MXPA06011328A - Azaindoles utiles como inhibidotes de roca y otras proteinas cinasas. - Google Patents

Azaindoles utiles como inhibidotes de roca y otras proteinas cinasas.

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Publication number
MXPA06011328A
MXPA06011328A MXPA06011328A MXPA06011328A MXPA06011328A MX PA06011328 A MXPA06011328 A MX PA06011328A MX PA06011328 A MXPA06011328 A MX PA06011328A MX PA06011328 A MXPA06011328 A MX PA06011328A MX PA06011328 A MXPA06011328 A MX PA06011328A
Authority
MX
Mexico
Prior art keywords
ppm
disease
compound according
chr6
agent
Prior art date
Application number
MXPA06011328A
Other languages
English (en)
Spanish (es)
Inventor
John J Court
Jeremy Green
Andrew Miller
Juan-Miguel Jimenez
Craig Marhefka
Jingrong Cao
Upul K Bandarage
Huai Gao
Suganthini Nanthakumar
Original Assignee
Vertex Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Vertex Pharma filed Critical Vertex Pharma
Publication of MXPA06011328A publication Critical patent/MXPA06011328A/es

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
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    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
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  • Heart & Thoracic Surgery (AREA)
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  • Ophthalmology & Optometry (AREA)
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MXPA06011328A 2004-04-02 2005-04-04 Azaindoles utiles como inhibidotes de roca y otras proteinas cinasas. MXPA06011328A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US55904104P 2004-04-02 2004-04-02
PCT/US2005/011358 WO2005103050A2 (en) 2004-04-02 2005-04-04 Azaindoles useful as inhibitors of rock and other protein kinases

Publications (1)

Publication Number Publication Date
MXPA06011328A true MXPA06011328A (es) 2006-12-15

Family

ID=34983212

Family Applications (1)

Application Number Title Priority Date Filing Date
MXPA06011328A MXPA06011328A (es) 2004-04-02 2005-04-04 Azaindoles utiles como inhibidotes de roca y otras proteinas cinasas.

Country Status (14)

Country Link
US (1) US7514448B2 (enExample)
EP (1) EP1756108A2 (enExample)
JP (1) JP5019612B2 (enExample)
KR (1) KR20070002081A (enExample)
CN (1) CN101014597A (enExample)
AR (1) AR049333A1 (enExample)
AU (1) AU2005236002A1 (enExample)
CA (1) CA2561724A1 (enExample)
IL (1) IL178414A0 (enExample)
MX (1) MXPA06011328A (enExample)
NO (1) NO20064976L (enExample)
RU (1) RU2006138621A (enExample)
TW (1) TW200604168A (enExample)
WO (1) WO2005103050A2 (enExample)

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WO2005066145A1 (en) 2004-01-06 2005-07-21 Novo Nordisk A/S Heteroaryl-ureas and their use as glucokinase activators
EP1708697A4 (en) * 2004-01-30 2007-11-28 Smithkline Beecham Corp CHEMICAL COMPOUNDS
EP2332940B1 (en) 2004-03-30 2012-10-31 Vertex Pharmaceuticals Incorporated Azaindoles useful as inhibitors of JAK and other protein kinases
US7498342B2 (en) 2004-06-17 2009-03-03 Plexxikon, Inc. Compounds modulating c-kit activity
MXPA06014415A (es) 2004-06-24 2007-02-19 Shionogi & Co Compuestos de sulfonamida.
WO2006004984A1 (en) * 2004-06-30 2006-01-12 Vertex Pharmaceuticals Incorporated Azaindoles useful as inhibitors of protein kinases
MX2007000092A (es) * 2004-06-30 2007-03-07 Vertex Pharma Azaindoles utiles como inhibidores de proteinas cinasas.
AU2005272815A1 (en) * 2004-08-13 2006-02-23 Genentech, Inc. Thiazole based inhibitors of ATP-utilizing enzymes
CN101098872B (zh) * 2004-11-22 2012-09-05 沃泰克斯药物股份有限公司 可用作蛋白激酶抑制剂的吡咯并吡嗪和吡唑并吡嗪
EP1864971A4 (en) * 2005-03-31 2010-02-10 Takeda Pharmaceutical PROPHYLACTIC / THERAPEUTIC AGENT AGAINST DIABETES
NZ564065A (en) * 2005-05-20 2011-03-31 Vertex Pharma Pyrrolopyridines useful as inhibitors of protein kinase
BRPI0613591A2 (pt) 2005-07-08 2011-01-18 Novo Nordisk As ativadores de dicicloalquil uréia glicocinase
EP2377856A1 (en) 2005-07-14 2011-10-19 Novo Nordisk A/S Urea glucokinase activators
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