MY142423A - Substituted aminoacetyl pyrrolidine compounds which are dipeptidyl peptidase iv inhibitors, and pharmaceutical compositions containing them - Google Patents
Substituted aminoacetyl pyrrolidine compounds which are dipeptidyl peptidase iv inhibitors, and pharmaceutical compositions containing themInfo
- Publication number
- MY142423A MY142423A MYPI20054654A MYPI20054654A MY142423A MY 142423 A MY142423 A MY 142423A MY PI20054654 A MYPI20054654 A MY PI20054654A MY PI20054654 A MYPI20054654 A MY PI20054654A MY 142423 A MY142423 A MY 142423A
- Authority
- MY
- Malaysia
- Prior art keywords
- inhibitors
- pharmaceutical compositions
- compositions containing
- dipeptidyl peptidase
- substituted
- Prior art date
Links
- 229940124213 Dipeptidyl peptidase 4 (DPP IV) inhibitor Drugs 0.000 title abstract 2
- 239000003603 dipeptidyl peptidase IV inhibitor Substances 0.000 title abstract 2
- 239000008194 pharmaceutical composition Substances 0.000 title abstract 2
- SJNAQBNIUKINQH-UHFFFAOYSA-N 2-amino-1-pyrrolidin-1-ylethanone Chemical class NCC(=O)N1CCCC1 SJNAQBNIUKINQH-UHFFFAOYSA-N 0.000 title 1
Classifications
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- C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
- C07D235/06—Benzimidazoles; Hydrogenated benzimidazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
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- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
- A61K31/4015—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil having oxo groups directly attached to the heterocyclic ring, e.g. piracetam, ethosuximide
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- A61K31/4025—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil not condensed and containing further heterocyclic rings, e.g. cromakalim
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- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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- C07C2601/08—Systems containing only non-condensed rings with a five-membered ring the ring being saturated
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- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2601/00—Systems containing only non-condensed rings
- C07C2601/06—Systems containing only non-condensed rings with a five-membered ring
- C07C2601/10—Systems containing only non-condensed rings with a five-membered ring the ring being unsaturated
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| US61810204P | 2004-10-12 | 2004-10-12 | |
| IN1096MU2004 | 2004-10-14 | ||
| US63526604P | 2004-12-10 | 2004-12-10 | |
| IN1332MU2004 | 2004-12-14 |
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| MY142423A true MY142423A (en) | 2010-11-30 |
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| MYPI20054654A MY142423A (en) | 2004-10-12 | 2005-10-03 | Substituted aminoacetyl pyrrolidine compounds which are dipeptidyl peptidase iv inhibitors, and pharmaceutical compositions containing them |
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| US (3) | US7205323B2 (https=) |
| EP (1) | EP1799639B1 (https=) |
| JP (1) | JP4959569B2 (https=) |
| KR (1) | KR20070073887A (https=) |
| AP (1) | AP2007003973A0 (https=) |
| AR (1) | AR053415A1 (https=) |
| AU (1) | AU2005293266B2 (https=) |
| BR (1) | BRPI0516340A (https=) |
| CA (1) | CA2583457C (https=) |
| EA (1) | EA013463B1 (https=) |
| IL (1) | IL182444A0 (https=) |
| MX (1) | MX2007004305A (https=) |
| MY (1) | MY142423A (https=) |
| NZ (1) | NZ554515A (https=) |
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| ATE368647T1 (de) | 2002-09-19 | 2007-08-15 | Abbott Lab | Pharmazeutische zusammensetzung und ihre verwendung als inhibitoren von der dipeptidyl peptidase iv (dpp-iv) |
| JP2006522109A (ja) * | 2003-03-31 | 2006-09-28 | 大正製薬株式会社 | 新規なキナゾリン誘導体及びそれらの使用に関連する治療方法 |
| US20050197350A1 (en) | 2003-03-31 | 2005-09-08 | Taisho Pharmaceutical Co., Ltd. | Novel quinoline, tetrahydroquinazoline, and pyrimidine derivatives and methods of treatment related to the use thereof |
| EP1627870A1 (en) | 2003-05-15 | 2006-02-22 | Taisho Pharmaceutical Co., Ltd | Cyanofluoropyrrolidine derivative |
| WO2005023762A1 (en) | 2003-09-04 | 2005-03-17 | Abbott Laboratories | Pyrrolidine-2-carbonitrile derivatives and their use as inhibitors of dipeptidyl peptidase-iv (dpp-iv) |
| US7230002B2 (en) * | 2004-02-03 | 2007-06-12 | Glenmark Pharmaceuticals Ltd. | Dipeptidyl peptidase IV inhibitors; processes for their preparation and compositions thereof |
| WO2005075426A1 (en) * | 2004-02-03 | 2005-08-18 | Glenmark Pharmaceuticals Ltd. | Novel dipeptidyl peptidase iv inhibitors; processes for their preparation and compositions thereof |
-
2005
- 2005-07-26 BR BRPI0516340-4A patent/BRPI0516340A/pt not_active IP Right Cessation
- 2005-07-26 CA CA2583457A patent/CA2583457C/en not_active Expired - Fee Related
- 2005-07-26 NZ NZ554515A patent/NZ554515A/en not_active IP Right Cessation
- 2005-07-26 JP JP2007536276A patent/JP4959569B2/ja not_active Expired - Fee Related
- 2005-07-26 KR KR1020077010262A patent/KR20070073887A/ko not_active Ceased
- 2005-07-26 AU AU2005293266A patent/AU2005293266B2/en not_active Ceased
- 2005-07-26 EP EP05784869.9A patent/EP1799639B1/en not_active Expired - Lifetime
- 2005-07-26 EA EA200700720A patent/EA013463B1/ru not_active IP Right Cessation
- 2005-07-26 WO PCT/IB2005/002204 patent/WO2006040625A1/en not_active Ceased
- 2005-07-26 AP AP2007003973A patent/AP2007003973A0/xx unknown
- 2005-07-26 MX MX2007004305A patent/MX2007004305A/es active IP Right Grant
- 2005-09-29 TW TW094134070A patent/TW200614988A/zh unknown
- 2005-10-03 MY MYPI20054654A patent/MY142423A/en unknown
- 2005-10-12 AR ARP050104282A patent/AR053415A1/es unknown
- 2005-10-12 US US11/250,195 patent/US7205323B2/en not_active Expired - Lifetime
-
2007
- 2007-02-15 US US11/675,180 patent/US7538128B2/en not_active Expired - Lifetime
- 2007-02-15 US US11/675,157 patent/US7524844B2/en not_active Expired - Lifetime
- 2007-04-10 IL IL182444A patent/IL182444A0/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| BRPI0516340A (pt) | 2008-09-16 |
| EP1799639A1 (en) | 2007-06-27 |
| JP4959569B2 (ja) | 2012-06-27 |
| EA013463B1 (ru) | 2010-04-30 |
| EA200700720A1 (ru) | 2007-08-31 |
| IL182444A0 (en) | 2007-07-24 |
| WO2006040625A1 (en) | 2006-04-20 |
| MX2007004305A (es) | 2007-06-18 |
| AP2007003973A0 (en) | 2007-07-30 |
| US7205323B2 (en) | 2007-04-17 |
| AU2005293266B2 (en) | 2011-09-29 |
| US7538128B2 (en) | 2009-05-26 |
| US20060142585A1 (en) | 2006-06-29 |
| KR20070073887A (ko) | 2007-07-10 |
| AR053415A1 (es) | 2007-05-09 |
| EP1799639B1 (en) | 2013-09-04 |
| US20070238728A1 (en) | 2007-10-11 |
| JP2008515962A (ja) | 2008-05-15 |
| CA2583457C (en) | 2013-01-29 |
| US20070232608A1 (en) | 2007-10-04 |
| NZ554515A (en) | 2009-12-24 |
| CA2583457A1 (en) | 2006-04-20 |
| US7524844B2 (en) | 2009-04-28 |
| AU2005293266A1 (en) | 2006-04-20 |
| TW200614988A (en) | 2006-05-16 |
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