MX2010013208A - Derivados de n-piperidinil acetamida como bloqueadores de canal de calcio. - Google Patents

Derivados de n-piperidinil acetamida como bloqueadores de canal de calcio.

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Publication number
MX2010013208A
MX2010013208A MX2010013208A MX2010013208A MX2010013208A MX 2010013208 A MX2010013208 A MX 2010013208A MX 2010013208 A MX2010013208 A MX 2010013208A MX 2010013208 A MX2010013208 A MX 2010013208A MX 2010013208 A MX2010013208 A MX 2010013208A
Authority
MX
Mexico
Prior art keywords
methyl
optionally substituted
compound
piperidin
alkyl
Prior art date
Application number
MX2010013208A
Other languages
English (en)
Spanish (es)
Inventor
Yongbao Zhu
Hassan Pajouhesh
Ramesh Kaul
Yanbing Ding
Lingyun Zhang
Nagasree Chakka
Mike Grimwood
Jason Tan
Yuanxi Zhou
Original Assignee
Zalicus Pharmaceuticals Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Zalicus Pharmaceuticals Ltd filed Critical Zalicus Pharmaceuticals Ltd
Publication of MX2010013208A publication Critical patent/MX2010013208A/es

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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/5375—1,4-Oxazines, e.g. morpholine
    • A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
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    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
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