NL7905810A - Werkwijze voor het bereiden van farmaceutisch preparaat op basis van een piperazinederivaat, dat actief is ten aanzien van het centrale zenuwstelsel en een pijnstil- lend middel is, werkwijze ter bereiding van het piperazinederivaat en het aldus bereide farmaceutische preparaat. - Google Patents

Werkwijze voor het bereiden van farmaceutisch preparaat op basis van een piperazinederivaat, dat actief is ten aanzien van het centrale zenuwstelsel en een pijnstil- lend middel is, werkwijze ter bereiding van het piperazinederivaat en het aldus bereide farmaceutische preparaat. Download PDF

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Publication number
NL7905810A
NL7905810A NL7905810A NL7905810A NL7905810A NL 7905810 A NL7905810 A NL 7905810A NL 7905810 A NL7905810 A NL 7905810A NL 7905810 A NL7905810 A NL 7905810A NL 7905810 A NL7905810 A NL 7905810A
Authority
NL
Netherlands
Prior art keywords
formula
radical
derivatives
preparing
piperazine derivative
Prior art date
Application number
NL7905810A
Other languages
English (en)
Dutch (nl)
Original Assignee
Synthelabo
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from FR7822672A external-priority patent/FR2432515A1/fr
Priority claimed from FR7833105A external-priority patent/FR2442234A2/fr
Application filed by Synthelabo filed Critical Synthelabo
Publication of NL7905810A publication Critical patent/NL7905810A/nl

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D295/00Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/04Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
    • C07D295/08Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms
    • C07D295/096Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms with the ring nitrogen atoms and the oxygen or sulfur atoms separated by carbocyclic rings or by carbon chains interrupted by carbocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/02Drugs for disorders of the nervous system for peripheral neuropathies
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/26Psychostimulants, e.g. nicotine, cocaine
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D295/00Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/04Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
    • C07D295/08Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms
    • C07D295/084Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms with the ring nitrogen atoms and the oxygen or sulfur atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings
    • C07D295/088Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms with the ring nitrogen atoms and the oxygen or sulfur atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings to an acyclic saturated chain

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
NL7905810A 1978-08-01 1979-07-27 Werkwijze voor het bereiden van farmaceutisch preparaat op basis van een piperazinederivaat, dat actief is ten aanzien van het centrale zenuwstelsel en een pijnstil- lend middel is, werkwijze ter bereiding van het piperazinederivaat en het aldus bereide farmaceutische preparaat. NL7905810A (nl)

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
FR7822672A FR2432515A1 (fr) 1978-08-01 1978-08-01 Derives de phenyl-1 piperazine et leur application en therapeutique
FR7822672 1978-08-01
FR7833105A FR2442234A2 (fr) 1978-08-01 1978-11-23 Derives de phenyl-1 piperazine et leur application en therapeutique
FR7833105 1978-11-23
FR7916029A FR2459797A2 (fr) 1978-08-01 1979-06-22 Derives de phenyl-1 piperazine et leur application en therapeutique
FR7916029 1979-06-22

Publications (1)

Publication Number Publication Date
NL7905810A true NL7905810A (nl) 1980-02-05

Family

ID=27250847

Family Applications (1)

Application Number Title Priority Date Filing Date
NL7905810A NL7905810A (nl) 1978-08-01 1979-07-27 Werkwijze voor het bereiden van farmaceutisch preparaat op basis van een piperazinederivaat, dat actief is ten aanzien van het centrale zenuwstelsel en een pijnstil- lend middel is, werkwijze ter bereiding van het piperazinederivaat en het aldus bereide farmaceutische preparaat.

Country Status (18)

Country Link
JP (1) JPS5522690A (da)
AU (1) AU4930979A (da)
BE (1) BE877994A (da)
DE (1) DE2930440A1 (da)
DK (1) DK321479A (da)
ES (1) ES483003A1 (da)
FI (1) FI792401A7 (da)
FR (1) FR2459797A2 (da)
GB (1) GB2027703A (da)
GR (1) GR69703B (da)
IL (1) IL57920A0 (da)
IT (1) IT1123497B (da)
LU (1) LU81562A1 (da)
NL (1) NL7905810A (da)
NO (1) NO792502L (da)
NZ (1) NZ191140A (da)
PT (1) PT70007A (da)
SE (1) SE7906507L (da)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2582288B1 (fr) * 1985-05-21 1987-08-07 Massonnet Henry Poubelle compacteuse perfectionnee
SE9904723D0 (sv) 1999-12-22 1999-12-22 Carlsson A Research Ab New modulators of dopamine neurotransmission II
USRE46117E1 (en) 1999-12-22 2016-08-23 Teva Pharmaceuticals International Gmbh Modulators of dopamine neurotransmission
SE9904724D0 (sv) * 1999-12-22 1999-12-22 Carlsson A Research Ab New modulators of dopamine neurotransmission I
DE602005021641D1 (de) 2004-06-08 2010-07-15 Nsab, Filial Af Neurosearch Sweden Ab Neue disubstituierte phenylpiperidine und piperazine als modulatoren der dopamin-neurotransmission
JP2008501749A (ja) 2004-06-08 2008-01-24 ニューロサーチ スウェーデン アクチボラゲット ドーパミン及びセロトニン神経伝達のモジュレーターとしての新規なジ置換フェニルピペリジン
US7851629B2 (en) 2004-06-08 2010-12-14 Nsab, Filial Af Neurosearch Sweden Ab, Sverige Disubstituted phenylpiperidines as modulators of dopamine and serotonin neurotransmission
CA2584831C (en) 2004-10-13 2013-09-17 Neurosearch Sweden Ab Process for the synthesis of 4-(3-methanesulfonylphenyl)-1-n-propyl-piperidine
SE529246C2 (sv) 2005-10-13 2007-06-12 Neurosearch Sweden Ab Nya disubstituerade fenyl-piperidiner som modulatorer för dopaminneurotransmission
MX347209B (es) 2011-12-08 2017-04-19 Teva Pharmaceuticals Int Gmbh La sal de bromhidrato de pridopidina.

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH353743A (fr) * 1955-06-29 1961-04-30 Parke Davis & Co Procédé de préparation de pipérazines
US2976290A (en) * 1959-04-24 1961-03-21 Parke Davis & Co Piperazine derivatives and methods for their production
FR2224464A1 (en) * 1973-04-05 1974-10-31 Synthelabo N-Phenyl-N'-beta-hydroxy-ethyl piperazines - as analgesic and anti-inflammatory agents

Also Published As

Publication number Publication date
DE2930440A1 (de) 1980-02-28
PT70007A (fr) 1979-08-01
AU4930979A (en) 1980-02-07
FI792401A7 (fi) 1981-01-01
FR2459797A2 (fr) 1981-01-16
BE877994A (fr) 1980-01-31
DK321479A (da) 1980-02-02
FR2459797B2 (da) 1982-05-14
GR69703B (da) 1982-07-09
LU81562A1 (fr) 1981-03-24
NZ191140A (en) 1981-01-23
GB2027703A (en) 1980-02-27
JPS5522690A (en) 1980-02-18
NO792502L (no) 1980-02-04
IT1123497B (it) 1986-04-30
IL57920A0 (en) 1979-11-30
ES483003A1 (es) 1980-04-16
IT7924749A0 (it) 1979-07-27
SE7906507L (sv) 1980-02-02

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