NL8202102A - Antracyclinen en werkwijze voor hun bereiding. - Google Patents

Antracyclinen en werkwijze voor hun bereiding. Download PDF

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Publication number
NL8202102A
NL8202102A NL8202102A NL8202102A NL8202102A NL 8202102 A NL8202102 A NL 8202102A NL 8202102 A NL8202102 A NL 8202102A NL 8202102 A NL8202102 A NL 8202102A NL 8202102 A NL8202102 A NL 8202102A
Authority
NL
Netherlands
Prior art keywords
formula
demethoxy
racemic
acid
mixture
Prior art date
Application number
NL8202102A
Other languages
English (en)
Dutch (nl)
Original Assignee
Erba Farmitalia
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Erba Farmitalia filed Critical Erba Farmitalia
Publication of NL8202102A publication Critical patent/NL8202102A/nl

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20—Carbocyclic rings
    • C07H15/24—Condensed ring systems having three or more rings
    • C07H15/252—Naphthacene radicals, e.g. daunomycins, adriamycins
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C50/00—Quinones
    • C07C50/38—Quinones containing —CHO or non—quinoid keto groups
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
NL8202102A 1981-05-28 1982-05-21 Antracyclinen en werkwijze voor hun bereiding. NL8202102A (nl)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
GB8116264 1981-05-28
GB8116264 1981-05-28
GB8125949 1981-08-22
GB8125949 1981-08-22

Publications (1)

Publication Number Publication Date
NL8202102A true NL8202102A (nl) 1982-12-16

Family

ID=26279611

Family Applications (1)

Application Number Title Priority Date Filing Date
NL8202102A NL8202102A (nl) 1981-05-28 1982-05-21 Antracyclinen en werkwijze voor hun bereiding.

Country Status (16)

Country Link
US (2) US4465671A (it)
AU (2) AU564016B2 (it)
CA (1) CA1210390A (it)
CH (1) CH652131A5 (it)
DE (2) DE3249834C2 (it)
DK (1) DK239382A (it)
FI (1) FI75833C (it)
FR (2) FR2506772B1 (it)
GB (1) GB2100257B (it)
HU (2) HU190015B (it)
IE (1) IE53120B1 (it)
IL (1) IL65858A (it)
IT (1) IT1210476B (it)
NL (1) NL8202102A (it)
SE (2) SE458685B (it)
YU (2) YU113082A (it)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5138042A (en) * 1981-05-28 1992-08-11 Farmitalia Carlo Erba S.P.A. 6-deoxyanthracyclines
GB8317037D0 (en) * 1983-06-23 1983-07-27 Erba Farmitalia 6-deoxyanthracyclines
IT1210476B (it) * 1981-05-28 1989-09-14 Erba Farmitalia Antracicline.
DE3233020A1 (de) * 1981-09-18 1983-04-07 Farmitalia Carlo Erba S.p.A., 20159 Milano Verfahren zur herstellung von 4-demethoxy-7,9-dideoxydaunomycinon
IT1155446B (it) * 1982-12-23 1987-01-28 Erba Farmitalia Procedimento per la purificazione di glucosidi antraciclinonici mediante adsobimento selettivo su resine
DE3422735C2 (de) * 1983-06-23 1996-07-11 Erba Carlo Spa Anthracyclinglykoside, Verfahren zu deren Herstellung und Arzneimittel, welche diese enthalten
FR2560600B1 (fr) * 1983-06-23 1988-01-15 Erba Farmitalia Glycosides d'anthracyclines, procede pour les preparer, medicament les contenant
FR2551057B1 (fr) * 1983-08-30 1986-07-18 Hoechst Lab Nouveaux aglycones utiles pour la preparation des antibiotiques et des antitumoraux de la serie des anthracyclines et leurs procedes de preparation
GB8421491D0 (en) * 1984-08-24 1984-09-26 Erba Farmitalia Anthracycline glycosides
GB8426672D0 (en) * 1984-10-22 1984-11-28 Erba Farmitalia Pharmaceutical compositions
US4634765A (en) * 1984-12-18 1987-01-06 Merrell Dow Pharmaceuticals Inc. Homodisaccharide hypoglycemic agents
GB2182926B (en) * 1985-11-19 1989-10-04 Erba Farmitalia Nitro anthracyclines, process for their preparation and use thereof
GB8905668D0 (en) * 1989-03-13 1989-04-26 Erba Carlo Spa New 3'-(4-morpholinyl)-and 3'-(2-methoxy-4-morpholinyl)-anthracycline derivatives
US5948896A (en) * 1997-08-13 1999-09-07 Gem Pharmaceuticals Processes for preparing 13-deoxy anthracycline derivatives
US5942605A (en) * 1998-03-03 1999-08-24 Gem Pharmaceuticals, Inc. 5-imino-13-deoxy anthracycline derivatives, their uses, and processes for preparing them

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE44954C (de) * FARBENFABRIKEN VORM. FRIEDR. BAYER & CO. in Elberfeld Verfahren zur Darstellung gelbbis rothbrauner, im alkalischen Bade färbender Azofarbstoffe aus Chrysoidin
GB1467383A (en) * 1974-06-12 1977-03-16 Farmaceutici Italia Daunomycin analogues
NL7900869A (nl) * 1978-02-09 1979-08-13 Erba Farmitalia Anthracyclinenantibiotica.
IT1098212B (it) * 1978-05-09 1985-09-07 Farmaceutici Italia Antracioline antitumorali sostituite
JPS5756494A (en) * 1980-09-22 1982-04-05 Microbial Chem Res Found New anthracyclin derivative
IT1210476B (it) * 1981-05-28 1989-09-14 Erba Farmitalia Antracicline.

Also Published As

Publication number Publication date
AU576684B2 (en) 1988-09-01
IL65858A (en) 1985-07-31
DK239382A (da) 1982-11-29
SE8203274L (sv) 1982-11-29
YU191984A (en) 1985-04-30
DE3219380A1 (de) 1982-12-16
IL65858A0 (en) 1982-08-31
AU8412782A (en) 1982-12-02
FI821833A0 (fi) 1982-05-24
SE8704116L (sv) 1987-10-22
AU564016B2 (en) 1987-07-30
IE821260L (en) 1982-11-28
GB2100257A (en) 1982-12-22
AU6173186A (en) 1987-01-08
FI75833B (fi) 1988-04-29
IT8220606A0 (it) 1982-04-06
FR2514754A1 (it) 1983-04-22
SE8704116D0 (sv) 1987-10-22
YU113082A (en) 1985-04-30
DE3219380C2 (de) 1986-12-04
DE3249834C2 (it) 1989-08-03
US4465671A (en) 1984-08-14
FR2506772B1 (fr) 1985-10-18
CH652131A5 (de) 1985-10-31
GB2100257B (en) 1985-09-25
SE458685B (sv) 1989-04-24
FR2514754B1 (it) 1985-12-13
FR2506772A1 (fr) 1982-12-03
IT1210476B (it) 1989-09-14
CA1210390A (en) 1986-08-26
US4600537A (en) 1986-07-15
IE53120B1 (en) 1988-07-06
FI75833C (fi) 1988-08-08
HU190015B (en) 1986-08-28
HU199767B (en) 1990-03-28

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Legal Events

Date Code Title Description
A85 Still pending on 85-01-01
BA A request for search or an international-type search has been filed
BB A search report has been drawn up
BC A request for examination has been filed
BV The patent application has lapsed