MX2009006001A - Derivados de 2,3-dihidroimidazo[1,2-c]quinazolina sustituidos de utilidad en el tratamiento de trastornos hiperproliferativos y enfermedades asociadas con la angiogenesis. - Google Patents

Derivados de 2,3-dihidroimidazo[1,2-c]quinazolina sustituidos de utilidad en el tratamiento de trastornos hiperproliferativos y enfermedades asociadas con la angiogenesis.

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Publication number
MX2009006001A
MX2009006001A MX2009006001A MX2009006001A MX2009006001A MX 2009006001 A MX2009006001 A MX 2009006001A MX 2009006001 A MX2009006001 A MX 2009006001A MX 2009006001 A MX2009006001 A MX 2009006001A MX 2009006001 A MX2009006001 A MX 2009006001A
Authority
MX
Mexico
Prior art keywords
dihydroimidazo
diseases associated
angiogenesis
substituted
proliferative disorders
Prior art date
Application number
MX2009006001A
Other languages
English (en)
Spanish (es)
Inventor
Martin Michels
Martin Hentemann
Jill Wood
William Scott
Ann-Marie Campbell
Ann-Marie Bullion
R Bruce Rowley
Aniko Redman
Original Assignee
Bayer Schering Pharma Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=39492563&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MX2009006001(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Bayer Schering Pharma Ag filed Critical Bayer Schering Pharma Ag
Publication of MX2009006001A publication Critical patent/MX2009006001A/es

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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/5375—1,4-Oxazines, e.g. morpholine
    • A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
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    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
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    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/517—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with carbocyclic ring systems, e.g. quinazoline, perimidine
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

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MX2009006001A 2006-12-05 2007-12-05 Derivados de 2,3-dihidroimidazo[1,2-c]quinazolina sustituidos de utilidad en el tratamiento de trastornos hiperproliferativos y enfermedades asociadas con la angiogenesis. MX2009006001A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US87309006P 2006-12-05 2006-12-05
PCT/US2007/024985 WO2008070150A1 (en) 2006-12-05 2007-12-05 Substituted 2,3-dihydroimidazo[1,2-c]quinazoline derivatives useful for treating hyper-proliferative disorders and diseases associated with angiogenesis

Publications (1)

Publication Number Publication Date
MX2009006001A true MX2009006001A (es) 2009-06-16

Family

ID=39492563

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2009006001A MX2009006001A (es) 2006-12-05 2007-12-05 Derivados de 2,3-dihidroimidazo[1,2-c]quinazolina sustituidos de utilidad en el tratamiento de trastornos hiperproliferativos y enfermedades asociadas con la angiogenesis.

Country Status (42)

Country Link
US (3) US8466283B2 (und)
EP (1) EP2096919B1 (und)
JP (1) JP5326092B2 (und)
KR (1) KR101501785B1 (und)
CN (4) CN105254634B (und)
AR (1) AR064106A1 (und)
AU (1) AU2007328008B2 (und)
BR (1) BRPI0720178B8 (und)
CA (1) CA2671614C (und)
CL (1) CL2007003508A1 (und)
CO (1) CO6220908A2 (und)
CR (1) CR10838A (und)
CU (1) CU23796B7 (und)
DK (1) DK2096919T3 (und)
DO (1) DOP2009000135A (und)
EA (1) EA018839B1 (und)
EC (1) ECSP099387A (und)
ES (1) ES2572189T3 (und)
GT (1) GT200900154A (und)
HK (1) HK1217953A1 (und)
HN (1) HN2009001131A (und)
HU (1) HUE028773T2 (und)
IL (1) IL198273A (und)
JO (1) JO3147B1 (und)
MA (1) MA31283B1 (und)
MX (1) MX2009006001A (und)
MY (1) MY157944A (und)
NO (1) NO342348B1 (und)
NZ (1) NZ577342A (und)
PA (1) PA8759601A1 (und)
PE (1) PE20081444A1 (und)
PL (1) PL2096919T3 (und)
RS (1) RS56045B1 (und)
SG (1) SG177170A1 (und)
SI (1) SI2096919T1 (und)
SV (1) SV2009003288A (und)
TN (1) TN2009000137A1 (und)
TW (1) TWI406662B (und)
UA (1) UA96965C2 (und)
UY (1) UY30761A1 (und)
WO (1) WO2008070150A1 (und)
ZA (1) ZA200904691B (und)

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