS mTOR INHIBITORS |
JP5440934B2 (en) | 2006-05-24 | 2014-03-12 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | Substituted pteridine |
WO2008009079A2 (en) | 2006-07-20 | 2008-01-24 | Gilead Sciences, Inc. | Substituted pteridines useful for the treatment and prevention of viral infections |
KR101438245B1 (en) | 2006-08-23 | 2014-09-04 | 쿠도스 파마슈티칼스 리미티드 | 2-methylmorpholine pyrido-, pyrazo- and pyrimido-pyrimidine derivatives as mtor inhibitors |
CA2728183C (en) | 2008-06-20 | 2016-10-25 | Astrazeneca Ab | Compositions with and process for methylmorpholin-substituted pyrido [2,3-d] pryimidines |
KR102335970B1 (en) | 2015-03-04 | 2021-12-07 | 길리애드 사이언시즈, 인코포레이티드 | Toll like receptor modulator compounds |
CA3035346A1 (en) | 2016-09-02 | 2018-03-08 | Gilead Sciences, Inc. | Toll like receptor modulator compounds |
EP3507288B1 (en) | 2016-09-02 | 2020-08-26 | Gilead Sciences, Inc. | 4,6-diamino-pyrido[3,2-d]pyrimidine derivaties as toll like receptor modulators |
TWI751517B (en) | 2019-04-17 | 2022-01-01 | 美商基利科學股份有限公司 | Solid forms of a toll-like receptor modulator |
TW202210480A (en) | 2019-04-17 | 2022-03-16 | 美商基利科學股份有限公司 | Solid forms of a toll-like receptor modulator |
TW202115056A (en) | 2019-06-28 | 2021-04-16 | 美商基利科學股份有限公司 | Processes for preparing toll-like receptor modulator compounds |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3159628A (en) * | 1962-05-28 | 1964-12-01 | Smith Kline French Lab | Pteridine-5-oxide derivatives |
DE3323932A1 (en) * | 1983-07-02 | 1985-01-10 | Dr. Karl Thomae Gmbh, 7950 Biberach | NEW 2-PIPERAZINO-PTERIDINE, METHOD FOR THE PRODUCTION THEREOF AND MEDICINAL PRODUCTS CONTAINING THIS COMPOUND |
-
1984
- 1984-12-12 DE DE19843445298 patent/DE3445298A1/en not_active Withdrawn
-
1985
- 1985-12-05 EP EP85115459A patent/EP0185259A3/en not_active Ceased
- 1985-12-10 FI FI854862A patent/FI82696C/en not_active IP Right Cessation
- 1985-12-11 IL IL77294A patent/IL77294A/en unknown
- 1985-12-11 PT PT81650A patent/PT81650B/en not_active IP Right Cessation
- 1985-12-11 DK DK572685A patent/DK161327C/en not_active IP Right Cessation
- 1985-12-11 PH PH33161A patent/PH24451A/en unknown
- 1985-12-11 ZA ZA859462A patent/ZA859462B/en unknown
- 1985-12-11 NO NO854965A patent/NO161373C/en unknown
- 1985-12-11 ES ES549806A patent/ES8707238A1/en not_active Expired
- 1985-12-11 CA CA000497336A patent/CA1252783A/en not_active Expired
- 1985-12-11 NZ NZ214522A patent/NZ214522A/en unknown
- 1985-12-11 JP JP60278859A patent/JPS61140585A/en active Pending
- 1985-12-12 AU AU51232/85A patent/AU576924B2/en not_active Ceased
- 1985-12-12 GR GR852996A patent/GR852996B/el unknown
Also Published As
Publication number | Publication date |
---|---|
FI82696C (en) | 1991-04-10 |
ES549806A0 (en) | 1987-07-16 |
FI854862A0 (en) | 1985-12-10 |
ES8707238A1 (en) | 1987-07-16 |
NO161373C (en) | 1989-08-09 |
PT81650A (en) | 1986-01-01 |
JPS61140585A (en) | 1986-06-27 |
DK572685A (en) | 1986-06-13 |
AU5123285A (en) | 1986-06-19 |
PT81650B (en) | 1988-04-21 |
IL77294A (en) | 1989-02-28 |
NO854965L (en) | 1986-06-13 |
AU576924B2 (en) | 1988-09-08 |
PH24451A (en) | 1990-06-25 |
DK161327C (en) | 1991-12-09 |
EP0185259A2 (en) | 1986-06-25 |
EP0185259A3 (en) | 1989-03-01 |
DK161327B (en) | 1991-06-24 |
FI82696B (en) | 1990-12-31 |
DE3445298A1 (en) | 1986-06-12 |
ZA859462B (en) | 1987-07-29 |
GR852996B (en) | 1986-04-16 |
CA1252783A (en) | 1989-04-18 |
NZ214522A (en) | 1988-07-28 |
DK572685D0 (en) | 1985-12-11 |
NO161373B (en) | 1989-05-02 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
MM | Patent lapsed |
Owner name: DR. KARL THOMAE GESELLSCHAFT MIT |