DK572685D0 - Hidtil ukendte pteridiner, deres fremstilling og anvendelse - Google Patents

Hidtil ukendte pteridiner, deres fremstilling og anvendelse

Info

Publication number
DK572685D0
DK572685D0 DK572685A DK572685A DK572685D0 DK 572685 D0 DK572685 D0 DK 572685D0 DK 572685 A DK572685 A DK 572685A DK 572685 A DK572685 A DK 572685A DK 572685 D0 DK572685 D0 DK 572685D0
Authority
DK
Denmark
Prior art keywords
pteridines
unknown
preparation
unknown pteridines
Prior art date
Application number
DK572685A
Other languages
English (en)
Other versions
DK161327B (da
DK161327C (da
DK572685A (da
Inventor
Josef Roch
Armin Heckel
Josef Nickl
Erich Mueller
Berthold Narr
Rainer Zimmermann
Weisenberger Hans
Original Assignee
Thomae Gmbh Dr K
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Thomae Gmbh Dr K filed Critical Thomae Gmbh Dr K
Publication of DK572685D0 publication Critical patent/DK572685D0/da
Publication of DK572685A publication Critical patent/DK572685A/da
Publication of DK161327B publication Critical patent/DK161327B/da
Application granted granted Critical
Publication of DK161327C publication Critical patent/DK161327C/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D475/00Heterocyclic compounds containing pteridine ring systems
    • C07D475/06Heterocyclic compounds containing pteridine ring systems with a nitrogen atom directly attached in position 4
    • C07D475/08Heterocyclic compounds containing pteridine ring systems with a nitrogen atom directly attached in position 4 with a nitrogen atom directly attached in position 2
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
DK572685A 1984-12-12 1985-12-11 Substituerede 2-piperazinopteridiner, fremgangsmaade til fremstilling deraf samt laegemidler indeholdende forbindelserne DK161327C (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE3445298 1984-12-12
DE19843445298 DE3445298A1 (de) 1984-12-12 1984-12-12 Neue pteridine, verfahren zu ihrer herstellung und deren verwendung als zwischenprodukte oder als arzneimittel

Publications (4)

Publication Number Publication Date
DK572685D0 true DK572685D0 (da) 1985-12-11
DK572685A DK572685A (da) 1986-06-13
DK161327B DK161327B (da) 1991-06-24
DK161327C DK161327C (da) 1991-12-09

Family

ID=6252576

Family Applications (1)

Application Number Title Priority Date Filing Date
DK572685A DK161327C (da) 1984-12-12 1985-12-11 Substituerede 2-piperazinopteridiner, fremgangsmaade til fremstilling deraf samt laegemidler indeholdende forbindelserne

Country Status (15)

Country Link
EP (1) EP0185259A3 (da)
JP (1) JPS61140585A (da)
AU (1) AU576924B2 (da)
CA (1) CA1252783A (da)
DE (1) DE3445298A1 (da)
DK (1) DK161327C (da)
ES (1) ES8707238A1 (da)
FI (1) FI82696C (da)
GR (1) GR852996B (da)
IL (1) IL77294A (da)
NO (1) NO161373C (da)
NZ (1) NZ214522A (da)
PH (1) PH24451A (da)
PT (1) PT81650B (da)
ZA (1) ZA859462B (da)

Families Citing this family (23)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7276506B2 (en) 1998-12-28 2007-10-02 4 Aza Bioscience Nv Immunosuppressive effects of pteridine derivatives
CN1543465A (zh) * 2001-06-28 2004-11-03 ��������ҽѧ���޹�˾ 用作选择性细菌dhfr抑制剂的新的杂环化合物及其应用
DE10202468A1 (de) * 2002-01-23 2004-09-30 Faustus Forschungs Cie. Translational Cancer Research Gmbh Pteridinderivate, Verfahren zu deren Herstellung und ihre Verwendung
EP1658081B1 (en) * 2003-08-29 2007-10-24 4 Aza Ip Nv Immunosuppressive effects of pteridine derivatives
WO2005039587A1 (en) * 2003-10-17 2005-05-06 4 Aza Bioscience Nv Heterocycle-substituted pteridine derivatives and their use in therapy
GB2407089A (en) * 2003-10-17 2005-04-20 4 Aza Bioscience Nv Pteridine derivatives
JP2007526323A (ja) * 2004-03-04 2007-09-13 ニューロジェン・コーポレーション アリールアルキルアミノ置換キナゾリン類縁体
DE102004057595A1 (de) 2004-11-29 2006-06-08 Boehringer Ingelheim Pharma Gmbh & Co. Kg Substituierte Pteridine zur Behandlung von entzündlichen Erkrankungen
DE102004057594A1 (de) 2004-11-29 2006-06-08 Boehringer Ingelheim Pharma Gmbh & Co. Kg Substitueirte Pteridine zur Behandlung von entzündlichen Erkrankungen
DE102004057618A1 (de) 2004-11-29 2006-06-01 Boehringer Ingelheim Pharma Gmbh & Co. Kg Substituierte Pteridine zur Behandlung von entzündlichen Erkrankungen
DE102004057645A1 (de) * 2004-11-29 2006-06-01 Boehringer Ingelheim Pharma Gmbh & Co. Kg Substituierte Pteridine zur Behandlung von entzündlichen Erkrankungen
CA2628920C (en) * 2005-11-22 2015-12-29 Kudos Pharmaceuticals Limited Pyrido-,pyrazo- and pyrimido-pyrimidine derivatives as mtor inhibitors
RU2445315C2 (ru) * 2005-11-22 2012-03-20 Кудос Фармасьютиклз Лимитед ПРОИЗВОДНЫЕ ПИРИДО-, ПИРАЗО- И ПИРИМИДО-ПИРИМИДИНА И ИХ ПРИМЕНЕНИЕ В КАЧЕСТВЕ ИНГИБИТОРОВ mTOR
WO2007135026A2 (de) 2006-05-24 2007-11-29 Boehringer Ingelheim International Gmbh Substituierte pteridine als therapeutika
US10144736B2 (en) 2006-07-20 2018-12-04 Gilead Sciences, Inc. Substituted pteridines useful for the treatment and prevention of viral infections
MY148688A (en) 2006-08-23 2013-05-31 Kudos Pharm Ltd 2-methylmorpholine pyrido-, pyrazo- and pyrimido-pyrimidine derivatives as mtor inhibitors
AU2009261688B2 (en) 2008-06-20 2012-07-05 Astrazeneca Ab Compositions with and process for methylmorpholin-substituted pyrido [2,3-D] pyrimidines
EP3722297A1 (en) 2015-03-04 2020-10-14 Gilead Sciences, Inc. Toll-like receptor modulating 4,6-diamino-pyrido[3,2-d]pyrimidine compounds
WO2018045150A1 (en) 2016-09-02 2018-03-08 Gilead Sciences, Inc. 4,6-diamino-pyrido[3,2-d]pyrimidine derivaties as toll like receptor modulators
AU2017318601B2 (en) 2016-09-02 2020-09-03 Gilead Sciences, Inc. Toll like receptor modulator compounds
TWI751517B (zh) 2019-04-17 2022-01-01 美商基利科學股份有限公司 類鐸受體調節劑之固體形式
TW202210480A (zh) 2019-04-17 2022-03-16 美商基利科學股份有限公司 類鐸受體調節劑之固體形式
TW202115056A (zh) 2019-06-28 2021-04-16 美商基利科學股份有限公司 類鐸受體調節劑化合物的製備方法

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3159628A (en) * 1962-05-28 1964-12-01 Smith Kline French Lab Pteridine-5-oxide derivatives
DE3323932A1 (de) * 1983-07-02 1985-01-10 Dr. Karl Thomae Gmbh, 7950 Biberach Neue 2-piperazino-pteridine, verfahren zu ihrer herstellung und diese verbindung enthaltende arzneimittel

Also Published As

Publication number Publication date
DK161327B (da) 1991-06-24
FI854862A0 (fi) 1985-12-10
IL77294A (en) 1989-02-28
EP0185259A2 (de) 1986-06-25
ES8707238A1 (es) 1987-07-16
PH24451A (en) 1990-06-25
DK161327C (da) 1991-12-09
NZ214522A (en) 1988-07-28
PT81650B (pt) 1988-04-21
NO161373B (no) 1989-05-02
CA1252783A (en) 1989-04-18
ZA859462B (en) 1987-07-29
GR852996B (da) 1986-04-16
DK572685A (da) 1986-06-13
JPS61140585A (ja) 1986-06-27
EP0185259A3 (de) 1989-03-01
FI854862A (fi) 1986-06-13
FI82696C (fi) 1991-04-10
NO161373C (no) 1989-08-09
AU576924B2 (en) 1988-09-08
ES549806A0 (es) 1987-07-16
AU5123285A (en) 1986-06-19
FI82696B (fi) 1990-12-31
NO854965L (no) 1986-06-13
PT81650A (de) 1986-01-01
DE3445298A1 (de) 1986-06-12

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