HK1175997A1 - 作為鈣通道阻斷劑的 -哌啶基乙酰胺衍生物 - Google Patents

作為鈣通道阻斷劑的 -哌啶基乙酰胺衍生物

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Publication number
HK1175997A1
HK1175997A1 HK13103155.0A HK13103155A HK1175997A1 HK 1175997 A1 HK1175997 A1 HK 1175997A1 HK 13103155 A HK13103155 A HK 13103155A HK 1175997 A1 HK1175997 A1 HK 1175997A1
Authority
HK
Hong Kong
Prior art keywords
calcium channel
channel blockers
acetamide derivatives
piperidinyl acetamide
piperidinyl
Prior art date
Application number
HK13103155.0A
Other languages
English (en)
Inventor
Hassan Pajouhesh
Ramesh Kaul
Yanbing Ding
Yongbao Zhu
Lingyun Zhang
Nagasree Chakka
Mike Grimwood
Jason Tan
Yuanxi Zhou
Original Assignee
Taro Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Taro Pharmaceuticals Inc filed Critical Taro Pharmaceuticals Inc
Publication of HK1175997A1 publication Critical patent/HK1175997A1/zh

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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/5375—1,4-Oxazines, e.g. morpholine
    • A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
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    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
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