MX389920B - Procesos novedosos para preparar estimuladores de guanilato ciclasa soluble. - Google Patents

Procesos novedosos para preparar estimuladores de guanilato ciclasa soluble.

Info

Publication number
MX389920B
MX389920B MX2019000105A MX2019000105A MX389920B MX 389920 B MX389920 B MX 389920B MX 2019000105 A MX2019000105 A MX 2019000105A MX 2019000105 A MX2019000105 A MX 2019000105A MX 389920 B MX389920 B MX 389920B
Authority
MX
Mexico
Prior art keywords
guanylate cyclase
soluble guanylate
preparation
novel processes
preparing soluble
Prior art date
Application number
MX2019000105A
Other languages
English (en)
Spanish (es)
Other versions
MX2019000105A (es
Inventor
Robert C Livingston
Song Xue
Vishnu Vardhan Reddy Karnati
Original Assignee
Cyclerion Therapeutics Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Cyclerion Therapeutics Inc filed Critical Cyclerion Therapeutics Inc
Publication of MX2019000105A publication Critical patent/MX2019000105A/es
Publication of MX389920B publication Critical patent/MX389920B/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Enzymes And Modification Thereof (AREA)
MX2019000105A 2016-07-07 2017-07-06 Procesos novedosos para preparar estimuladores de guanilato ciclasa soluble. MX389920B (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201662359453P 2016-07-07 2016-07-07
PCT/US2017/040810 WO2018009597A1 (en) 2016-07-07 2017-07-06 Novel processes for preparation of soluble guanylate cyclase stimulators

Publications (2)

Publication Number Publication Date
MX2019000105A MX2019000105A (es) 2019-04-22
MX389920B true MX389920B (es) 2025-03-20

Family

ID=59416789

Family Applications (2)

Application Number Title Priority Date Filing Date
MX2019000105A MX389920B (es) 2016-07-07 2017-07-06 Procesos novedosos para preparar estimuladores de guanilato ciclasa soluble.
MX2022001495A MX2022001495A (es) 2016-07-07 2019-01-07 Procesos novedosos para preparar estimuladores de guanilato ciclasa soluble.

Family Applications After (1)

Application Number Title Priority Date Filing Date
MX2022001495A MX2022001495A (es) 2016-07-07 2019-01-07 Procesos novedosos para preparar estimuladores de guanilato ciclasa soluble.

Country Status (16)

Country Link
US (3) US11319308B2 (enExample)
EP (2) EP3481818B1 (enExample)
JP (1) JP7112384B2 (enExample)
KR (1) KR102487872B1 (enExample)
CN (1) CN109563077A (enExample)
AU (1) AU2017291827B2 (enExample)
BR (1) BR112019000291A2 (enExample)
CA (1) CA3029375A1 (enExample)
CL (2) CL2019000016A1 (enExample)
EA (1) EA201990237A1 (enExample)
ES (1) ES2963563T3 (enExample)
IL (1) IL263995B (enExample)
MA (1) MA45603A (enExample)
MX (2) MX389920B (enExample)
SG (1) SG11201900096QA (enExample)
WO (1) WO2018009597A1 (enExample)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MX382762B (es) 2016-07-07 2025-03-13 Cyclerion Therapeutics Inc Procesos novedosos para preparacion de estimuladores de guanilato ciclasa soluble.
AU2017291827B2 (en) 2016-07-07 2021-10-21 Cyclerion Therapeutics, Inc. Novel processes for preparation of soluble guanylate cyclase stimulators
EP4570797A3 (en) 2018-01-10 2025-09-03 Cyclerion Therapeutics, Inc. Novel processes and intermediates for the preparation of soluble guanylate cyclase stimulators
WO2019161534A1 (en) * 2018-02-22 2019-08-29 Ironwood Pharmaceuticals, Inc. Novel processes and intermediates for preparation of soluble guanylate cyclase stimulators

Family Cites Families (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2011150156A2 (en) * 2010-05-26 2011-12-01 Sunovion Pharmaceuticals Inc. Heteroaryl compounds and methods of use thereof
JP5860459B2 (ja) 2010-06-30 2016-02-16 アイアンウッド ファーマシューティカルズ インコーポレイテッド sGC刺激薬
US9139564B2 (en) * 2011-12-27 2015-09-22 Ironwood Pharmaceuticals, Inc. 2-benzyl, 3-(pyrimidin-2-yl) substituted pyrazoles useful as sGC stimulators
EP2897953B8 (en) * 2012-09-19 2019-06-26 Cyclerion Therapeutics, Inc. Sgc stimulators
RS59981B1 (sr) * 2013-03-15 2020-03-31 Cyclerion Therapeutics Inc Sgc stimulatori
US20160311826A1 (en) * 2013-12-11 2016-10-27 Ironwood Pharmaceuticals, Inc. Sgc stimulators
US20170298055A1 (en) * 2014-09-17 2017-10-19 Ironwood Pharmaceuticals, Inc. sGC STIMULATORS
AU2015317824A1 (en) * 2014-09-17 2017-03-23 Cyclerion Therapeutics, Inc. Pyrazole derivatives as sGC stimulators
KR20170055531A (ko) * 2014-09-17 2017-05-19 아이언우드 파마슈티컬스, 인코포레이티드 에스지씨 자극제
US10844064B2 (en) * 2014-09-17 2020-11-24 Cyclerion Therapeutics, Inc. sGC stimulators
EP3383372B1 (en) * 2015-11-30 2023-11-01 Cyclerion Therapeutics, Inc. Solid dispersions comprising a sgc stimulator
MX382762B (es) 2016-07-07 2025-03-13 Cyclerion Therapeutics Inc Procesos novedosos para preparacion de estimuladores de guanilato ciclasa soluble.
JP2019524710A (ja) * 2016-07-07 2019-09-05 アイアンウッド ファーマシューティカルズ インコーポレイテッド Sgc刺激剤の固体形態
AU2017291827B2 (en) 2016-07-07 2021-10-21 Cyclerion Therapeutics, Inc. Novel processes for preparation of soluble guanylate cyclase stimulators
EA202091502A1 (ru) * 2017-12-19 2020-11-12 Сайклерион Терапьютикс, Инк. СТИМУЛЯТОРЫ sGC
EP4570797A3 (en) * 2018-01-10 2025-09-03 Cyclerion Therapeutics, Inc. Novel processes and intermediates for the preparation of soluble guanylate cyclase stimulators

Also Published As

Publication number Publication date
AU2017291827A1 (en) 2019-02-07
SG11201900096QA (en) 2019-02-27
IL263995A (en) 2019-02-28
KR20190025986A (ko) 2019-03-12
CL2019000016A1 (es) 2019-05-03
BR112019000291A2 (pt) 2019-04-16
WO2018009597A1 (en) 2018-01-11
CA3029375A1 (en) 2018-01-11
MA45603A (fr) 2019-05-15
CL2023000228A1 (es) 2023-09-29
US11773089B2 (en) 2023-10-03
US20240059684A1 (en) 2024-02-22
MX2022001495A (es) 2022-03-11
AU2017291827B2 (en) 2021-10-21
CN109563077A (zh) 2019-04-02
JP7112384B2 (ja) 2022-08-03
EP4249488A3 (en) 2023-12-20
EP3481818C0 (en) 2023-09-06
EP4249488A2 (en) 2023-09-27
US20220227748A1 (en) 2022-07-21
US11319308B2 (en) 2022-05-03
EA201990237A1 (ru) 2019-08-30
EP3481818B1 (en) 2023-09-06
IL263995B (en) 2021-02-28
EP3481818A1 (en) 2019-05-15
US20210323951A1 (en) 2021-10-21
ES2963563T3 (es) 2024-03-27
NZ750123A (en) 2025-02-28
MX2019000105A (es) 2019-04-22
JP2019525913A (ja) 2019-09-12
KR102487872B1 (ko) 2023-01-12

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