NL7207820A - - Google Patents

Info

Publication number
NL7207820A
NL7207820A NL7207820A NL7207820A NL7207820A NL 7207820 A NL7207820 A NL 7207820A NL 7207820 A NL7207820 A NL 7207820A NL 7207820 A NL7207820 A NL 7207820A NL 7207820 A NL7207820 A NL 7207820A
Authority
NL
Netherlands
Application number
NL7207820A
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Publication of NL7207820A publication Critical patent/NL7207820A/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C51/00—Preparation of carboxylic acids or their salts, halides or anhydrides
    • C07C51/16—Preparation of carboxylic acids or their salts, halides or anhydrides by oxidation
    • C07C51/31—Preparation of carboxylic acids or their salts, halides or anhydrides by oxidation of cyclic compounds with ring-splitting
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/87—Benzo [c] furans; Hydrogenated benzo [c] furans
    • C07D307/88—Benzo [c] furans; Hydrogenated benzo [c] furans with one oxygen atom directly attached in position 1 or 3
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D317/00—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms
    • C07D317/08—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3
    • C07D317/44—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D317/46—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • C07D317/48—Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring
    • C07D317/50—Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to atoms of the carbocyclic ring
    • C07D317/58—Radicals substituted by nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D333/72—Benzo[c]thiophenes; Hydrogenated benzo[c]thiophenes
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Cephalosporin Compounds (AREA)
NL7207820A 1971-06-09 1972-06-08 NL7207820A (cg-RX-API-DMAC7.html)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB1960471A GB1364672A (en) 1971-06-09 1971-06-09 Penicillins

Publications (1)

Publication Number Publication Date
NL7207820A true NL7207820A (cg-RX-API-DMAC7.html) 1972-12-12

Family

ID=10132139

Family Applications (2)

Application Number Title Priority Date Filing Date
NLAANVRAGE7207626,A NL178006C (nl) 1971-06-09 1972-06-05 Werkwijze voor het bereiden of vervaardigen van een antibacterieel werkend geneesmiddel, alsmede werkwijze voor het bereiden van een ester van 6-(d(-)-alfa-aminofenylaceetamido)penicillanzuur.
NL7207820A NL7207820A (cg-RX-API-DMAC7.html) 1971-06-09 1972-06-08

Family Applications Before (1)

Application Number Title Priority Date Filing Date
NLAANVRAGE7207626,A NL178006C (nl) 1971-06-09 1972-06-05 Werkwijze voor het bereiden of vervaardigen van een antibacterieel werkend geneesmiddel, alsmede werkwijze voor het bereiden van een ester van 6-(d(-)-alfa-aminofenylaceetamido)penicillanzuur.

Country Status (33)

Country Link
US (7) US3860579A (cg-RX-API-DMAC7.html)
JP (8) JPS5235678B1 (cg-RX-API-DMAC7.html)
AR (2) AR192944A1 (cg-RX-API-DMAC7.html)
AT (4) AT317427B (cg-RX-API-DMAC7.html)
AU (2) AU476038B2 (cg-RX-API-DMAC7.html)
BE (2) BE784698A (cg-RX-API-DMAC7.html)
CA (3) CA1126260A (cg-RX-API-DMAC7.html)
CH (4) CH605986A5 (cg-RX-API-DMAC7.html)
CS (1) CS198111B2 (cg-RX-API-DMAC7.html)
CY (1) CY861A (cg-RX-API-DMAC7.html)
DD (1) DD99802A5 (cg-RX-API-DMAC7.html)
DE (2) DE2228012C3 (cg-RX-API-DMAC7.html)
DK (1) DK140597B (cg-RX-API-DMAC7.html)
ES (4) ES403667A1 (cg-RX-API-DMAC7.html)
FI (3) FI58642C (cg-RX-API-DMAC7.html)
FR (3) FR2140617B1 (cg-RX-API-DMAC7.html)
GB (1) GB1364672A (cg-RX-API-DMAC7.html)
HK (1) HK71676A (cg-RX-API-DMAC7.html)
HU (1) HU166360B (cg-RX-API-DMAC7.html)
IE (3) IE37758B1 (cg-RX-API-DMAC7.html)
IL (3) IL39772A (cg-RX-API-DMAC7.html)
IS (1) IS923B6 (cg-RX-API-DMAC7.html)
KE (2) KE2631A (cg-RX-API-DMAC7.html)
MY (2) MY7600195A (cg-RX-API-DMAC7.html)
NL (2) NL178006C (cg-RX-API-DMAC7.html)
NO (1) NO144169C (cg-RX-API-DMAC7.html)
OA (1) OA04101A (cg-RX-API-DMAC7.html)
PL (2) PL87735B1 (cg-RX-API-DMAC7.html)
SE (7) SE432102B (cg-RX-API-DMAC7.html)
SU (2) SU507244A3 (cg-RX-API-DMAC7.html)
YU (2) YU36029B (cg-RX-API-DMAC7.html)
ZA (2) ZA723800B (cg-RX-API-DMAC7.html)
ZM (1) ZM9172A1 (cg-RX-API-DMAC7.html)

Families Citing this family (30)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1377661A (en) * 1971-06-05 1974-12-18 Yamanouchi Pharma Co Ltd Oxofuryl ester derivatives of penicillin and cephalosporin
GB1364672A (en) * 1971-06-09 1974-08-29 Beecham Group Ltd Penicillins
GB1450043A (en) * 1972-09-08 1976-09-22 Beecham Group Ltd Penicillins
US4092476A (en) * 1974-02-21 1978-05-30 Beecham Group Limited Phthalidyl esters of 7-[(α amino, 2 substituted acetamido)-3-(heterocyclic-thio methyl)]cephalosporins
US4115646A (en) * 1975-02-22 1978-09-19 Beecham Group Limited Process for preparing 7-aminocephalosporanic acid derivatives
GB1565656A (en) * 1975-12-13 1980-04-23 Beecham Group Ltd Preparation of substituted penicillin acid esters
NZ189945A (en) * 1978-04-01 1981-04-24 Beecham Group Ltd Ampicillin phthalidyl ester naphthalene 2-sulphonate also pharmaceutical compositions
US4206218A (en) * 1978-08-31 1980-06-03 E. R. Squibb & Sons, Inc. Phthalidyl esters of the acetone adduct of epicillin
EP0014651B1 (fr) * 1979-02-05 1982-08-04 Sanofi S.A. 2-Méthoxyphénoxyacétate de talampicilline, procédé pour sa préparation et médicaments le renfermant
DE3001590A1 (de) * 1980-01-11 1981-07-23 E.R. Squibb & Sons, Inc., 08540 Princeton, N.J. Phthalidylester des aceton-addukts von epicillin und diese verbindungen enthaltende arzneimittel
US4340539A (en) * 1980-01-21 1982-07-20 Bristol-Myers Company Derivatives of 6-bromo penicillanic acid
IT1130969B (it) * 1980-03-14 1986-06-18 Dob Far Spa Esteri della cefapirina,loro sali e procedimento per il loro ottenimento
CA1212105A (en) 1980-04-30 1986-09-30 Shoji Ikeda Ampicillin esters and production thereof
IT1190897B (it) * 1982-06-29 1988-02-24 Opos Biochimica Srl Procedimento per la preparazione dell'estere 1-etossicarbonilossietilico dell'acido 6-(d(-)-alfa aminoalfa fenilacetamido)-penicillanico
GB2157284B (en) * 1984-04-11 1987-11-04 Leo Pharm Prod Ltd 6-b-halopenicillanic acid salts
IT1180207B (it) * 1984-07-30 1987-09-23 Istituto Biochimico Italiano Procedimento per la preparazione, con resa e purezza elevate, di antibiotici beta-lattamici
US4675210A (en) * 1984-10-10 1987-06-23 Hercules Incorporated Maleic modified butene copolymers for adhering polypropylene
JPH01148353A (ja) * 1987-12-02 1989-06-09 Sadami Ujima 遠心脱水機
US5695473A (en) * 1994-07-27 1997-12-09 Sims Deltec, Inc. Occlusion detection system for an infusion pump
US7186855B2 (en) 2001-06-11 2007-03-06 Xenoport, Inc. Prodrugs of GABA analogs, compositions and uses thereof
AU2002310409C1 (en) 2001-06-11 2008-04-17 Xenoport, Inc. Orally administered dosage forms of GABA analog prodrugs having reduced toxicity
US8048917B2 (en) * 2005-04-06 2011-11-01 Xenoport, Inc. Prodrugs of GABA analogs, compositions and uses thereof
US7232924B2 (en) * 2001-06-11 2007-06-19 Xenoport, Inc. Methods for synthesis of acyloxyalkyl derivatives of GABA analogs
US6818787B2 (en) * 2001-06-11 2004-11-16 Xenoport, Inc. Prodrugs of GABA analogs, compositions and uses thereof
AU2004267100B2 (en) * 2003-08-20 2010-10-07 Xenoport, Inc. Acyloxyalkyl carbamate prodrugs, methods of synthesis and use
EP2354120A1 (en) 2003-08-20 2011-08-10 XenoPort, Inc. Synthesis of acyloxyalkyl carbamate prodrugs and intermediates thereof
EP1811986B1 (en) * 2004-11-04 2014-03-26 XenoPort, Inc. Gabapentin prodrug sustained release oral dosage forms
EP1919859B1 (en) 2005-06-20 2010-06-02 Xenoport, Inc. Acyloxyalkyl carbamate prodrugs of tranexamic acid and use
WO2011028234A1 (en) * 2009-09-04 2011-03-10 Xenoport, Inc. Uses of acyloxyalkyl carbamate prodrugs of tranexamic acid
WO2011091164A1 (en) * 2010-01-22 2011-07-28 Xenoport, Inc. Oral dosage forms having a high loading of a tranexamic acid prodrug

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2985648A (en) * 1958-10-06 1961-05-23 Doyle Frank Peter Alpha-aminobenzylpenicillins
US3652546A (en) * 1965-07-22 1972-03-28 Bristol Myers Co Esters of 6-aminopenicillanic acid
GB1175590A (en) * 1967-08-09 1969-12-23 Beecham Group Ltd Therapeutic Compositions
US3697507A (en) * 1968-09-26 1972-10-10 Leo Pharm Prod Ltd Esters of {60 -aminobenzylpenicillin
FR2020209A1 (en) * 1968-10-09 1970-07-10 Sarath Antibiotic acylxymethyl 7-(alpha-amino-alpha-phenyl- - acetamido)-3-methyl-delta-3-cephem-4-carboxylates
GB1234426A (cg-RX-API-DMAC7.html) * 1968-10-23 1971-06-03
IE34019B1 (en) * 1969-03-18 1975-01-08 Leo Pharm Prod Ltd New semi-synthetic penicillin esters
BE754141A (fr) * 1969-08-04 1971-02-01 Pfizer Esters d'alpha-carboxyarylmethyl penicillines
BE758782A (fr) * 1969-11-11 1971-05-10 Leo Pharm Prod Ltd Nouveaux derives d'acide 6-amidino penicillanique leur procede de preparation et leurs applications comme antibiotiques
US3726861A (en) * 1971-06-03 1973-04-10 American Home Prod Ureido derivatives of 6-aminopenicillanic acid saccharimide
GB1377661A (en) * 1971-06-05 1974-12-18 Yamanouchi Pharma Co Ltd Oxofuryl ester derivatives of penicillin and cephalosporin
GB1364672A (en) * 1971-06-09 1974-08-29 Beecham Group Ltd Penicillins

Also Published As

Publication number Publication date
BE784699A (fr) 1972-12-11
ES431087A1 (es) 1976-11-01
CH605986A5 (cg-RX-API-DMAC7.html) 1978-10-13
SE433939B (sv) 1984-06-25
USRE29650E (en) 1978-05-30
IE36461L (en) 1972-12-09
PL96668B1 (pl) 1978-01-31
CA1131620A (en) 1982-09-14
CA1126260A (en) 1982-06-22
US3919196A (en) 1975-11-11
IS923B6 (is) 1976-03-30
JPS5659780A (en) 1981-05-23
ES403667A1 (es) 1976-01-01
FR2299857B1 (cg-RX-API-DMAC7.html) 1978-11-17
IE37758B1 (en) 1977-10-12
SU578887A3 (ru) 1977-10-30
DE2228012C3 (de) 1980-01-17
ZM9172A1 (en) 1973-01-22
IE37757L (en) 1972-12-09
NL7207626A (cg-RX-API-DMAC7.html) 1972-12-12
IL39771A (en) 1975-12-31
JPS5253889A (en) 1977-04-30
DE2228255C2 (de) 1983-12-08
IL39772A0 (en) 1972-08-30
JPS5235678B1 (cg-RX-API-DMAC7.html) 1977-09-10
PL87735B1 (en) 1976-07-31
FI792791A7 (fi) 1981-01-01
AT318147B (de) 1974-09-25
GB1364672A (en) 1974-08-29
SU507244A3 (ru) 1976-03-15
IL39771A0 (en) 1972-08-30
AT320155B (de) 1975-01-27
HK71676A (en) 1976-11-26
YU36029B (en) 1981-11-13
FR2299857A1 (fr) 1976-09-03
MY7600196A (en) 1976-12-31
NO144169C (no) 1981-07-08
YU186679A (en) 1981-11-13
SE390415B (sv) 1976-12-20
ES403672A1 (es) 1975-07-01
ZA723799B (en) 1973-03-28
MY7600195A (en) 1976-12-31
DE2228012B2 (de) 1979-05-23
US4036829A (en) 1977-07-19
US3963702A (en) 1976-06-15
CS198111B2 (en) 1980-05-30
CH577514A5 (cg-RX-API-DMAC7.html) 1976-07-15
IS2078A7 (is) 1972-12-10
AU476038B2 (en) 1976-09-09
AR192944A1 (es) 1973-03-21
FR2140617A1 (cg-RX-API-DMAC7.html) 1973-01-19
SE430606B (sv) 1983-11-28
KE2631A (en) 1976-06-11
SE430605B (sv) 1983-11-28
JPS6021593B2 (ja) 1985-05-28
FR2140616B1 (cg-RX-API-DMAC7.html) 1976-08-20
SE7809241L (sv) 1978-09-01
US3963704A (en) 1976-06-15
YU153772A (en) 1981-04-30
AU4331372A (en) 1973-12-13
DK140597C (cg-RX-API-DMAC7.html) 1980-02-25
US3860579A (en) 1975-01-14
FI792790A7 (fi) 1981-01-01
FR2140617B1 (cg-RX-API-DMAC7.html) 1976-07-02
JPS5253886A (en) 1977-04-30
AT317427B (de) 1974-08-26
AT318806B (de) 1974-11-25
JPS5659779A (en) 1981-05-23
SE7809236L (sv) 1978-09-01
SE7809237L (sv) 1978-09-01
YU36377B (en) 1983-06-30
IE36461B1 (en) 1976-11-10
OA04101A (fr) 1979-11-15
SE433938B (sv) 1984-06-25
DD99802A5 (cg-RX-API-DMAC7.html) 1973-08-20
IE37757B1 (en) 1977-10-12
US3939180A (en) 1976-02-17
FR2140616A1 (cg-RX-API-DMAC7.html) 1973-01-19
ZA723800B (en) 1973-03-28
AR193581A1 (es) 1973-04-30
SE7600561L (sv) 1976-01-20
JPS5253888A (en) 1977-04-30
DK140597B (da) 1979-10-08
JPS6021594B2 (ja) 1985-05-28
AU4331472A (en) 1973-12-13
NL178006B (nl) 1985-08-01
FI58642C (fi) 1981-03-10
IL47578A (en) 1975-12-31
SE432102B (sv) 1984-03-19
NL178006C (nl) 1986-01-02
KE2632A (en) 1976-06-11
AU463395B2 (en) 1975-07-24
CH587267A5 (cg-RX-API-DMAC7.html) 1977-04-29
CA1126258A (en) 1982-06-22
SE7600562L (sv) 1976-01-20
CY861A (en) 1976-12-17
JPS602310B1 (cg-RX-API-DMAC7.html) 1985-01-21
NO144169B (no) 1981-03-30
DE2228012A1 (de) 1972-12-28
FI58642B (fi) 1980-11-28
CH587265A5 (cg-RX-API-DMAC7.html) 1977-04-29
IL39772A (en) 1977-03-31
BE784698A (fr) 1972-12-11
DE2228255A1 (de) 1972-12-28
ES431086A1 (es) 1976-11-01
JPS5253887A (en) 1977-04-30
HU166360B (cg-RX-API-DMAC7.html) 1975-03-28

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Legal Events

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