DK161327C - SUBSTITUTED 2-PIPERAZINOPTERIDINES, PROCEDURES FOR PREPARING THEREOF, AND MEDICINALS CONTAINING THE COMPOUNDS - Google Patents

SUBSTITUTED 2-PIPERAZINOPTERIDINES, PROCEDURES FOR PREPARING THEREOF, AND MEDICINALS CONTAINING THE COMPOUNDS

Info

Publication number
DK161327C
DK161327C DK572685A DK572685A DK161327C DK 161327 C DK161327 C DK 161327C DK 572685 A DK572685 A DK 572685A DK 572685 A DK572685 A DK 572685A DK 161327 C DK161327 C DK 161327C
Authority
DK
Denmark
Prior art keywords
piperazinopteridines
procedures
substituted
preparing
compounds
Prior art date
Application number
DK572685A
Other languages
Danish (da)
Other versions
DK572685D0 (en
DK161327B (en
DK572685A (en
Inventor
Josef Roch
Armin Heckel
Josef Nickl
Erich Mueller
Berthold Narr
Rainer Zimmermann
Hans Weisenberger
Original Assignee
Thomae Gmbh Dr K
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Thomae Gmbh Dr K filed Critical Thomae Gmbh Dr K
Publication of DK572685D0 publication Critical patent/DK572685D0/en
Publication of DK572685A publication Critical patent/DK572685A/en
Publication of DK161327B publication Critical patent/DK161327B/en
Application granted granted Critical
Publication of DK161327C publication Critical patent/DK161327C/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D475/00—Heterocyclic compounds containing pteridine ring systems
    • C07D475/06—Heterocyclic compounds containing pteridine ring systems with a nitrogen atom directly attached in position 4
    • C07D475/08—Heterocyclic compounds containing pteridine ring systems with a nitrogen atom directly attached in position 4 with a nitrogen atom directly attached in position 2
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Hematology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
DK572685A 1984-12-12 1985-12-11 SUBSTITUTED 2-PIPERAZINOPTERIDINES, PROCEDURES FOR PREPARING THEREOF, AND MEDICINALS CONTAINING THE COMPOUNDS DK161327C (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE3445298 1984-12-12
DE19843445298 DE3445298A1 (en) 1984-12-12 1984-12-12 NEW PTERIDINE, METHOD FOR THE PRODUCTION AND USE THEREOF AS INTERMEDIATE PRODUCTS OR AS A MEDICINAL PRODUCT

Publications (4)

Publication Number Publication Date
DK572685D0 DK572685D0 (en) 1985-12-11
DK572685A DK572685A (en) 1986-06-13
DK161327B DK161327B (en) 1991-06-24
DK161327C true DK161327C (en) 1991-12-09

Family

ID=6252576

Family Applications (1)

Application Number Title Priority Date Filing Date
DK572685A DK161327C (en) 1984-12-12 1985-12-11 SUBSTITUTED 2-PIPERAZINOPTERIDINES, PROCEDURES FOR PREPARING THEREOF, AND MEDICINALS CONTAINING THE COMPOUNDS

Country Status (15)

Country Link
EP (1) EP0185259A3 (en)
JP (1) JPS61140585A (en)
AU (1) AU576924B2 (en)
CA (1) CA1252783A (en)
DE (1) DE3445298A1 (en)
DK (1) DK161327C (en)
ES (1) ES8707238A1 (en)
FI (1) FI82696C (en)
GR (1) GR852996B (en)
IL (1) IL77294A (en)
NO (1) NO161373C (en)
NZ (1) NZ214522A (en)
PH (1) PH24451A (en)
PT (1) PT81650B (en)
ZA (1) ZA859462B (en)

Families Citing this family (24)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7276506B2 (en) 1998-12-28 2007-10-02 4 Aza Bioscience Nv Immunosuppressive effects of pteridine derivatives
WO2003001887A2 (en) 2001-06-28 2003-01-09 Essential Therapeutics, Inc. Fused pyrimidines as d-alanyl-d-alanine ligase inhibitors
DE10202468A1 (en) * 2002-01-23 2004-09-30 Faustus Forschungs Cie. Translational Cancer Research Gmbh Pteridine derivatives, process for their preparation and their use
DE602004009696T2 (en) * 2003-08-29 2008-08-28 4 Aza Ip Nv IMMUNOSUPPRESSIVE EFFECTS OF PTERIDINE DERIVATIVES
DE602004008312T2 (en) * 2003-10-17 2008-04-17 4 Aza Ip Nv Heterocyclic-substituted pteridine derivatives and their use in therapy
GB2407089A (en) * 2003-10-17 2005-04-20 4 Aza Bioscience Nv Pteridine derivatives
AU2005221614A1 (en) * 2004-03-04 2005-09-22 Neurogen Corporation Arylalkylamino-substituted quinazoline analogues
DE102004057645A1 (en) 2004-11-29 2006-06-01 Boehringer Ingelheim Pharma Gmbh & Co. Kg New substituted pteridine compounds, useful as phosphodiesterase 4 inhibitors for treating e.g. inflammatory diseases, cancer, asthma, ulcerative colitis, depression and schizophrenia
DE102004057595A1 (en) 2004-11-29 2006-06-08 Boehringer Ingelheim Pharma Gmbh & Co. Kg Substituted pteridines for the treatment of inflammatory diseases
DE102004057594A1 (en) 2004-11-29 2006-06-08 Boehringer Ingelheim Pharma Gmbh & Co. Kg Substitute pteridine for the treatment of inflammatory diseases
DE102004057618A1 (en) 2004-11-29 2006-06-01 Boehringer Ingelheim Pharma Gmbh & Co. Kg Substituted pteridines for the treatment of inflammatory diseases
WO2007060404A1 (en) * 2005-11-22 2007-05-31 Kudos Pharmaceuticals Limited PYRIDO-,PYRAZO- AND PYRIMIDO-PYRIMIDINE DERIVATIVES AS mTOR INHIBITORS
RU2445315C2 (en) * 2005-11-22 2012-03-20 Кудос Фармасьютиклз Лимитед PYRIDO-, PYRAZO- AND PYRIMIDO-PYRIMIDINE DERIVATIVES AND USE THEREOF AS mTOR INHIBITORS
JP5440934B2 (en) 2006-05-24 2014-03-12 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング Substituted pteridine
US10144736B2 (en) 2006-07-20 2018-12-04 Gilead Sciences, Inc. Substituted pteridines useful for the treatment and prevention of viral infections
WO2008009078A2 (en) 2006-07-20 2008-01-24 Gilead Sciences, Inc. 4,6-dl- and 2,4,6-trisubstituted quinazoline derivatives useful for treating viral infections
HUE033894T2 (en) 2006-08-23 2018-01-29 Kudos Pharm Ltd 2-methylmorpholine pyrido-,pyrazo- and pyrimido-pyrimidine derivatives as mtor inhibitors
MX2010014230A (en) 2008-06-20 2011-03-29 Astrazeneca Ab Compositions with and process for methylmorpholin-subsituted pyrido [2, 3-d] pyrimidines.
CA2978188C (en) 2015-03-04 2020-05-12 Gilead Sciences, Inc. Toll-like receptor modulating 4,6-diamino-pyrido[3,2-d]pyrimidine compounds
WO2018045144A1 (en) 2016-09-02 2018-03-08 Gilead Sciences, Inc. Toll like receptor modulator compounds
US10640499B2 (en) 2016-09-02 2020-05-05 Gilead Sciences, Inc. Toll like receptor modulator compounds
TW202210480A (en) 2019-04-17 2022-03-16 美商基利科學股份有限公司 Solid forms of a toll-like receptor modulator
TW202212339A (en) 2019-04-17 2022-04-01 美商基利科學股份有限公司 Solid forms of a toll-like receptor modulator
TW202115056A (en) 2019-06-28 2021-04-16 美商基利科學股份有限公司 Processes for preparing toll-like receptor modulator compounds

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3159628A (en) * 1962-05-28 1964-12-01 Smith Kline French Lab Pteridine-5-oxide derivatives
DE3323932A1 (en) * 1983-07-02 1985-01-10 Dr. Karl Thomae Gmbh, 7950 Biberach NEW 2-PIPERAZINO-PTERIDINE, METHOD FOR THE PRODUCTION THEREOF AND MEDICINAL PRODUCTS CONTAINING THIS COMPOUND

Also Published As

Publication number Publication date
NO161373B (en) 1989-05-02
AU5123285A (en) 1986-06-19
NO854965L (en) 1986-06-13
ZA859462B (en) 1987-07-29
FI82696C (en) 1991-04-10
PT81650B (en) 1988-04-21
NZ214522A (en) 1988-07-28
PH24451A (en) 1990-06-25
GR852996B (en) 1986-04-16
EP0185259A3 (en) 1989-03-01
AU576924B2 (en) 1988-09-08
PT81650A (en) 1986-01-01
CA1252783A (en) 1989-04-18
EP0185259A2 (en) 1986-06-25
NO161373C (en) 1989-08-09
DK572685D0 (en) 1985-12-11
DE3445298A1 (en) 1986-06-12
FI854862A (en) 1986-06-13
FI854862A0 (en) 1985-12-10
ES549806A0 (en) 1987-07-16
ES8707238A1 (en) 1987-07-16
IL77294A (en) 1989-02-28
FI82696B (en) 1990-12-31
DK161327B (en) 1991-06-24
DK572685A (en) 1986-06-13
JPS61140585A (en) 1986-06-27

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