NO162188C - ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE IMIDAZOKINOLINES. - Google Patents

ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE IMIDAZOKINOLINES.

Info

Publication number
NO162188C
NO162188C NO853099A NO853099A NO162188C NO 162188 C NO162188 C NO 162188C NO 853099 A NO853099 A NO 853099A NO 853099 A NO853099 A NO 853099A NO 162188 C NO162188 C NO 162188C
Authority
NO
Norway
Prior art keywords
imidazokinolines
preparation
therapeutic active
analogue procedure
analogue
Prior art date
Application number
NO853099A
Other languages
Norwegian (no)
Other versions
NO853099L (en
NO162188B (en
Inventor
Pascal George
Danielle De Peretti
Original Assignee
Synthelabo
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Synthelabo filed Critical Synthelabo
Publication of NO853099L publication Critical patent/NO853099L/en
Publication of NO162188B publication Critical patent/NO162188B/en
Publication of NO162188C publication Critical patent/NO162188C/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/08Antiepileptics; Anticonvulsants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Pain & Pain Management (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Anesthesiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
NO853099A 1984-08-07 1985-08-06 ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE IMIDAZOKINOLINES. NO162188C (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR8412446A FR2568879B1 (en) 1984-08-07 1984-08-07 IMIDAZO (1,2-A) QUINOLINES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION

Publications (3)

Publication Number Publication Date
NO853099L NO853099L (en) 1986-02-10
NO162188B NO162188B (en) 1989-08-14
NO162188C true NO162188C (en) 1989-11-29

Family

ID=9306855

Family Applications (1)

Application Number Title Priority Date Filing Date
NO853099A NO162188C (en) 1984-08-07 1985-08-06 ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE IMIDAZOKINOLINES.

Country Status (20)

Country Link
EP (1) EP0172097B1 (en)
JP (1) JPS6147484A (en)
KR (1) KR860001814A (en)
AR (1) AR240674A1 (en)
AT (1) ATE41001T1 (en)
AU (1) AU573880B2 (en)
CA (1) CA1263389A (en)
DE (1) DE3568430D1 (en)
DK (1) DK161963B (en)
ES (1) ES8604593A1 (en)
FI (1) FI79314C (en)
FR (1) FR2568879B1 (en)
GR (1) GR851929B (en)
HU (1) HU199838B (en)
IL (1) IL76019A0 (en)
MX (1) MX161035A (en)
NO (1) NO162188C (en)
NZ (1) NZ213014A (en)
PT (1) PT80920B (en)
ZA (1) ZA855937B (en)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2593179B1 (en) * 1986-01-22 1988-04-01 Synthelabo IMIDAZO (1,2-A) QUINOLEINS DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION
FR2606410B1 (en) * 1986-11-07 1989-02-24 Synthelabo IMIDAZOPYRIDINES, THEIR PREPARATION AND THEIR APPLICATION IN THERAPEUTICS
FR2700547B1 (en) * 1993-01-15 1995-02-17 Synthelabo Imidazo [2,1-b] benzoselenazole-3-acetamide derivatives, their preparation and their therapeutic use.
FR2700544B1 (en) * 1993-01-15 1995-02-17 Synthelabo 9H-imidazo [1,2-a] benzimidazole-3-acetamide derivatives, their preparation and their therapeutic use.
FR2707987B1 (en) * 1993-07-22 1995-09-08 Synthelabo 9H-imidazo [1,2-a] benzimidazole-3-acetamide derivatives, their preparation and their therapeutic use.
EP0607076A1 (en) * 1993-01-15 1994-07-20 Synthelabo 9H-Imidazo 1,2-a benzimidazole derivatives with GABA activity
FR2719843B1 (en) * 1994-05-10 1996-06-07 Synthelabo Derivatives of 5,6-dihydro-4h-imidazo [2 ', 1': 2,3] imidazo- [4,5,1-ij] quinoline and 4,5-dihydroimidazo [1,2-a] pyrrolo- [1,2,3-cd] benzimidazole, their preparation and their therapeutic application.
FR2722501B1 (en) * 1994-07-13 1996-08-09 Synthelabo 9H-IMIDAZO (1,2-A) BENZIMIDAZOLE-3-ACETAMIDE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2492382A1 (en) * 1980-10-22 1982-04-23 Synthelabo IMIDAZO (1,2-A) PYRIDINE DERIVATIVES, THEIR PREPARATION AND THERAPEUTIC USE THEREOF

Also Published As

Publication number Publication date
DK356985D0 (en) 1985-08-06
KR860001814A (en) 1986-03-22
FI853027L (en) 1986-02-08
AR240674A1 (en) 1990-08-31
DK161963B (en) 1991-09-02
ES545929A0 (en) 1986-02-01
FI79314C (en) 1989-12-11
IL76019A0 (en) 1985-12-31
AU573880B2 (en) 1988-06-23
DK356985A (en) 1986-02-08
MX161035A (en) 1990-07-11
ES8604593A1 (en) 1986-02-01
FI79314B (en) 1989-08-31
NO853099L (en) 1986-02-10
AU4581485A (en) 1986-02-13
FI853027A0 (en) 1985-08-06
FR2568879B1 (en) 1986-12-12
GR851929B (en) 1985-12-09
ATE41001T1 (en) 1989-03-15
EP0172097B1 (en) 1989-03-01
NO162188B (en) 1989-08-14
HUT38636A (en) 1986-06-30
CA1263389A (en) 1989-11-28
FR2568879A1 (en) 1986-02-14
EP0172097A1 (en) 1986-02-19
PT80920B (en) 1987-12-30
DE3568430D1 (en) 1989-04-06
JPS6147484A (en) 1986-03-07
NZ213014A (en) 1988-05-30
PT80920A (en) 1985-09-01
ZA855937B (en) 1986-03-26
HU199838B (en) 1990-03-28

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